CN100384791C - 碳-杂原子双键的催化氢化 - Google Patents

碳-杂原子双键的催化氢化 Download PDF

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Publication number
CN100384791C
CN100384791C CNB2003801045565A CN200380104556A CN100384791C CN 100384791 C CN100384791 C CN 100384791C CN B2003801045565 A CNB2003801045565 A CN B2003801045565A CN 200380104556 A CN200380104556 A CN 200380104556A CN 100384791 C CN100384791 C CN 100384791C
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Chinese (zh)
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CN1717376A (zh
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F·M·诺德
U·皮特尔科夫
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Solvias AG
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Solvias AG
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B41/00—Formation or introduction of functional groups containing oxygen
    • C07B41/02—Formation or introduction of functional groups containing oxygen of hydroxy or O-metal groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B43/00—Formation or introduction of functional groups containing nitrogen
    • C07B43/04—Formation or introduction of functional groups containing nitrogen of amino groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B53/00—Asymmetric syntheses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/16—Radicals substituted by singly bound hetero atoms other than halogen by oxygen atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Catalysts (AREA)
  • Production Of Liquid Hydrocarbon Mixture For Refining Petroleum (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
CNB2003801045565A 2002-12-02 2003-11-27 碳-杂原子双键的催化氢化 Expired - Lifetime CN100384791C (zh)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH20332002 2002-12-02
CH2033/02 2002-12-02

Publications (2)

Publication Number Publication Date
CN1717376A CN1717376A (zh) 2006-01-04
CN100384791C true CN100384791C (zh) 2008-04-30

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CNB2003801045565A Expired - Lifetime CN100384791C (zh) 2002-12-02 2003-11-27 碳-杂原子双键的催化氢化

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US (1) US7446236B2 (cg-RX-API-DMAC7.html)
EP (1) EP1567464B1 (cg-RX-API-DMAC7.html)
JP (1) JP2006508161A (cg-RX-API-DMAC7.html)
CN (1) CN100384791C (cg-RX-API-DMAC7.html)
AT (1) ATE359986T1 (cg-RX-API-DMAC7.html)
AU (1) AU2003298328A1 (cg-RX-API-DMAC7.html)
CA (1) CA2507908A1 (cg-RX-API-DMAC7.html)
DE (1) DE60313357T2 (cg-RX-API-DMAC7.html)
ES (1) ES2283867T3 (cg-RX-API-DMAC7.html)
WO (1) WO2004050585A1 (cg-RX-API-DMAC7.html)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2004298453A1 (en) 2003-12-19 2005-06-30 Altana Pharma Ag Intermediates for the preparation of tricyclic dihydropyrano -imidazo -pyridines derivatives
KR101337045B1 (ko) 2005-02-16 2013-12-05 아나코르 파마슈티칼스 인코포레이티드 보론함유 소분자
EP1976536A4 (en) 2005-12-30 2011-03-02 Anacor Pharmaceuticals Inc SMALL MOLECULES CONTAINING BORON
KR20150013941A (ko) 2006-02-16 2015-02-05 아나코르 파마슈티칼스 인코포레이티드 항염증제로서 보론함유 소분자
CA2645107A1 (en) * 2006-03-10 2007-09-20 Solvias Ag Asymmetric catalytic hydrogenation of prochiral ketones and aldehydes
EP2564857B1 (en) 2008-03-06 2017-05-03 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-inflammatory agents
WO2010027975A1 (en) 2008-09-04 2010-03-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
US8461336B2 (en) * 2008-09-04 2013-06-11 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
ES2863542T3 (es) * 2009-03-17 2021-10-11 Johnson Matthey Plc Proceso para la hidrogenación de cetonas en presencia de catalizadores de Ru (II)
US9440994B2 (en) * 2009-08-14 2016-09-13 Anacor Pharmaceuticals, Inc. Boron containing small molecules as antiprotozoal agents
WO2011049971A1 (en) 2009-10-20 2011-04-28 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as antiprotozoal agents
WO2011060196A1 (en) * 2009-11-11 2011-05-19 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
US8716478B2 (en) 2010-01-27 2014-05-06 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
WO2011116348A1 (en) 2010-03-19 2011-09-22 Anacor Pharmaceuticals, Inc. Boron-containing small molecules as anti-protozoal agent
EA021532B1 (ru) * 2010-04-07 2015-07-30 ГЛАКСОСМИТКЛАЙН ЭлЭлСи Способ получения бензоксаборолов
CA2810021C (en) 2010-09-07 2018-05-29 Anacor Pharmaceuticals, Inc. Boron-containing small molecules
CA2919888C (en) 2013-08-09 2022-10-18 Anacor Pharmaceuticals, Inc. Tricyclic benzoxaborole compounds and uses thereof
GB201401230D0 (en) * 2014-01-24 2014-03-12 Givaudan Sa Improvements in or relating to organic compounds
MA41494B1 (fr) 2015-02-12 2020-10-28 Glaxosmithkline Ip No 2 Ltd Composés benzoxaborole substitués en position 4 et utilisations associées

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002004466A2 (en) * 2000-07-07 2002-01-17 Dsm N.V. Catalyst for asymmetric (transfer) hydrogenation
WO2002022526A2 (en) * 2000-09-13 2002-03-21 Firmenich S.A. Catalytic hydrogenation processes

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2693190B1 (fr) * 1992-07-02 1994-09-23 Elf Aquitaine Procédé d'hydrogénation énantiosélectif de la double liaison C=O OXO.
US6476233B1 (en) * 1998-11-12 2002-11-05 The Penn State Research Foundation Transition metal-catalyzed reactions based on chiral amine oxazolinyl ligands and related compounds

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2002004466A2 (en) * 2000-07-07 2002-01-17 Dsm N.V. Catalyst for asymmetric (transfer) hydrogenation
WO2002022526A2 (en) * 2000-09-13 2002-03-21 Firmenich S.A. Catalytic hydrogenation processes

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
extremely high enantioselectvie redox reaction of ketones ansalcohols catalyzed by RuCl2(PPh3)3(oxazolinylferrocenylphosphine). Yoshiaki Nishibayashi et al.Organometallics,Vol.18 . 1999 *
Ruthenium(II)-catalyzed asymmetric transfer hydrogention ofketones using chiral oxazolinylferrocenylphosphines and oneof their Ru(II) complex. Yasuyoshi Arikawa et al.Journal of Organometallic Chemistry,Vol.572 No.2. 1999 *

Also Published As

Publication number Publication date
DE60313357D1 (de) 2007-05-31
US20060106247A1 (en) 2006-05-18
EP1567464A1 (en) 2005-08-31
EP1567464B1 (en) 2007-04-18
CA2507908A1 (en) 2004-06-17
CN1717376A (zh) 2006-01-04
JP2006508161A (ja) 2006-03-09
WO2004050585A1 (en) 2004-06-17
US7446236B2 (en) 2008-11-04
ATE359986T1 (de) 2007-05-15
DE60313357T2 (de) 2008-01-03
AU2003298328A1 (en) 2004-06-23
ES2283867T3 (es) 2007-11-01

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