CN101189248A - 新型含磷拟甲状腺素药 - Google Patents
新型含磷拟甲状腺素药 Download PDFInfo
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- CN101189248A CN101189248A CNA2006800177325A CN200680017732A CN101189248A CN 101189248 A CN101189248 A CN 101189248A CN A2006800177325 A CNA2006800177325 A CN A2006800177325A CN 200680017732 A CN200680017732 A CN 200680017732A CN 101189248 A CN101189248 A CN 101189248A
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Classifications
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- C07F9/4461—Amides thereof the amide moiety containing a substituent or a structure which is considered as characteristic
- C07F9/4465—Amides thereof the amide moiety containing a substituent or a structure which is considered as characteristic of aliphatic amines
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- C07F9/657163—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and oxygen atoms as the only ring hetero atoms the ring phosphorus atom being bound to at least one carbon atom
- C07F9/657181—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having phosphorus atoms, with or without nitrogen, oxygen, sulfur, selenium or tellurium atoms, as ring hetero atoms having phosphorus and oxygen atoms as the only ring hetero atoms the ring phosphorus atom being bound to at least one carbon atom the ring phosphorus atom and, at least, one ring oxygen atom being part of a (thio)phosphonic acid derivative
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Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US11/137,773 | 2005-05-26 | ||
US11/137,773 US7514419B2 (en) | 2003-11-19 | 2005-05-26 | Phosphorus-containing thyromimetics |
US72517005P | 2005-10-06 | 2005-10-06 | |
US60/725,170 | 2005-10-06 | ||
PCT/US2006/020607 WO2006128055A2 (fr) | 2005-05-26 | 2006-05-26 | Nouvelles substances thyromimetiques contenant du phosphore |
Publications (1)
Publication Number | Publication Date |
---|---|
CN101189248A true CN101189248A (zh) | 2008-05-28 |
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ID=37057345
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CNA2006800177325A Pending CN101189248A (zh) | 2005-05-26 | 2006-05-26 | 新型含磷拟甲状腺素药 |
Country Status (7)
Country | Link |
---|---|
EP (1) | EP1891080A2 (fr) |
JP (1) | JP2008545710A (fr) |
CN (1) | CN101189248A (fr) |
AU (1) | AU2006249347A1 (fr) |
CA (1) | CA2606497A1 (fr) |
MX (1) | MX2007014493A (fr) |
WO (1) | WO2006128055A2 (fr) |
Cited By (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN110726801A (zh) * | 2019-10-31 | 2020-01-24 | 山东泰星新材料股份有限公司 | 一种监测烷基次膦酸反应状态的方法 |
WO2020118564A1 (fr) * | 2018-12-12 | 2020-06-18 | Autobahn Therapeutics, Inc. | Nouveaux thyromimétiques |
CN112300211A (zh) * | 2019-07-26 | 2021-02-02 | 广东东阳光药业有限公司 | 一种作为甲状腺激素β受体激动剂的化合物及其用途 |
CN113336792A (zh) * | 2020-02-18 | 2021-09-03 | 甘莱制药有限公司 | 一种环状膦酸酯化合物的制备方法 |
CN114315902A (zh) * | 2020-09-30 | 2022-04-12 | 甘莱制药有限公司 | 一种甲状腺激素β受体激动剂的晶体及其制备方法和用途 |
CN114763363A (zh) * | 2021-01-12 | 2022-07-19 | 上海喀露蓝科技有限公司 | 磷酸或磷酸酯类衍生物及其制备方法和其在医药上的用途 |
US11667606B2 (en) | 2019-03-01 | 2023-06-06 | Autobahn Therapeutics, Inc. | Thyromimetics |
US11827596B2 (en) | 2018-12-12 | 2023-11-28 | Autobahn Therapeutics, Inc. | Thyromimetics |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
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CN1882327A (zh) | 2003-11-19 | 2006-12-20 | 症变治疗公司 | 含磷的新的拟甲状腺素药 |
CA2606499C (fr) | 2005-05-26 | 2017-06-13 | Metabasis Therapeutics, Inc. | Composes thyromimetiques utilises pour traiter les maladies hepatiques graisseuses |
