CN101687809A - 过渡金属催化的2h-吲唑合成 - Google Patents

过渡金属催化的2h-吲唑合成 Download PDF

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Publication number
CN101687809A
CN101687809A CN200880021936A CN200880021936A CN101687809A CN 101687809 A CN101687809 A CN 101687809A CN 200880021936 A CN200880021936 A CN 200880021936A CN 200880021936 A CN200880021936 A CN 200880021936A CN 101687809 A CN101687809 A CN 101687809A
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China
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substituted
alkyl
replace
phenyl
another
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Chinese (zh)
Inventor
N·哈兰
M·纳扎雷
A·林登施密德
J·阿朗索
O·勒克亚克
M·乌尔曼
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Sanofi Aventis France
Sanofi Aventis SpA
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Sanofi Aventis SpA
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Publication of CN101687809A publication Critical patent/CN101687809A/zh
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Catalysts (AREA)
CN200880021936A 2007-06-26 2008-06-11 过渡金属催化的2h-吲唑合成 Pending CN101687809A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP07290799.1 2007-06-26
EP07290799 2007-06-26
PCT/EP2008/004637 WO2009000411A1 (en) 2007-06-26 2008-06-11 A transition metal catalyzed synthesis of 2h-indazoles

Publications (1)

Publication Number Publication Date
CN101687809A true CN101687809A (zh) 2010-03-31

Family

ID=38577414

Family Applications (1)

Application Number Title Priority Date Filing Date
CN200880021936A Pending CN101687809A (zh) 2007-06-26 2008-06-11 过渡金属催化的2h-吲唑合成

Country Status (12)

Country Link
US (1) US8283476B2 (https=)
EP (1) EP2170833B1 (https=)
JP (1) JP5250029B2 (https=)
KR (1) KR20100024963A (https=)
CN (1) CN101687809A (https=)
AT (1) ATE511501T1 (https=)
AU (1) AU2008267442A1 (https=)
BR (1) BRPI0813870A2 (https=)
CA (1) CA2693024A1 (https=)
IL (1) IL202825A0 (https=)
MX (1) MX2009014203A (https=)
WO (1) WO2009000411A1 (https=)

Cited By (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2012139495A1 (en) * 2011-04-13 2012-10-18 Merck Sharp & Dohme Corp. Mineralocorticoid receptor antagonists
CN104812755A (zh) * 2012-10-31 2015-07-29 拉夸里亚创药株式会社 作为ttx-s阻断剂的吡唑并吡啶衍生物
TWI646102B (zh) * 2016-12-30 2019-01-01 新加坡商沙特基礎工業愛思開奈克斯林恩私人有限公司 新穎環戊［Ｂ］苯硫基過渡金屬化合物、包含該化合物的過渡金屬催化劑組合物、以及使用該化合物製備乙烯均聚物或乙烯與α-烯烴的共聚物的方法
CN110317204A (zh) * 2019-08-02 2019-10-11 安徽农业大学 吡唑并嘧啶酮类衍生物及其制备方法和应用
CN113698349A (zh) * 2021-09-02 2021-11-26 河南师范大学 一种2-(2-苯基-2h-吲唑-3-基)乙酸酯类化合物的水相光催化制备方法
CN114920699A (zh) * 2022-05-31 2022-08-19 甘肃皓天化学科技有限公司 一种制备6-氯-2-甲基-2h-吲唑-5-胺的方法
CN116457349A (zh) * 2020-11-16 2023-07-18 先正达农作物保护股份公司 除草n-杂芳基吡唑化合物

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN103232462B (zh) * 2013-05-13 2016-03-02 湖北科技学院 香豆素-吡咯类化合物的合成方法
WO2016144678A1 (en) * 2015-03-12 2016-09-15 E I Du Pont De Nemours And Company Heterocycle-substituted bicyclic azole pesticides
KR101931234B1 (ko) 2016-02-12 2018-12-21 주식회사 엘지화학 신규한 리간드 화합물 및 전이금속 화합물
WO2017138783A1 (ko) * 2016-02-12 2017-08-17 주식회사 엘지화학 신규한 리간드 화합물 및 전이금속 화합물
KR102095007B1 (ko) * 2016-02-12 2020-03-30 주식회사 엘지화학 신규한 리간드 화합물 및 전이금속 화합물의 제조방법
WO2019233994A1 (en) 2018-06-04 2019-12-12 Exscientia Ltd Pyrazolopyrimidine compounds as adenosine receptor antagonists

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1999043643A2 (en) * 1998-02-26 1999-09-02 Massachusetts Institute Of Technology Metal-catalyzed arylations and vinylations of hydrazines, hydrazones, hydroxylamines and oximes

Cited By (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2012139495A1 (en) * 2011-04-13 2012-10-18 Merck Sharp & Dohme Corp. Mineralocorticoid receptor antagonists
CN104812755A (zh) * 2012-10-31 2015-07-29 拉夸里亚创药株式会社 作为ttx-s阻断剂的吡唑并吡啶衍生物
CN104812755B (zh) * 2012-10-31 2017-08-08 拉夸里亚创药株式会社 作为ttx‑s阻断剂的吡唑并吡啶衍生物
TWI646102B (zh) * 2016-12-30 2019-01-01 新加坡商沙特基礎工業愛思開奈克斯林恩私人有限公司 新穎環戊［Ｂ］苯硫基過渡金屬化合物、包含該化合物的過渡金屬催化劑組合物、以及使用該化合物製備乙烯均聚物或乙烯與α-烯烴的共聚物的方法
CN110317204A (zh) * 2019-08-02 2019-10-11 安徽农业大学 吡唑并嘧啶酮类衍生物及其制备方法和应用
CN110317204B (zh) * 2019-08-02 2022-02-08 安徽农业大学 吡唑并嘧啶酮类衍生物及其制备方法和应用
CN116457349A (zh) * 2020-11-16 2023-07-18 先正达农作物保护股份公司 除草n-杂芳基吡唑化合物
CN113698349A (zh) * 2021-09-02 2021-11-26 河南师范大学 一种2-(2-苯基-2h-吲唑-3-基)乙酸酯类化合物的水相光催化制备方法
CN113698349B (zh) * 2021-09-02 2023-08-01 河南师范大学 一种2-(2-苯基-2h-吲唑-3-基)乙酸酯类化合物的水相光催化制备方法
CN114920699A (zh) * 2022-05-31 2022-08-19 甘肃皓天化学科技有限公司 一种制备6-氯-2-甲基-2h-吲唑-5-胺的方法
CN114920699B (zh) * 2022-05-31 2024-03-19 甘肃皓天科技股份有限公司 一种制备6-氯-2-甲基-2h-吲唑-5-胺的方法

Also Published As

Publication number Publication date
JP5250029B2 (ja) 2013-07-31
EP2170833B1 (en) 2011-06-01
IL202825A0 (en) 2010-06-30
JP2010531311A (ja) 2010-09-24
US20100234601A1 (en) 2010-09-16
AU2008267442A1 (en) 2008-12-31
BRPI0813870A2 (pt) 2015-01-06
ATE511501T1 (de) 2011-06-15
WO2009000411A1 (en) 2008-12-31
US8283476B2 (en) 2012-10-09
EP2170833A1 (en) 2010-04-07
MX2009014203A (es) 2010-01-28
KR20100024963A (ko) 2010-03-08
CA2693024A1 (en) 2008-12-31

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