CN102791135B - 噻唑并[5,4-d]嘧啶以及它们作为农用化学品的用途 - Google Patents

噻唑并[5,4-d]嘧啶以及它们作为农用化学品的用途 Download PDF

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Publication number
CN102791135B
CN102791135B CN201180012818.XA CN201180012818A CN102791135B CN 102791135 B CN102791135 B CN 102791135B CN 201180012818 A CN201180012818 A CN 201180012818A CN 102791135 B CN102791135 B CN 102791135B
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CN
China
Prior art keywords
spp
compound
compounds
ethyl
thiazolo
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Expired - Fee Related
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CN201180012818.XA
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English (en)
Chinese (zh)
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CN102791135A (zh
Inventor
W.布鲁斯特
C.克里蒂科
B.里德
T.西德尔
姚成林
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Corteva Agriscience LLC
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Dow AgroSciences LLC
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/429—Thiazoles condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Zoology (AREA)
  • Dentistry (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pretreatment Of Seeds And Plants (AREA)
CN201180012818.XA 2010-01-07 2011-01-06 噻唑并[5,4-d]嘧啶以及它们作为农用化学品的用途 Expired - Fee Related CN102791135B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US29301410P 2010-01-07 2010-01-07
US61/293,014 2010-01-07
PCT/US2011/020351 WO2011085084A1 (en) 2010-01-07 2011-01-06 THIAZOLO[5,4-d] PYRIMIDINES AND THEIR USE AS AGROCHEMICALS

Publications (2)

Publication Number Publication Date
CN102791135A CN102791135A (zh) 2012-11-21
CN102791135B true CN102791135B (zh) 2015-05-20

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Country Link
US (1) US8921382B2 (cg-RX-API-DMAC7.html)
EP (1) EP2521452B1 (cg-RX-API-DMAC7.html)
JP (1) JP5781090B2 (cg-RX-API-DMAC7.html)
KR (1) KR101814835B1 (cg-RX-API-DMAC7.html)
CN (1) CN102791135B (cg-RX-API-DMAC7.html)
BR (1) BR112012016866A2 (cg-RX-API-DMAC7.html)
CA (1) CA2786250A1 (cg-RX-API-DMAC7.html)
CL (1) CL2012001851A1 (cg-RX-API-DMAC7.html)
CO (1) CO6612238A2 (cg-RX-API-DMAC7.html)
ES (1) ES2529247T3 (cg-RX-API-DMAC7.html)
IN (1) IN2012DN06323A (cg-RX-API-DMAC7.html)
MX (1) MX2012007954A (cg-RX-API-DMAC7.html)
PL (1) PL2521452T3 (cg-RX-API-DMAC7.html)
PT (1) PT2521452E (cg-RX-API-DMAC7.html)
RU (1) RU2547721C2 (cg-RX-API-DMAC7.html)
UA (1) UA109780C2 (cg-RX-API-DMAC7.html)
WO (1) WO2011085084A1 (cg-RX-API-DMAC7.html)
ZA (1) ZA201204871B (cg-RX-API-DMAC7.html)