WO2010093601A1 (fr) | 2009-02-10 | 2010-08-19 | Metabasis Therapeutics, Inc. | Nouveaux thyromimetiques contenant de l'acide sulfonique et methodes d'utilisation associees |
CA3044059A1 (fr) * | 2016-11-21 | 2018-05-24 | Viking Therapeutics, Inc. | Methodes de traitement de glycogenose |
BR112019025659A2 (pt) * | 2017-06-05 | 2020-08-25 | Viking Therapeutics, Inc. | composições para o tratamento de fibrose |
AU2019238090A1 (en) * | 2018-03-22 | 2020-10-08 | Viking Therapeutics, Inc. | Crystalline forms and methods of producing crystalline forms of a compound |
EP4019524A4 (fr) * | 2019-08-19 | 2024-01-03 | Hepagene Therapeutics (HK) Limited | Composé agoniste du récepteur thr-bêta hétérocyclique, son procédé de préparation et son utilisation |
US11752161B2 (en) | 2020-03-27 | 2023-09-12 | Gannex Pharma Co., Ltd. | Pharmaceutical compositions, method of making and method of using thereof |
WO2023158607A1 (fr) * | 2022-02-18 | 2023-08-24 | Viking Therapeutics, Inc. | Formes polymorphes et procédés de production de formes polymorphes d'un composé |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3357887A (en) * | 1962-12-03 | 1967-12-12 | Upjohn Co | 4-phenoxy-3, 5-dihalophenylalkanols and hypocholesteremic compositions containing the same |
GB9713739D0 (en) * | 1997-06-27 | 1997-09-03 | Karobio Ab | Thyroid receptor ligands |
IL137672A0 (en) * | 2000-08-03 | 2001-10-31 | Dpharm Ltd | Derivatives of branched-chain lipophilic molecules and uses thereof |
AU2003216054B2 (en) * | 2002-01-18 | 2007-01-04 | Merck & Co., Inc. | Selective S1P1/Edg1 receptor agonists |
CN1882327A (zh) * | 2003-11-19 | 2006-12-20 | 症变治疗公司 | 含磷的新的拟甲状腺素药 |
-
2006
- 2006-05-26 WO PCT/US2006/020607 patent/WO2006128055A2/fr active Application Filing
- 2006-05-26 EP EP06760469A patent/EP1891080A2/fr not_active Withdrawn
- 2006-05-26 CN CNA2006800177325A patent/CN101189248A/zh active Pending
- 2006-05-26 MX MX2007014493A patent/MX2007014493A/es not_active Application Discontinuation
- 2006-05-26 CA CA002606497A patent/CA2606497A1/fr not_active Abandoned
- 2006-05-26 AU AU2006249347A patent/AU2006249347A1/en not_active Abandoned
- 2006-05-26 JP JP2008513783A patent/JP2008545710A/ja not_active Withdrawn
Cited By (9)
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WO2020118564A1 (fr) * | 2018-12-12 | 2020-06-18 | Autobahn Therapeutics, Inc. | Nouveaux thyromimétiques |
US11827596B2 (en) | 2018-12-12 | 2023-11-28 | Autobahn Therapeutics, Inc. | Thyromimetics |
US11667606B2 (en) | 2019-03-01 | 2023-06-06 | Autobahn Therapeutics, Inc. | Thyromimetics |
CN112300211A (zh) * | 2019-07-26 | 2021-02-02 | 广东东阳光药业有限公司 | 一种作为甲状腺激素β受体激动剂的化合物及其用途 |
CN112300211B (zh) * | 2019-07-26 | 2023-12-08 | 广东东阳光药业股份有限公司 | 一种作为甲状腺激素β受体激动剂的化合物及其用途 |
CN110726801A (zh) * | 2019-10-31 | 2020-01-24 | 山东泰星新材料股份有限公司 | 一种监测烷基次膦酸反应状态的方法 |
CN113336792A (zh) * | 2020-02-18 | 2021-09-03 | 甘莱制药有限公司 | 一种环状膦酸酯化合物的制备方法 |
CN114315902A (zh) * | 2020-09-30 | 2022-04-12 | 甘莱制药有限公司 | 一种甲状腺激素β受体激动剂的晶体及其制备方法和用途 |
CN114763363A (zh) * | 2021-01-12 | 2022-07-19 | 上海喀露蓝科技有限公司 | 磷酸或磷酸酯类衍生物及其制备方法和其在医药上的用途 |
Also Published As
Publication number | Publication date |
---|---|
WO2006128055A2 (fr) | 2006-11-30 |
JP2008545710A (ja) | 2008-12-18 |
MX2007014493A (es) | 2008-02-07 |
AU2006249347A1 (en) | 2006-11-30 |
EP1891080A2 (fr) | 2008-02-27 |
CA2606497A1 (fr) | 2006-11-30 |
WO2006128055A3 (fr) | 2007-05-24 |
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