CN102056485A - 用于局部治疗免疫相关疾病的局部lfa-1拮抗剂 - Google Patents

用于局部治疗免疫相关疾病的局部lfa-1拮抗剂 Download PDF

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CN102056485A
CN102056485A CN2009801216301A CN200980121630A CN102056485A CN 102056485 A CN102056485 A CN 102056485A CN 2009801216301 A CN2009801216301 A CN 2009801216301A CN 200980121630 A CN200980121630 A CN 200980121630A CN 102056485 A CN102056485 A CN 102056485A
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lfa
antagonist
aliphatic
preparation
aryl
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CN2009801216301A
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Chinese (zh)
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J·伯尼尔
T·盖德克
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Sarcode Bioscience Inc
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Sarcode Corp
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Priority to CN201610115732.4A priority Critical patent/CN105943534A/zh
Publication of CN102056485A publication Critical patent/CN102056485A/zh
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    • A—HUMAN NECESSITIES
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    • A61K9/0014—Skin, i.e. galenical aspects of topical compositions
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
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  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
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  • Nitrogen Condensed Heterocyclic Rings (AREA)
CN2009801216301A 2008-04-15 2009-04-15 用于局部治疗免疫相关疾病的局部lfa-1拮抗剂 Pending CN102056485A (zh)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CN201610115732.4A CN105943534A (zh) 2008-04-15 2009-04-15 用于局部治疗免疫相关疾病的局部lfa-1拮抗剂

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Application Number Priority Date Filing Date Title
US4524008P 2008-04-15 2008-04-15
US61/045,240 2008-04-15
PCT/US2009/002389 WO2009128934A1 (en) 2008-04-15 2009-04-15 Topical lfa-1 antagonists for use in localized treatment of immune related disorders

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CN201610115732.4A Division CN105943534A (zh) 2008-04-15 2009-04-15 用于局部治疗免疫相关疾病的局部lfa-1拮抗剂

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US (2) US20090258070A1 (cg-RX-API-DMAC7.html)
EP (2) EP2265125B1 (cg-RX-API-DMAC7.html)
JP (2) JP2011521896A (cg-RX-API-DMAC7.html)
CN (1) CN102056485A (cg-RX-API-DMAC7.html)
ES (1) ES2763703T3 (cg-RX-API-DMAC7.html)
WO (1) WO2009128934A1 (cg-RX-API-DMAC7.html)

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WO2025223511A1 (zh) * 2024-04-25 2025-10-30 上海翊石医药科技有限公司 一类苯甲酰基甘氨酸衍生物及其制备方法和应用

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US20090257957A1 (en) * 2008-04-15 2009-10-15 John Burnier Aerosolized LFA-1 antagonists for use in localized treatment of immune related disorders
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TW201920956A (zh) * 2017-09-29 2019-06-01 日商參天製藥股份有限公司 淚液中之muc5ac量之測定方法
CN111787918A (zh) * 2017-11-29 2020-10-16 洛克菲勒大学 用于皮肤病学病况增强治疗的局部和全身性治疗的组合
KR20220003555A (ko) * 2019-04-18 2022-01-10 아주라 오프탈믹스 엘티디 안구 장애의 치료를 위한 화합물 및 방법
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