CL2004001921A1 - Compuestos derivados de pirimidina; composicion que los cintoene utiles como insecticidas y antihelminticos. - Google Patents

Compuestos derivados de pirimidina; composicion que los cintoene utiles como insecticidas y antihelminticos.

Info

Publication number
CL2004001921A1
CL2004001921A1 CL200401921A CL2004001921A CL2004001921A1 CL 2004001921 A1 CL2004001921 A1 CL 2004001921A1 CL 200401921 A CL200401921 A CL 200401921A CL 2004001921 A CL2004001921 A CL 2004001921A CL 2004001921 A1 CL2004001921 A1 CL 2004001921A1
Authority
CL
Chile
Prior art keywords
cintoene
antihelmintics
insecticides
pyrimidine
useful
Prior art date
Application number
CL200401921A
Other languages
English (en)
Inventor
Hyun Lee Martha Jane Lar Byung
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of CL2004001921A1 publication Critical patent/CL2004001921A1/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06Antimalarials
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/10Anthelmintics
    • A61P33/12Schistosomicides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/14Ectoparasiticides, e.g. scabicides
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/50Three nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)
CL200401921A 2003-08-07 2004-07-29 Compuestos derivados de pirimidina; composicion que los cintoene utiles como insecticidas y antihelminticos. CL2004001921A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US49329603P 2003-08-07 2003-08-07

Publications (1)

Publication Number Publication Date
CL2004001921A1 true CL2004001921A1 (es) 2005-06-03

Family

ID=34135225

Family Applications (1)

Application Number Title Priority Date Filing Date
CL200401921A CL2004001921A1 (es) 2003-08-07 2004-07-29 Compuestos derivados de pirimidina; composicion que los cintoene utiles como insecticidas y antihelminticos.

Country Status (9)

Country Link
US (1) US20050032810A1 (es)
EP (1) EP1654249A1 (es)
JP (1) JP2007501781A (es)
AR (1) AR045223A1 (es)
AU (1) AU2004263373A1 (es)
CA (1) CA2534975A1 (es)
CL (1) CL2004001921A1 (es)
TW (1) TW200509794A (es)
WO (1) WO2005014573A1 (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1692939A1 (en) * 2005-02-19 2006-08-23 Bayer CropScience S.A. Pesticidal substituted piperidines
EP1869007A1 (en) * 2005-04-14 2007-12-26 Teva Pharmaceutical Industries Ltd Process for preparing quetiapine fumarate
CN101597278B (zh) 2008-06-04 2013-04-17 中国中化股份有限公司 酰胺类化合物及其制备与应用
JP2014237589A (ja) * 2011-09-28 2014-12-18 日本曹達株式会社 環状アミン化合物および有害生物防除剤
RU2014131951A (ru) * 2012-02-03 2016-03-27 Зоэтис Ллс Производные дигидрофуран азетидина в качестве противопаразитарных агентов
US9357782B2 (en) * 2012-08-08 2016-06-07 Novartis Tiergesundheit Ag Substituted azines as pesticides
CA3138859A1 (en) * 2019-05-02 2020-11-05 Constellation Pharmaceuticals, Inc. Modulators of trex1
US20240132464A1 (en) * 2022-09-28 2024-04-25 Accutar Biotechnology Inc. Heterocyclic compounds as e3 ligase inhibitors

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8929022D0 (en) * 1989-12-22 1990-02-28 Ici Plc Diazine derivatives
EP0506270A1 (en) * 1991-03-28 1992-09-30 Zeneca Limited Nematocide pyrimidine derivatives
GB9219635D0 (en) * 1992-09-16 1992-10-28 Ici Plc Heterocyclic compounds
KR100342275B1 (ko) * 1993-10-21 2002-12-05 지.디. 썰 엘엘씨 산화질소신타제저해제로서유용한아미디노유도체
IL116893A (en) * 1995-02-10 2000-02-29 Yamanouchi Pharma Co Ltd Piperazine derivatives and pharmaceutical compositions containing them
ZA974584B (en) * 1996-06-07 1998-11-26 Upjohn Co Method for discovering novel anthelmintic compounds
FR2783519B1 (fr) * 1998-09-23 2003-01-24 Sod Conseils Rech Applic Nouveaux derives d'amidines, leur preparation, leur application a titre de medicaments et les compositions pharmaceutiques les contenant
EP1437348A1 (fr) * 2003-01-13 2004-07-14 L'oreal Dérivés de de la 6-méthyl-pyrimidine-2,4-diamine, procédé de synthèse, compositions les comprenant et utilisations comme agents neutralisants basiques

Also Published As

Publication number Publication date
CA2534975A1 (en) 2005-02-17
JP2007501781A (ja) 2007-02-01
AU2004263373A1 (en) 2005-02-17
US20050032810A1 (en) 2005-02-10
WO2005014573A1 (en) 2005-02-17
EP1654249A1 (en) 2006-05-10
TW200509794A (en) 2005-03-16
AR045223A1 (es) 2005-10-19

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