CN107073011A - 利用噻吩并三唑并二氮杂*化合物治疗淋巴瘤的方法 - Google Patents

利用噻吩并三唑并二氮杂*化合物治疗淋巴瘤的方法 Download PDF

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Publication number
CN107073011A
CN107073011A CN201580045068.4A CN201580045068A CN107073011A CN 107073011 A CN107073011 A CN 107073011A CN 201580045068 A CN201580045068 A CN 201580045068A CN 107073011 A CN107073011 A CN 107073011A
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compound
thienotriazolodiazepine
dlbcl
carbons
group
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CN201580045068.4A
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Chinese (zh)
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弗朗切斯科·贝尔托尼
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Oncoethix GmbH
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Oncoethix GmbH
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
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    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
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CN201580045068.4A 2014-08-19 2015-08-19 利用噻吩并三唑并二氮杂*化合物治疗淋巴瘤的方法 Pending CN107073011A (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US201462039072P 2014-08-19 2014-08-19
US62/039,072 2014-08-19
US201462086609P 2014-12-02 2014-12-02
US62/086,609 2014-12-02
PCT/EP2015/069092 WO2016026912A1 (en) 2014-08-19 2015-08-19 Methods of treating lymphoma using thienotriazolodiazepine compounds

Publications (1)

Publication Number Publication Date
CN107073011A true CN107073011A (zh) 2017-08-18

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CN201580045068.4A Pending CN107073011A (zh) 2014-08-19 2015-08-19 利用噻吩并三唑并二氮杂*化合物治疗淋巴瘤的方法

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US (1) US9968620B2 (enExample)
EP (1) EP3182976A1 (enExample)
JP (1) JP2017528446A (enExample)
KR (1) KR20170037670A (enExample)
CN (1) CN107073011A (enExample)
WO (1) WO2016026912A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN108057036B (zh) * 2016-11-07 2023-06-13 正大天晴药业集团股份有限公司 一种egfr抑制剂的固体药物组合物
US12162870B2 (en) 2021-06-08 2024-12-10 The Regents Of The University Of California Anticancer compounds
WO2025120552A1 (ko) * 2023-12-07 2025-06-12 제이더블유중외제약 주식회사 헤테로사이클 유도체 함유 고체분산체, 이의 제조 방법, 이를 포함하는 약학적 조성물

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1297836A1 (en) * 2000-06-16 2003-04-02 Mitsubishi Pharma Corporation COMPOSITIONS CONTROLLING RELEASE pH RANGE AND/OR SPEED
CN101910182A (zh) * 2007-12-28 2010-12-08 田边三菱制药株式会社 抗癌剂
WO2014001356A1 (en) * 2012-06-25 2014-01-03 Oncoethix Sa Method of treating lymphoma using thienotriazolodiazepine compounds
WO2015018520A1 (en) * 2013-08-06 2015-02-12 Oncoethix Sa A bet-brd inhibitor represents a novel agent for alk positive anaplastic large cell lymphoma
CN105899212A (zh) * 2013-08-06 2016-08-24 翁科埃斯克斯有限公司 利用β溴结构域抑制剂治疗弥漫性大B细胞淋巴瘤(DLBCL)的方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2015115634A (ru) * 2012-09-28 2016-11-20 Онкоэтикс Гмбх Фармацевтический состав, содержащий соединения тиенотриазолодиазепина
EP3137086A4 (en) * 2014-05-02 2017-12-27 Oncoethix GmbH Method of treating resistant non-hodgkin lymphoma, medulloblastoma, and/or alk+non-small cell lung cancer using thienotriazolodiazepine compounds

Patent Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1297836A1 (en) * 2000-06-16 2003-04-02 Mitsubishi Pharma Corporation COMPOSITIONS CONTROLLING RELEASE pH RANGE AND/OR SPEED
CN101910182A (zh) * 2007-12-28 2010-12-08 田边三菱制药株式会社 抗癌剂
WO2014001356A1 (en) * 2012-06-25 2014-01-03 Oncoethix Sa Method of treating lymphoma using thienotriazolodiazepine compounds
CN105050605A (zh) * 2012-06-25 2015-11-11 翁科埃蒂克斯股份公司 使用噻吩并三唑并二氮杂*化合物治疗淋巴瘤的方法
WO2015018520A1 (en) * 2013-08-06 2015-02-12 Oncoethix Sa A bet-brd inhibitor represents a novel agent for alk positive anaplastic large cell lymphoma
CN105899212A (zh) * 2013-08-06 2016-08-24 翁科埃斯克斯有限公司 利用β溴结构域抑制剂治疗弥漫性大B细胞淋巴瘤(DLBCL)的方法

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Publication number Publication date
US9968620B2 (en) 2018-05-15
US20170273988A1 (en) 2017-09-28
EP3182976A1 (en) 2017-06-28
WO2016026912A1 (en) 2016-02-25
JP2017528446A (ja) 2017-09-28
KR20170037670A (ko) 2017-04-04

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Application publication date: 20170818