CN106459120A - 作为asgpr靶向剂的被取代的‑6,8‑二氧杂双环[3.2.1]辛烷‑2,3‑二醇化合物 - Google Patents

作为asgpr靶向剂的被取代的‑6,8‑二氧杂双环[3.2.1]辛烷‑2,3‑二醇化合物 Download PDF

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Publication number
CN106459120A
CN106459120A CN201580028359.2A CN201580028359A CN106459120A CN 106459120 A CN106459120 A CN 106459120A CN 201580028359 A CN201580028359 A CN 201580028359A CN 106459120 A CN106459120 A CN 106459120A
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base
dihydroxy
octyl
bicyclic
oxa
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CN201580028359.2A
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Chinese (zh)
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V·马希蒂
B·丘马
S·利拉斯
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SmithKline Beecham Ltd
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SmithKline Beecham Ltd
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    • A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
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CN201580028359.2A 2014-05-19 2015-05-05 作为asgpr靶向剂的被取代的‑6,8‑二氧杂双环[3.2.1]辛烷‑2,3‑二醇化合物 Pending CN106459120A (zh)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201462000211P 2014-05-19 2014-05-19
US62/000,211 2014-05-19
US201462001540P 2014-05-21 2014-05-21
US62/001,540 2014-05-21
US201562139254P 2015-03-27 2015-03-27
US62/139,254 2015-03-27
PCT/IB2015/053282 WO2015177668A1 (en) 2014-05-19 2015-05-05 Substituted-6,8-dioxabicyclo[3.2.1]octane-2,3-diol compounds as targeting agents of asgpr

Publications (1)

Publication Number Publication Date
CN106459120A true CN106459120A (zh) 2017-02-22

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CN201580028359.2A Pending CN106459120A (zh) 2014-05-19 2015-05-05 作为asgpr靶向剂的被取代的‑6,8‑二氧杂双环[3.2.1]辛烷‑2,3‑二醇化合物

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EP (1) EP3145934B1 (https=)
JP (2) JP6193513B2 (https=)
KR (1) KR102149572B1 (https=)
CN (1) CN106459120A (https=)
AU (1) AU2015262993B2 (https=)
BR (1) BR112016026809A2 (https=)
CA (1) CA2891717C (https=)
DK (1) DK3145934T5 (https=)
ES (1) ES2841400T3 (https=)
HU (1) HUE052146T2 (https=)
IL (1) IL248667B (https=)
MX (1) MX381383B (https=)
MY (1) MY181586A (https=)
NZ (1) NZ725600A (https=)
PE (1) PE20170024A1 (https=)
PH (1) PH12016502304A1 (https=)
PL (1) PL3145934T3 (https=)
PT (1) PT3145934T (https=)
RU (1) RU2696490C2 (https=)
SA (1) SA516380328B1 (https=)
SG (1) SG11201608936UA (https=)
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Cited By (2)

* Cited by examiner, † Cited by third party
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CN109232690A (zh) * 2018-09-10 2019-01-18 南方医科大学南方医院 一种正电子显像剂标准品前体及其制备方法
WO2025157263A1 (zh) * 2024-01-26 2025-07-31 浙江养生堂天然药物研究所有限公司 偶联物及其制备方法和用途

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