CN103857405B - 用于调节血清磷的治疗剂 - Google Patents

用于调节血清磷的治疗剂 Download PDF

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Publication number
CN103857405B
CN103857405B CN201280038112.5A CN201280038112A CN103857405B CN 103857405 B CN103857405 B CN 103857405B CN 201280038112 A CN201280038112 A CN 201280038112A CN 103857405 B CN103857405 B CN 103857405B
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hours
hemodialysis
seq
dialysis
amino acid
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CN201280038112.5A
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Chinese (zh)
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CN103857405A (zh
Inventor
F.凯林
G.贝尔
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Kai Pharmaceuticals Inc
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Kai Pharmaceuticals Inc
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/08—Peptides having 5 to 11 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00—Drugs for skeletal disorders
    • A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
    • A61P3/14—Drugs for disorders of the metabolism for electrolyte homeostasis for calcium homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/18—Drugs for disorders of the endocrine system of the parathyroid hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/08—Plasma substitutes; Perfusion solutions; Dialytics or haemodialytics; Drugs for electrolytic or acid-base disorders, e.g. hypovolemic shock
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/06—Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00—Preparations for use in therapy

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Urology & Nephrology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Rheumatology (AREA)
  • Obesity (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Endocrinology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
CN201280038112.5A 2011-06-08 2012-06-08 用于调节血清磷的治疗剂 Active CN103857405B (zh)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201161494874P 2011-06-08 2011-06-08
US61/494,874 2011-06-08
US61/494874 2011-06-08
PCT/US2012/041759 WO2012170955A1 (en) 2011-06-08 2012-06-08 Therapeutic agents for regulating serum phosphorus

Publications (2)

Publication Number Publication Date
CN103857405A CN103857405A (zh) 2014-06-11
CN103857405B true CN103857405B (zh) 2015-12-02

Family

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Family Applications (1)

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CN201280038112.5A Active CN103857405B (zh) 2011-06-08 2012-06-08 用于调节血清磷的治疗剂

Country Status (23)

Country Link
US (1) US8969299B2 (https=)
EP (1) EP2717896B1 (https=)
JP (1) JP5982473B2 (https=)
KR (1) KR102057508B1 (https=)
CN (1) CN103857405B (https=)
AU (1) AU2012267470C1 (https=)
BR (1) BR112013031539A2 (https=)
CA (1) CA2837445C (https=)
CY (1) CY1118430T1 (https=)
DK (1) DK2717896T3 (https=)
ES (1) ES2607986T3 (https=)
HR (1) HRP20161566T1 (https=)
HU (1) HUE032087T2 (https=)
LT (1) LT2717896T (https=)
MX (1) MX337613B (https=)
PL (1) PL2717896T3 (https=)
PT (1) PT2717896T (https=)
RS (1) RS55503B1 (https=)
RU (1) RU2612912C2 (https=)
SG (1) SG195290A1 (https=)
SI (1) SI2717896T1 (https=)
SM (2) SMT201700081T1 (https=)
WO (1) WO2012170955A1 (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2729051T3 (es) 2009-07-29 2019-10-30 Kai Pharmaceuticals Inc Agentes terapéuticos para reducir los niveles de hormona paratiroidea
SMT201700401T1 (it) 2013-06-28 2017-09-07 Amgen Inc Formulazione liquida stabile di amg 416 (velcalcetide)
RU2686086C1 (ru) * 2018-05-17 2019-04-24 федеральное государственное бюджетное образовательное учреждение высшего образования "Первый Санкт-Петербургский государственный медицинский университет имени академика И.П. Павлова" Министерства здравоохранения Российской Федерации Способ коррекции пресаркопении или саркопении у пациента с адекватным потреблением основных нутриентов, получающего лечение программным гемодиализом
CN114222578B (zh) * 2019-12-09 2024-06-25 北京拓界生物医药科技有限公司 钙敏感受体激动剂化合物及其应用
KR20230066044A (ko) * 2020-09-10 2023-05-12 샨시 마이콧 테크놀로지 컴퍼니 리미티드 이중특이적 융합 폴리펩타이드 화합물

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WO2011014707A2 (en) * 2009-07-29 2011-02-03 Kai Pharmaceuticals, Inc. Therapeutic agents for reducing parathyroid hormone levels

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Publication number Publication date
DK2717896T3 (en) 2016-12-19
RU2612912C2 (ru) 2017-03-13
ES2607986T3 (es) 2017-04-05
RS55503B1 (sr) 2017-05-31
MX337613B (es) 2016-03-10
WO2012170955A1 (en) 2012-12-13
AU2012267470B2 (en) 2017-06-15
US20130150301A1 (en) 2013-06-13
PT2717896T (pt) 2016-12-23
SI2717896T1 (sl) 2017-04-26
KR20140035456A (ko) 2014-03-21
CY1118430T1 (el) 2017-06-28
SG195290A1 (en) 2013-12-30
CA2837445A1 (en) 2012-12-13
AU2012267470C1 (en) 2017-09-21
LT2717896T (lt) 2017-02-27
CN103857405A (zh) 2014-06-11
HRP20161566T1 (hr) 2017-02-24
EP2717896A1 (en) 2014-04-16
BR112013031539A2 (pt) 2019-07-30
MX2013014249A (es) 2014-01-24
PL2717896T3 (pl) 2017-05-31
JP2014522414A (ja) 2014-09-04
HUE032087T2 (en) 2017-08-28
SMT201700081B (it) 2017-03-08
KR102057508B1 (ko) 2019-12-19
CA2837445C (en) 2022-10-04
EP2717896B1 (en) 2016-08-24
US8969299B2 (en) 2015-03-03
SMT201700081T1 (it) 2017-03-08
RU2013157928A (ru) 2015-07-20
JP5982473B2 (ja) 2016-08-31

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