CN102791135B - 噻唑并[5,4-d]嘧啶以及它们作为农用化学品的用途 - Google Patents

噻唑并[5,4-d]嘧啶以及它们作为农用化学品的用途 Download PDF

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Publication number
CN102791135B
CN102791135B CN201180012818.XA CN201180012818A CN102791135B CN 102791135 B CN102791135 B CN 102791135B CN 201180012818 A CN201180012818 A CN 201180012818A CN 102791135 B CN102791135 B CN 102791135B
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China
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spp
compound
compounds
ethyl
thiazolo
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Expired - Fee Related
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CN201180012818.XA
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English (en)
Chinese (zh)
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CN102791135A (zh
Inventor
W.布鲁斯特
C.克里蒂科
B.里德
T.西德尔
姚成林
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Corteva Agriscience LLC
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Dow AgroSciences LLC
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/429—Thiazoles condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Zoology (AREA)
  • Dentistry (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pretreatment Of Seeds And Plants (AREA)
  • Plural Heterocyclic Compounds (AREA)
CN201180012818.XA 2010-01-07 2011-01-06 噻唑并[5,4-d]嘧啶以及它们作为农用化学品的用途 Expired - Fee Related CN102791135B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US29301410P 2010-01-07 2010-01-07
US61/293,014 2010-01-07
PCT/US2011/020351 WO2011085084A1 (en) 2010-01-07 2011-01-06 THIAZOLO[5,4-d] PYRIMIDINES AND THEIR USE AS AGROCHEMICALS

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Publication Number Publication Date
CN102791135A CN102791135A (zh) 2012-11-21
CN102791135B true CN102791135B (zh) 2015-05-20

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Country Link
US (1) US8921382B2 (https=)
EP (1) EP2521452B1 (https=)
JP (1) JP5781090B2 (https=)
KR (1) KR101814835B1 (https=)
CN (1) CN102791135B (https=)
BR (1) BR112012016866A2 (https=)
CA (1) CA2786250A1 (https=)
CL (1) CL2012001851A1 (https=)
CO (1) CO6612238A2 (https=)
ES (1) ES2529247T3 (https=)
IN (1) IN2012DN06323A (https=)
MX (1) MX2012007954A (https=)
PL (1) PL2521452T3 (https=)
PT (1) PT2521452E (https=)
RU (1) RU2547721C2 (https=)
UA (1) UA109780C2 (https=)
WO (1) WO2011085084A1 (https=)
ZA (1) ZA201204871B (https=)

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AR088218A1 (es) 2011-07-19 2014-05-21 Infinity Pharmaceuticals Inc Compuestos heterociclicos utiles como inhibidores de pi3k
WO2013031694A1 (ja) * 2011-08-26 2013-03-07 富山化学工業株式会社 アミン化合物またはその塩
PT3513793T (pt) 2011-09-02 2021-05-10 Incyte Holdings Corp Heterociclilaminas como inibidores de pi3k
AU2013214353A1 (en) 2012-02-03 2014-08-21 Basf Se Fungicidal pyrimidine compounds
AU2013214137A1 (en) 2012-02-03 2014-08-21 Basf Se Fungicidal pyrimidine compounds
WO2013135672A1 (en) 2012-03-13 2013-09-19 Basf Se Fungicidal pyrimidine compounds
AR090548A1 (es) 2012-04-02 2014-11-19 Incyte Corp Azaheterociclobencilaminas biciclicas como inhibidores de pi3k
CN103668956B (zh) * 2012-09-21 2015-08-12 上海韬鸿化工科技有限公司 防螨虫整理剂、织物的防螨虫整理方法及防螨虫织物
BR112015023640A2 (pt) * 2013-03-15 2017-07-18 Univ California métodos para identificar repelentes e atraentes de artrópodes e compostos e composições identificados por tais métodos
WO2015191677A1 (en) * 2014-06-11 2015-12-17 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as pi3k inhibitors
CN105594748A (zh) * 2014-10-15 2016-05-25 浙江新安化工集团股份有限公司 一种精准定向、高效的防治鳞翅目害虫的杀虫组合物及其使用方法
CN104391070B (zh) * 2014-12-05 2016-06-08 山东省城市供排水水质监测中心 一种水中烷基汞的检测方法
SG10201907576SA (en) 2015-02-27 2019-09-27 Incyte Corp Salts of pi3k inhibitor and processes for their preparation
US20160272612A1 (en) 2015-03-18 2016-09-22 The Regents Of The University Of California Anthropod repellent chemicals
US9988401B2 (en) 2015-05-11 2018-06-05 Incyte Corporation Crystalline forms of a PI3K inhibitor
CN105606755A (zh) * 2016-01-30 2016-05-25 郭庆龙 一种胺苯吡唑酮残留量的gc-nci-ms测定方法
TWI760428B (zh) 2017-01-26 2022-04-11 日商三井化學Agro股份有限公司 吡啶酮化合物及以吡啶酮化合物作為有效成分的農園藝用殺菌劑
JP7134946B2 (ja) 2017-04-10 2022-09-12 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
US11147272B2 (en) 2017-04-10 2021-10-19 Mitsui Chemicals Argro, Inc. Pyridone compounds and agricultural and horticultural fungicides comprising the same as active ingredients
BR112019021388B1 (pt) 2017-04-11 2023-10-31 Mitsui Chemicals Crop & Life Solutions, Inc Compostos, agente de controle de pragas agrícolas e hortícolas, fungicida agrícola e hortícola e métodos para prevenção e/ou tratamento de uma doença de plantas
JP7157738B2 (ja) 2017-06-08 2022-10-20 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
SG11202011680YA (en) 2018-06-01 2020-12-30 Incyte Corp Dosing regimen for the treatment of pi3k related disorders
EP3828177B1 (en) 2018-07-25 2023-11-29 Mitsui Chemicals Crop & Life Solutions, Inc. Pyridone compound and agricultural and horticultural fungicide having this as active component
PH12022552032A1 (en) 2020-02-11 2023-11-29 Syngenta Crop Protection Ag Method of controlling fungi
CN112010848B (zh) * 2020-09-29 2021-12-24 南通大学 含三氟甲基吡啶联芳氧基结构的1,3,4-噁二唑类化合物的制备方法和应用
CN116250525B (zh) * 2023-03-08 2024-12-24 内蒙古民族大学 一种小型哺乳类剥制标本安全防腐剂及其制备方法

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Publication number Publication date
CN102791135A (zh) 2012-11-21
UA109780C2 (uk) 2015-10-12
WO2011085084A1 (en) 2011-07-14
BR112012016866A2 (pt) 2015-09-01
JP2013516476A (ja) 2013-05-13
RU2012133570A (ru) 2014-02-20
EP2521452A1 (en) 2012-11-14
PT2521452E (pt) 2015-02-24
US8921382B2 (en) 2014-12-30
EP2521452B1 (en) 2014-12-24
KR20120115538A (ko) 2012-10-18
MX2012007954A (es) 2012-08-03
CL2012001851A1 (es) 2012-12-14
JP5781090B2 (ja) 2015-09-16
ZA201204871B (en) 2013-09-25
PL2521452T3 (pl) 2015-05-29
CO6612238A2 (es) 2013-02-01
KR101814835B1 (ko) 2018-01-04
ES2529247T3 (es) 2015-02-18
IN2012DN06323A (https=) 2015-10-02
EP2521452A4 (en) 2013-07-03
CA2786250A1 (en) 2011-07-14
US20110166164A1 (en) 2011-07-07
HK1176236A1 (en) 2013-07-26
RU2547721C2 (ru) 2015-04-10

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