CN108349946B - 作为PI3Kβ抑制剂的喹喔啉和吡啶并吡嗪衍生物 - Google Patents

作为PI3Kβ抑制剂的喹喔啉和吡啶并吡嗪衍生物 Download PDF

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CN108349946B
CN108349946B CN201680058332.2A CN201680058332A CN108349946B CN 108349946 B CN108349946 B CN 108349946B CN 201680058332 A CN201680058332 A CN 201680058332A CN 108349946 B CN108349946 B CN 108349946B
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CN108349946A (zh
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P.R.安吉鲍德
O.A.G.奎尔罗勒
D.J-C.保特洛特
C.梅耶
M.P.V.维罗特
L.米尔波伊
T.F.A.J.乔斯塞奥梅
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Janssen Pharmaceutica NV
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CN201680058332.2A 2015-10-09 2016-10-07 作为PI3Kβ抑制剂的喹喔啉和吡啶并吡嗪衍生物 Active CN108349946B (zh)

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Application Number Priority Date Filing Date Title
EP15189163 2015-10-09
EP15189163.7 2015-10-09
EP16174710.0 2016-06-16
EP16174710 2016-06-16
PCT/EP2016/073962 WO2017060406A1 (en) 2015-10-09 2016-10-07 Quinoxaline and pyridopyrazine derivatives as pi3kbeta inhibitors

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CN108349946A CN108349946A (zh) 2018-07-31
CN108349946B true CN108349946B (zh) 2021-05-18

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US10526316B2 (en) 2020-01-07
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BR112018007068A2 (pt) 2018-10-23
BR112018007068B1 (pt) 2024-01-02
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