CL2007002511A1 - Compuestos derivados de pirrolo[2,3-f]isoquinolina, inhibidores de cinasa-2; proceso de preparacion; composicion farmaceutica; combinacion farmaceutica; y uso para el tratamiento de una enfermedad autoinmune. - Google Patents
Compuestos derivados de pirrolo[2,3-f]isoquinolina, inhibidores de cinasa-2; proceso de preparacion; composicion farmaceutica; combinacion farmaceutica; y uso para el tratamiento de una enfermedad autoinmune.Info
- Publication number
- CL2007002511A1 CL2007002511A1 CL200702511A CL2007002511A CL2007002511A1 CL 2007002511 A1 CL2007002511 A1 CL 2007002511A1 CL 200702511 A CL200702511 A CL 200702511A CL 2007002511 A CL2007002511 A CL 2007002511A CL 2007002511 A1 CL2007002511 A1 CL 2007002511A1
- Authority
- CL
- Chile
- Prior art keywords
- isoquinolina
- pirrolo
- kinase
- inhibitors
- treatment
- Prior art date
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- A61K31/5365—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines ortho- or peri-condensed with heterocyclic ring systems
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D498/14—Ortho-condensed systems
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
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EP06119817 | 2006-08-30 |
Publications (1)
Publication Number | Publication Date |
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CL2007002511A1 true CL2007002511A1 (es) | 2008-05-16 |
Family
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Family Applications (1)
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CL200702511A CL2007002511A1 (es) | 2006-08-30 | 2007-08-29 | Compuestos derivados de pirrolo[2,3-f]isoquinolina, inhibidores de cinasa-2; proceso de preparacion; composicion farmaceutica; combinacion farmaceutica; y uso para el tratamiento de una enfermedad autoinmune. |
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US (1) | US20100069360A1 (es) |
EP (1) | EP2064212A1 (es) |
JP (1) | JP2010501605A (es) |
KR (1) | KR20090046891A (es) |
CN (1) | CN101506208A (es) |
AR (1) | AR062564A1 (es) |
AU (1) | AU2007291575B2 (es) |
BR (1) | BRPI0716198A2 (es) |
CA (1) | CA2660980A1 (es) |
CL (1) | CL2007002511A1 (es) |
MX (1) | MX2009002278A (es) |
PE (1) | PE20080668A1 (es) |
RU (1) | RU2009111382A (es) |
TW (1) | TW200819449A (es) |
WO (1) | WO2008025512A1 (es) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8299271B2 (en) | 2006-08-30 | 2012-10-30 | Phenomix Corporation | Solid tartrate salts of DPP-IV inhibitors |
Families Citing this family (9)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2009067493A2 (en) * | 2007-11-19 | 2009-05-28 | Envivo Pharmaceuticals, Inc. | 1,3,5 tri-subtituted benzenes for treatment of alzheimer's disease and other disorders |
KR20100135711A (ko) | 2007-12-20 | 2010-12-27 | 엔비보 파마슈티칼즈, 인코퍼레이티드 | 사중치환된 벤젠 |
ES2445896T3 (es) * | 2009-03-20 | 2014-03-05 | Nerviano Medical Sciences S.R.L. | Uso de un inhibidor de quinasa para el tratamiento del timoma |
EP3072555B1 (en) | 2011-09-02 | 2020-03-25 | The Trustees of Columbia University in the City of New York | Mk2/3 inhibitors to treat metabolic disturbances of obesity |
CA2908098A1 (en) | 2013-03-15 | 2014-09-25 | Celgene Avilomics Research, Inc. | Mk2 inhibitors and uses thereof |
US9951026B2 (en) | 2013-09-17 | 2018-04-24 | Pharmakea, Inc. | Heterocyclic vinyl autotaxin inhibitor compounds |
EP3046905A4 (en) | 2013-09-17 | 2017-03-22 | Pharmakea Inc. | Vinyl autotaxin inhibitor compounds |
CN104140393B (zh) * | 2013-12-10 | 2016-09-21 | 郑州泰基鸿诺医药股份有限公司 | 一种芳环/芳杂环叔丁醇酯类化合物的制备方法 |
CN107082780B (zh) * | 2017-04-14 | 2020-08-14 | 山东省医学科学院药物研究所 | 一种具有吡咯骈异喹啉结构的生物碱及其制备方法与应用 |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
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BR0317430A (pt) * | 2002-12-20 | 2005-10-25 | Pharmacia Corp | Compostos inibidores de quinase-2 de proteìna ativada por quinase de proteìna ativada por mitógeno |
US20050143371A1 (en) * | 2003-07-23 | 2005-06-30 | Pharmacia Corporation | Beta-carboline compounds and analogues thereof as mitogen-activated protein kinase-activated protein kinase-2 inhibitors |
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2007
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- 2007-08-28 MX MX2009002278A patent/MX2009002278A/es not_active Application Discontinuation
- 2007-08-28 WO PCT/EP2007/007510 patent/WO2008025512A1/en active Application Filing
- 2007-08-28 RU RU2009111382/04A patent/RU2009111382A/ru not_active Application Discontinuation
- 2007-08-28 US US12/439,603 patent/US20100069360A1/en not_active Abandoned
- 2007-08-28 AR ARP070103811A patent/AR062564A1/es unknown
- 2007-08-28 EP EP07801933A patent/EP2064212A1/en not_active Withdrawn
- 2007-08-28 BR BRPI0716198-0A2A patent/BRPI0716198A2/pt not_active IP Right Cessation
- 2007-08-28 JP JP2009525966A patent/JP2010501605A/ja active Pending
- 2007-08-28 CN CNA2007800310152A patent/CN101506208A/zh active Pending
- 2007-08-28 KR KR1020097004142A patent/KR20090046891A/ko not_active Application Discontinuation
- 2007-08-28 CA CA002660980A patent/CA2660980A1/en not_active Abandoned
- 2007-08-28 AU AU2007291575A patent/AU2007291575B2/en not_active Expired - Fee Related
- 2007-08-29 CL CL200702511A patent/CL2007002511A1/es unknown
- 2007-08-29 TW TW096132111A patent/TW200819449A/zh unknown
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
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US8299271B2 (en) | 2006-08-30 | 2012-10-30 | Phenomix Corporation | Solid tartrate salts of DPP-IV inhibitors |
Also Published As
Publication number | Publication date |
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CN101506208A (zh) | 2009-08-12 |
US20100069360A1 (en) | 2010-03-18 |
AU2007291575B2 (en) | 2011-02-10 |
KR20090046891A (ko) | 2009-05-11 |
AU2007291575A1 (en) | 2008-03-06 |
WO2008025512A1 (en) | 2008-03-06 |
PE20080668A1 (es) | 2008-07-17 |
AR062564A1 (es) | 2008-11-19 |
CA2660980A1 (en) | 2008-03-06 |
RU2009111382A (ru) | 2010-10-10 |
JP2010501605A (ja) | 2010-01-21 |
BRPI0716198A2 (pt) | 2013-11-12 |
EP2064212A1 (en) | 2009-06-03 |
TW200819449A (en) | 2008-05-01 |
MX2009002278A (es) | 2009-03-20 |
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