AU2016335086B2 - Quinoxaline and pyridopyrazine derivatives as pI3Kbeta inhibitors - Google Patents

Quinoxaline and pyridopyrazine derivatives as pI3Kbeta inhibitors Download PDF

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AU2016335086B2
AU2016335086B2 AU2016335086A AU2016335086A AU2016335086B2 AU 2016335086 B2 AU2016335086 B2 AU 2016335086B2 AU 2016335086 A AU2016335086 A AU 2016335086A AU 2016335086 A AU2016335086 A AU 2016335086A AU 2016335086 B2 AU2016335086 B2 AU 2016335086B2
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4alkyl
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AU2016335086A1 (en
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Patrick Rene Angibaud
Didier Jean-Claude Berthelot
Thierry François Alain Jean Jousseaume
Lieven Meerpoel
Christophe Meyer
Olivier Alexis Georges Querolle
Matthieu Philippe Victor Willot
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Janssen Pharmaceutica NV
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AU2016335086A 2015-10-09 2016-10-07 Quinoxaline and pyridopyrazine derivatives as pI3Kbeta inhibitors Active AU2016335086B2 (en)

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EP15189163 2015-10-09
EP15189163.7 2015-10-09
EP16174710.0 2016-06-16
EP16174710 2016-06-16
PCT/EP2016/073962 WO2017060406A1 (en) 2015-10-09 2016-10-07 Quinoxaline and pyridopyrazine derivatives as pi3kbeta inhibitors

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AU2016335086A1 AU2016335086A1 (en) 2018-04-12
AU2016335086B2 true AU2016335086B2 (en) 2020-08-27

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EP (1) EP3359533B1 (enExample)
JP (1) JP6912460B2 (enExample)
KR (1) KR102630111B1 (enExample)
CN (1) CN108349946B (enExample)
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BR (1) BR112018007068B1 (enExample)
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EA (1) EA037401B1 (enExample)
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Families Citing this family (8)

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Publication number Priority date Publication date Assignee Title
AU2016335086B2 (en) * 2015-10-09 2020-08-27 Janssen Pharmaceutica Nv Quinoxaline and pyridopyrazine derivatives as pI3Kbeta inhibitors
LT3472160T (lt) 2016-06-16 2021-04-26 Janssen Pharmaceutica Nv Biciklinio piridino, pirazino ir pirimidino dariniai kaip pi3k beta inhibitoriai
CN110461827A (zh) 2017-03-29 2019-11-15 詹森药业有限公司 作为PI3K-β抑制剂的喹喔啉和吡啶并吡嗪衍生物
MD3762368T2 (ro) 2018-03-08 2022-07-31 Incyte Corp Compuși diol aminopirazină ca inhibitori ai PI3K-Y
WO2020010003A1 (en) 2018-07-02 2020-01-09 Incyte Corporation AMINOPYRAZINE DERIVATIVES AS PI3K-γ INHIBITORS
CN111892597B (zh) * 2020-09-01 2023-07-25 山西天宏达安医药科技有限公司 一种喹喔啉基吡啶并吡嗪类化合物及其制备方法与应用
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