CN108503582A - 2-(1h)-喹啉酮类化合物的微波辅助合成方法 - Google Patents
2-(1h)-喹啉酮类化合物的微波辅助合成方法 Download PDFInfo
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- CN108503582A CN108503582A CN201810056840.8A CN201810056840A CN108503582A CN 108503582 A CN108503582 A CN 108503582A CN 201810056840 A CN201810056840 A CN 201810056840A CN 108503582 A CN108503582 A CN 108503582A
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- Prior art keywords
- quinoline
- reaction
- microwave
- synthesizing method
- raw material
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C07D215/22—Oxygen atoms attached in position 2 or 4
- C07D215/227—Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
Description
Claims (10)
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
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CN201810056840.8A CN108503582B (zh) | 2018-01-19 | 2018-01-19 | 2-(1h)-喹啉酮类化合物的微波辅助合成方法 |
Applications Claiming Priority (1)
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CN201810056840.8A CN108503582B (zh) | 2018-01-19 | 2018-01-19 | 2-(1h)-喹啉酮类化合物的微波辅助合成方法 |
Publications (2)
Publication Number | Publication Date |
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CN108503582A true CN108503582A (zh) | 2018-09-07 |
CN108503582B CN108503582B (zh) | 2020-01-07 |
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CN201810056840.8A Expired - Fee Related CN108503582B (zh) | 2018-01-19 | 2018-01-19 | 2-(1h)-喹啉酮类化合物的微波辅助合成方法 |
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CN (1) | CN108503582B (zh) |
Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN106588765A (zh) * | 2016-09-06 | 2017-04-26 | 天津科技大学 | 一种氮氧化物c2‑位羟基化的方法 |
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2018
- 2018-01-19 CN CN201810056840.8A patent/CN108503582B/zh not_active Expired - Fee Related
Patent Citations (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN106588765A (zh) * | 2016-09-06 | 2017-04-26 | 天津科技大学 | 一种氮氧化物c2‑位羟基化的方法 |
Non-Patent Citations (3)
Title |
---|
P. TOMASIK,等: "A NOVEL NUCLEOPHILIC SUBSTITUTION OF THE PYRIDINE RING", 《TETRAHEDRON LETTERS》 * |
PATRICK S. FIER,等: "Synthesis and Late-Stage Functionalization of Complex Molecules through C−H Fluorination and Nucleophilic Aromatic Substitution", 《J. AM. CHEM. SOC.》 * |
PATRICK S. FIER: "A Bifunctional Reagent Designed for the Mild, Nucleophilic Functionalization of Pyridines", 《J. AM. CHEM. SOC.》 * |
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Publication number | Publication date |
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CN108503582B (zh) | 2020-01-07 |
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Inventor after: Wang Yi Inventor after: Cao Zhong Inventor after: Lu Linghui Inventor after: Peng Sha Inventor after: He Weibao Inventor after: Zeng Fei Inventor after: Bao Wenhu Inventor after: He Weimin Inventor before: He Weimin Inventor before: Cao Zhong Inventor before: Lu Linghui Inventor before: Peng Sha Inventor before: He Weibao Inventor before: Zeng Fei Inventor before: Bao Wenhu Inventor before: Wang Yi |
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CF01 | Termination of patent right due to non-payment of annual fee |
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CF01 | Termination of patent right due to non-payment of annual fee |