CL2020001791A1 - Composiciones farmacéuticas para la piel tópicas que contienen cerdulatinib y usos de estas. - Google Patents

Composiciones farmacéuticas para la piel tópicas que contienen cerdulatinib y usos de estas.

Info

Publication number
CL2020001791A1
CL2020001791A1 CL2020001791A CL2020001791A CL2020001791A1 CL 2020001791 A1 CL2020001791 A1 CL 2020001791A1 CL 2020001791 A CL2020001791 A CL 2020001791A CL 2020001791 A CL2020001791 A CL 2020001791A CL 2020001791 A1 CL2020001791 A1 CL 2020001791A1
Authority
CL
Chile
Prior art keywords
cerdulatinib
pharmaceutical compositions
topical skin
skin pharmaceutical
disclosed
Prior art date
Application number
CL2020001791A
Other languages
English (en)
Inventor
Charles Rodney Greenaway Evans
Cameron Robert Stevenson
Marc Barry Brown
Original Assignee
Dermavant Sciences GmbH
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dermavant Sciences GmbH filed Critical Dermavant Sciences GmbH
Publication of CL2020001791A1 publication Critical patent/CL2020001791A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/08Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
    • A61K47/10Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38Cellulose; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/06Ointments; Bases therefor; Other semi-solid forms, e.g. creams, sticks, gels
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/14Drugs for dermatological disorders for baldness or alopecia

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Dermatology (AREA)
  • Inorganic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Se divulgan formas de realización de formulaciones tópicas para administrar cerdulatinib o una sal, hidrato o solvato aceptable desde el punto de vista farmacéutico de este. También se divulgan formas de realización de métodos para preparar las formulaciones tópicas. Las formulaciones divulgadas son adecuadas para el tratamiento de afecciones dermatológicas tales como dermatitis atópica.
CL2020001791A 2018-01-09 2020-07-03 Composiciones farmacéuticas para la piel tópicas que contienen cerdulatinib y usos de estas. CL2020001791A1 (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US201862615261P 2018-01-09 2018-01-09
US201862686509P 2018-06-18 2018-06-18
US201862765133P 2018-08-16 2018-08-16
US201862772415P 2018-11-28 2018-11-28

Publications (1)

Publication Number Publication Date
CL2020001791A1 true CL2020001791A1 (es) 2020-12-04

Family

ID=65685834

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2020001791A CL2020001791A1 (es) 2018-01-09 2020-07-03 Composiciones farmacéuticas para la piel tópicas que contienen cerdulatinib y usos de estas.

Country Status (17)

Country Link
US (1) US20200390689A1 (es)
EP (1) EP3737354A2 (es)
JP (1) JP2021510159A (es)
KR (1) KR20200108297A (es)
CN (1) CN111818910A (es)
AU (1) AU2019208049A1 (es)
BR (1) BR112020013976A2 (es)
CA (1) CA3087124A1 (es)
CL (1) CL2020001791A1 (es)
CO (1) CO2020008244A2 (es)
IL (1) IL275899A (es)
MX (1) MX2020007062A (es)
RU (1) RU2020124293A (es)
SG (1) SG11202005781WA (es)
TW (1) TW201938167A (es)
WO (1) WO2019138291A2 (es)
ZA (1) ZA202004104B (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3810144A4 (en) * 2018-06-04 2022-08-17 Chemistryrx TOPICAL HAIR GROWTH STIMULATING COMPOSITIONS

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2003244098A1 (en) 2002-06-28 2004-01-19 Yamanouchi Pharmaceutical Co., Ltd. Diaminopyrimidinecarboxa mide derivative
US8138339B2 (en) 2008-04-16 2012-03-20 Portola Pharmaceuticals, Inc. Inhibitors of protein kinases
EP2574168B9 (en) * 2010-05-21 2016-10-05 Incyte Holdings Corporation Topical formulation for a jak inhibitor
AU2012241018B2 (en) * 2011-04-08 2015-11-12 Pfizer Inc. Crystalline and non- crystalline forms of tofacitinib, and a pharmaceutical composition comprising tofacitinib and a penetration enhancer
JP6247223B2 (ja) * 2011-12-08 2017-12-13 ライジェル ファーマシューティカルズ, インコーポレイテッド 化合物を投与するための局所用製剤
KR20180002838A (ko) * 2015-05-07 2018-01-08 더 트러스티스 오브 콜롬비아 유니버시티 인 더 시티 오브 뉴욕 모발 생장을 촉진하기 위한 방법 및 조성물
WO2017027829A1 (en) * 2015-08-12 2017-02-16 Portola Pharmaceuticals, Inc. Cerdulatinib for treating myeloma
CN108367006B (zh) * 2015-12-04 2021-12-31 博尔托拉制药公司 用于治疗血液癌症的赛度替尼
BR112018075202A2 (pt) * 2016-06-07 2019-03-19 Dermavant Sciences GmbH formulação tópica e método de tratamento de uma condição dermatológica em um sujeito
US11957931B2 (en) * 2017-04-26 2024-04-16 Yale University Compositions and methods for treating vitiligo

Also Published As

Publication number Publication date
TW201938167A (zh) 2019-10-01
JP2021510159A (ja) 2021-04-15
BR112020013976A2 (pt) 2020-12-08
CO2020008244A2 (es) 2020-10-30
US20200390689A1 (en) 2020-12-17
SG11202005781WA (en) 2020-07-29
AU2019208049A1 (en) 2020-07-23
WO2019138291A3 (en) 2019-08-22
KR20200108297A (ko) 2020-09-17
CN111818910A (zh) 2020-10-23
CA3087124A1 (en) 2019-07-18
MX2020007062A (es) 2021-03-09
IL275899A (en) 2020-08-31
EP3737354A2 (en) 2020-11-18
WO2019138291A2 (en) 2019-07-18
ZA202004104B (en) 2022-01-26
RU2020124293A (ru) 2022-02-10

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