CN103501610A - Pi3激酶抑制剂和其用途 - Google Patents

Pi3激酶抑制剂和其用途 Download PDF

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Publication number
CN103501610A
CN103501610A CN201280021536.0A CN201280021536A CN103501610A CN 103501610 A CN103501610 A CN 103501610A CN 201280021536 A CN201280021536 A CN 201280021536A CN 103501610 A CN103501610 A CN 103501610A
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ring
nhc
nitrogen
compound
optionally substituted
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Chinese (zh)
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乔立新
牛德强
拉塞尔·C·彼得
朱振东
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Avila Therapeutics Inc
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Avila Therapeutics Inc
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CN201280021536.0A 2011-03-09 2012-03-08 Pi3激酶抑制剂和其用途 Pending CN103501610A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201161451022P 2011-03-09 2011-03-09
US61/451,022 2011-03-09
PCT/US2012/028293 WO2012122383A2 (en) 2011-03-09 2012-03-08 Pi3 kinase inhibitors and uses thereof

Publications (1)

Publication Number Publication Date
CN103501610A true CN103501610A (zh) 2014-01-08

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CN201280021536.0A Pending CN103501610A (zh) 2011-03-09 2012-03-08 Pi3激酶抑制剂和其用途

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US (1) US20120258967A1 (https=)
EP (1) EP2683243A4 (https=)
JP (1) JP2014511395A (https=)
CN (1) CN103501610A (https=)
AU (1) AU2012225382B2 (https=)
CA (1) CA2829558A1 (https=)
WO (1) WO2012122383A2 (https=)

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EP3877371A4 (en) 2018-11-07 2022-07-27 Dana-Farber Cancer Institute, Inc. IMIDAZOPYRIDINE DERIVATIVES AND AZA-IMIDAZOPYRIDINE DERIVATIVES AS JANUS KINASE 2 INHIBITORS AND USES THEREOF
WO2020097398A1 (en) 2018-11-07 2020-05-14 Dana-Farber Cancer Institute, Inc. Benzothiazole derivatives and 7-aza-benzothiazole derivatives as janus kinase 2 inhibitors and uses thereof
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AU2021324684A1 (en) * 2020-08-11 2023-04-20 Board Of Trustees Of Michigan State University Proteasome enhancers and uses thereof
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TW202325289A (zh) 2021-11-09 2023-07-01 美商雅捷可斯治療公司 Ｊａｋ２抑制劑之形式及組合物
JP7782035B2 (ja) 2021-11-09 2025-12-08 エイジャックス セラピューティクス， インコーポレイテッド Ｊａｋ２阻害剤としての６－ヘテロアリールオキシベンゾイミダゾール及びアザベンゾイミダゾール
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