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WO2013031694A1 (ja) * 2011-08-26 2013-03-07 富山化学工業株式会社 アミン化合物またはその塩
MX389479B (es) 2011-09-02 2025-03-20 Incyte Holdings Corp Heterociclilaminas como inhibidores de fosfoinositida 3-cinasas (pi3k)
IN2014DN07224A (cg-RX-API-DMAC7.html) 2012-02-03 2015-04-24 Basf Se
CA2862354A1 (en) 2012-02-03 2013-08-08 Basf Se Fungicidal pyrimidine compounds
WO2013135672A1 (en) 2012-03-13 2013-09-19 Basf Se Fungicidal pyrimidine compounds
AR090548A1 (es) 2012-04-02 2014-11-19 Incyte Corp Azaheterociclobencilaminas biciclicas como inhibidores de pi3k
CN103668956B (zh) * 2012-09-21 2015-08-12 上海韬鸿化工科技有限公司 防螨虫整理剂、织物的防螨虫整理方法及防螨虫织物
BR112015023640A2 (pt) * 2013-03-15 2017-07-18 Univ California métodos para identificar repelentes e atraentes de artrópodes e compostos e composições identificados por tais métodos
US10077277B2 (en) 2014-06-11 2018-09-18 Incyte Corporation Bicyclic heteroarylaminoalkyl phenyl derivatives as PI3K inhibitors
CN105594748A (zh) * 2014-10-15 2016-05-25 浙江新安化工集团股份有限公司 一种精准定向、高效的防治鳞翅目害虫的杀虫组合物及其使用方法
CN104391070B (zh) * 2014-12-05 2016-06-08 山东省城市供排水水质监测中心 一种水中烷基汞的检测方法
SG10201912302VA (en) 2015-02-27 2020-02-27 Incyte Corp Salts of pi3k inhibitor and processes for their preparation
EP3270692A4 (en) 2015-03-18 2019-02-13 The Regents of the University of California CHEMICALS FOR PROTECTION AGAINST BRANCHES
US9988401B2 (en) 2015-05-11 2018-06-05 Incyte Corporation Crystalline forms of a PI3K inhibitor
CN105606755A (zh) * 2016-01-30 2016-05-25 郭庆龙 一种胺苯吡唑酮残留量的gc-nci-ms测定方法
JP7037507B2 (ja) 2017-01-26 2022-03-16 三井化学アグロ株式会社 ピリドン化合物およびそれを有効成分とする農園芸用殺菌剤
TWI793113B (zh) 2017-04-10 2023-02-21 日商三井化學Agro股份有限公司 吡啶酮化合物及以吡啶酮化合物作為有效成分的農園藝用殺菌劑
CA3059675A1 (en) 2017-04-10 2018-10-18 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides comprising the same as active ingredients
KR102498819B1 (ko) 2017-04-11 2023-02-10 미쓰이가가쿠 아그로 가부시키가이샤 피리돈 화합물 및 그것을 유효성분으로 하는 농원예용 살균제
US11117863B2 (en) 2017-06-08 2021-09-14 Mitsui Chemicals Agro, Inc. Pyridone compounds and agricultural and horticultural fungicides containing the same as active ingredients
IL278889B2 (en) 2018-06-01 2025-11-01 Incyte Corp Dosing regimen for the treatment of pi3k related disorders
EP3828177B1 (en) 2018-07-25 2023-11-29 Mitsui Chemicals Crop & Life Solutions, Inc. Pyridone compound and agricultural and horticultural fungicide having this as active component
US12317896B2 (en) 2020-02-11 2025-06-03 Syngenta Crop Protection Ag Method of controlling fungi
CN112010848B (zh) * 2020-09-29 2021-12-24 南通大学 含三氟甲基吡啶联芳氧基结构的1,3,4-噁二唑类化合物的制备方法和应用
CN116250525B (zh) * 2023-03-08 2024-12-24 内蒙古民族大学 一种小型哺乳类剥制标本安全防腐剂及其制备方法
CN122422314A (zh) 2023-12-08 2026-07-17 三井化学植保株式会社 双环式杂环化合物以及以双环式杂环化合物作为有效成分的农业园艺用杀菌剂
CN117903168A (zh) * 2024-01-26 2024-04-19 南开大学 一类含吡咯并[2,3-d]噻唑衍生物及其制备方法和用途

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JP5781090B2 (ja) 2015-09-16
US8921382B2 (en) 2014-12-30
CO6612238A2 (es) 2013-02-01
MX2012007954A (es) 2012-08-03
IN2012DN06323A (cg-RX-API-DMAC7.html) 2015-10-02
JP2013516476A (ja) 2013-05-13
WO2011085084A1 (en) 2011-07-14
RU2547721C2 (ru) 2015-04-10
KR101814835B1 (ko) 2018-01-04
ES2529247T3 (es) 2015-02-18
BR112012016866A2 (pt) 2015-09-01
RU2012133570A (ru) 2014-02-20
CN102791135A (zh) 2012-11-21
US20110166164A1 (en) 2011-07-07
CL2012001851A1 (es) 2012-12-14
EP2521452A1 (en) 2012-11-14
PL2521452T3 (pl) 2015-05-29
UA109780C2 (uk) 2015-10-12
PT2521452E (pt) 2015-02-24
HK1176236A1 (en) 2013-07-26
KR20120115538A (ko) 2012-10-18
ZA201204871B (en) 2013-09-25
EP2521452A4 (en) 2013-07-03
EP2521452B1 (en) 2014-12-24
CA2786250A1 (en) 2011-07-14

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