CN102625660B - 亚氨基糖以及治疗沙粒病毒感染的方法 - Google Patents

亚氨基糖以及治疗沙粒病毒感染的方法 Download PDF

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Publication number
CN102625660B
CN102625660B CN201080017592.8A CN201080017592A CN102625660B CN 102625660 B CN102625660 B CN 102625660B CN 201080017592 A CN201080017592 A CN 201080017592A CN 102625660 B CN102625660 B CN 102625660B
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virus
use according
dnj
pharmaceutically acceptable
acceptable salt
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Chinese (zh)
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CN102625660A (zh
Inventor
厄本·拉姆斯泰特
布伦南·克洛斯
妮科尔·齐兹曼
雷蒙德·A·德韦克
特里·D·巴特斯
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University of Oxford
United Therapeutics Corp
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University of Oxford
United Therapeutics Corp
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/10—Dispersions; Emulsions
    • A61K9/12—Aerosols; Foams
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00—Preparations for use in therapy

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Dispersion Chemistry (AREA)
  • Molecular Biology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
CN201080017592.8A 2009-02-24 2010-02-22 亚氨基糖以及治疗沙粒病毒感染的方法 Expired - Fee Related CN102625660B (zh)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US20239109P 2009-02-24 2009-02-24
US61/202,391 2009-02-24
US27225109P 2009-09-04 2009-09-04
US61/272,251 2009-09-04
PCT/US2010/024914 WO2010099064A1 (en) 2009-02-24 2010-02-22 Iminosugars and methods of treating arenaviral infections

Publications (2)

Publication Number Publication Date
CN102625660A CN102625660A (zh) 2012-08-01
CN102625660B true CN102625660B (zh) 2015-03-11

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CN201080017592.8A Expired - Fee Related CN102625660B (zh) 2009-02-24 2010-02-22 亚氨基糖以及治疗沙粒病毒感染的方法

Country Status (8)

Country Link
US (1) US20100222384A1 (https=)
EP (1) EP2400843B1 (https=)
JP (1) JP5951996B2 (https=)
KR (2) KR20170117614A (https=)
CN (1) CN102625660B (https=)
CA (1) CA2753194A1 (https=)
ES (1) ES2562635T3 (https=)
WO (1) WO2010099064A1 (https=)

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CA2753195C (en) 2009-02-23 2015-06-02 United Therapeutics Corporation Iminosugars and methods of treating viral diseases
IN2014MN02539A (https=) 2012-06-06 2015-07-24 Unither Virology Llc
CN102775384B (zh) * 2012-07-27 2015-05-27 中国科学院化学研究所 小钩树碱i和j类似物及其制备方法与应用
CN106102464A (zh) * 2013-05-02 2016-11-09 牛津大学之校长及学者 采用亚氨基糖的糖脂抑制
KR20160055916A (ko) 2013-09-16 2016-05-18 이머전트 바이롤로지 엘엘씨 데옥시노지리마이신 유도체 및 그의 이용 방법
IT202000008917A1 (it) * 2020-04-24 2021-10-24 Biovalley Invest Partner S R L Composizioni antivirali
KR20250160378A (ko) 2024-05-06 2025-11-13 문제정 가구재용 서랍 조립시스템

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Also Published As

Publication number Publication date
WO2010099064A1 (en) 2010-09-02
CA2753194A1 (en) 2010-09-02
US20100222384A1 (en) 2010-09-02
HK1165675A1 (en) 2012-10-12
JP2012518648A (ja) 2012-08-16
CN102625660A (zh) 2012-08-01
KR20170117614A (ko) 2017-10-23
EP2400843B1 (en) 2015-11-11
KR20120042718A (ko) 2012-05-03
KR101787434B1 (ko) 2017-11-15
EP2400843A1 (en) 2012-01-04
JP5951996B2 (ja) 2016-07-13
ES2562635T3 (es) 2016-03-07
EP2400843A4 (en) 2012-01-04

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Termination date: 20190222