CN105899505B - 用于治疗自身免疫病症的吡唑 - Google Patents

用于治疗自身免疫病症的吡唑 Download PDF

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CN105899505B
CN105899505B CN201480072420.9A CN201480072420A CN105899505B CN 105899505 B CN105899505 B CN 105899505B CN 201480072420 A CN201480072420 A CN 201480072420A CN 105899505 B CN105899505 B CN 105899505B
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alkyl
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aromatic heterocyclic
optionally
optionally substituted
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CN105899505A (zh
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吉田雅都
高见和明
富成祐介
塩川善右
涉谷章人
佐佐木悠祐
东尼·吉普森
高木辉文
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Takeda Pharmaceutical Co Ltd
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    • A61K9/06—Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
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    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
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  • Physical Education & Sports Medicine (AREA)
  • Psychiatry (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
CN201480072420.9A 2013-11-08 2014-11-05 用于治疗自身免疫病症的吡唑 Active CN105899505B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP2013232571 2013-11-08
JP2013-232571 2013-11-08
JP2014-128562 2014-06-23
JP2014128562 2014-06-23
PCT/JP2014/080005 WO2015068856A1 (en) 2013-11-08 2014-11-05 Pyrazole for the treatment autoimmune disorders

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CN105899505A CN105899505A (zh) 2016-08-24
CN105899505B true CN105899505B (zh) 2018-08-28

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US (2) US9321757B2 (enExample)
EP (1) EP3066094B1 (enExample)
JP (1) JP6412148B2 (enExample)
CN (1) CN105899505B (enExample)
BR (1) BR112016010041B1 (enExample)
CA (1) CA2929316C (enExample)
EA (1) EA201690952A1 (enExample)
ES (1) ES2777123T3 (enExample)
TW (1) TW201605847A (enExample)
UY (1) UY35821A (enExample)
WO (1) WO2015068856A1 (enExample)

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KR102625224B1 (ko) 2018-10-31 2024-01-15 주식회사 큐로젠 피라졸-온 유도체를 유효성분으로 포함하는 자가면역질환의 예방, 개선 또는 치료용 조성물
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EP3066094B1 (en) 2020-01-08
TW201605847A (zh) 2016-02-16
US20160311811A1 (en) 2016-10-27
WO2015068856A1 (en) 2015-05-14
BR112016010041B1 (pt) 2023-04-18
EP3066094A1 (en) 2016-09-14
US9321757B2 (en) 2016-04-26
UY35821A (es) 2015-06-30
CN105899505A (zh) 2016-08-24
BR112016010041A2 (pt) 2020-10-27
US20150133451A1 (en) 2015-05-14
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JP2016535772A (ja) 2016-11-17
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