AR045223A1 - Compuestos derivados de pirimidina y composiciones antihelminticas e insecticidas que los contienen como principios activos. - Google Patents

Compuestos derivados de pirimidina y composiciones antihelminticas e insecticidas que los contienen como principios activos.

Info

Publication number
AR045223A1
AR045223A1 ARP040102787A ARP040102787A AR045223A1 AR 045223 A1 AR045223 A1 AR 045223A1 AR P040102787 A ARP040102787 A AR P040102787A AR P040102787 A ARP040102787 A AR P040102787A AR 045223 A1 AR045223 A1 AR 045223A1
Authority
AR
Argentina
Prior art keywords
pyrimidine
compounds derived
alkyl
antihelmintic
compositions containing
Prior art date
Application number
ARP040102787A
Other languages
English (en)
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of AR045223A1 publication Critical patent/AR045223A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • A61P33/06—Antimalarials
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A61P33/12—Schistosomicides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/14—Ectoparasiticides, e.g. scabicides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/50—Three nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

Compuestos derivados de pirimidina como ingredientes activos de composiciones antihelmínticas e insecticidas utilizables para el tratamiento de enfermedades parasitarias como así también el control de parásitos en una planta o cosecha agrícola. Reivindicación 1: Un compuesto de fórmula (1) que comprende: en la A y B se seleccionan independientemente del grupo comprendido por H, alquilo C1-6, NRR´, y alcoxi C1-6; X es uno a tres sustituyentes seleccionados del grupo que comprende halógeno, alquilo C1-6, -OH, alcoxi C1-6, tioalcoxi C1-6, -NRR´, -CO2R, -CONRR´, -CN, -NO2 y -SO2NRR´; R y R´ son independientemente H, alquilo C1-6 o, tomados conjuntamente, forman un anillo de 5 a 7 miembros que contiene opcionalmente un heteroátomo adicional de NR, O o S; m es 1 o 2; n es 1, 2 o 3; cuando m y n son 2, Z es -N-, -CH- o -COR-; cuando m es 1 o 2 y n es 1 o 3, Z es -CH- o -COR-.
ARP040102787A 2003-08-07 2004-08-05 Compuestos derivados de pirimidina y composiciones antihelminticas e insecticidas que los contienen como principios activos. AR045223A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US49329603P 2003-08-07 2003-08-07

Publications (1)

Publication Number Publication Date
AR045223A1 true AR045223A1 (es) 2005-10-19

Family

ID=34135225

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP040102787A AR045223A1 (es) 2003-08-07 2004-08-05 Compuestos derivados de pirimidina y composiciones antihelminticas e insecticidas que los contienen como principios activos.

Country Status (9)

Country Link
US (1) US20050032810A1 (es)
EP (1) EP1654249A1 (es)
JP (1) JP2007501781A (es)
AR (1) AR045223A1 (es)
AU (1) AU2004263373A1 (es)
CA (1) CA2534975A1 (es)
CL (1) CL2004001921A1 (es)
TW (1) TW200509794A (es)
WO (1) WO2005014573A1 (es)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1692939A1 (en) * 2005-02-19 2006-08-23 Bayer CropScience S.A. Pesticidal substituted piperidines
EP1869007A1 (en) * 2005-04-14 2007-12-26 Teva Pharmaceutical Industries Ltd Process for preparing quetiapine fumarate
CN101597278B (zh) 2008-06-04 2013-04-17 中国中化股份有限公司 酰胺类化合物及其制备与应用
JP2014237589A (ja) * 2011-09-28 2014-12-18 日本曹達株式会社 環状アミン化合物および有害生物防除剤
PL2814825T3 (pl) * 2012-02-03 2016-08-31 Zoetis Services Llc Dihydrofuranowe pochodne azetydyny jako środki przeciwpasożytnicze
WO2014023723A1 (en) * 2012-08-08 2014-02-13 Novartis Ag Subtituted azines as pesticides
KR20220004671A (ko) * 2019-05-02 2022-01-11 콘스텔레이션 파마슈티칼스, 인크. Trex1의 조절제
WO2024073502A1 (en) * 2022-09-28 2024-04-04 Accutar Biotechnology Inc. Heterocyclic compounds as e3 ligase inhibitors

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8929022D0 (en) * 1989-12-22 1990-02-28 Ici Plc Diazine derivatives
GB9205484D0 (en) * 1991-03-28 1992-04-29 Ici Plc Heterocyclic compounds
GB9219635D0 (en) * 1992-09-16 1992-10-28 Ici Plc Heterocyclic compounds
RU2136661C1 (ru) * 1993-10-21 1999-09-10 Джи Ди Сирл энд Ко. Амидинопроизводные, их применение и фармацевтическая композиция
IL116893A (en) * 1995-02-10 2000-02-29 Yamanouchi Pharma Co Ltd Piperazine derivatives and pharmaceutical compositions containing them
ZA974584B (en) * 1996-06-07 1998-11-26 Upjohn Co Method for discovering novel anthelmintic compounds
FR2783519B1 (fr) * 1998-09-23 2003-01-24 Sod Conseils Rech Applic Nouveaux derives d'amidines, leur preparation, leur application a titre de medicaments et les compositions pharmaceutiques les contenant
EP1437348A1 (fr) * 2003-01-13 2004-07-14 L'oreal Dérivés de de la 6-méthyl-pyrimidine-2,4-diamine, procédé de synthèse, compositions les comprenant et utilisations comme agents neutralisants basiques

Also Published As

Publication number Publication date
JP2007501781A (ja) 2007-02-01
CL2004001921A1 (es) 2005-06-03
TW200509794A (en) 2005-03-16
CA2534975A1 (en) 2005-02-17
US20050032810A1 (en) 2005-02-10
WO2005014573A1 (en) 2005-02-17
EP1654249A1 (en) 2006-05-10
AU2004263373A1 (en) 2005-02-17

Similar Documents

Publication Publication Date Title
AR042984A1 (es) Pirimidinas substituidas
AR031879A1 (es) Un derivado triazolona biciclico y un herbicida conteniendo dicho derivado
AR036047A1 (es) Composicion herbicida selectiva y metodo para controlar selectivamente malezas y pastos en cultivos de plantas utiles
PE20181198A1 (es) Derivados de heterociclos biciclicos condensados como agentes de control de plagas
CO2022005257A2 (es) Compuestos heteroaromáticos bicíclicos condensados activos como pesticidas
EA201071294A1 (ru) Химические соединения
PE20070054A1 (es) Mezclas pesticidas
PE20090189A1 (es) Derivados de aza-piridopirimidinona como agonistas de hm74a
AR083235A1 (es) Derivados de tiazol como pesticidas
CR7920A (es) Amino -1,3,5- triazinas sustituidad en n con radicales biciclicos quirales, procedimiento para su preparacion, composiciones de las mismas y su uso como herbicida y reguladores del crecimiento de las plantas
EA201200442A1 (ru) Гербицидная композиция
ECSP055935A (es) Medicamento para la profilaxis y el tratamiento de arteriosclerosis e hipertension
ECSP10010726A (es) Composición fungicida y
UY30316A1 (es) Derivados sustituidos de benzamidas, nicotinamidas, propanamidas, acetamidas y carboxamidas n-(2-(piperidin-1-ilmetil)ciclohexil)sustituidas, procesos de preparacion, composiciones conteniéndolos y aplicaciones
PE20211275A1 (es) Compuestos heterociclicos antihelminticos
PE20091349A1 (es) Compuestos derivados de espiro 1,3,4-tiadiazol como inhibidores de la actividad quinesina ksp
UY39515A (es) Compuestos herbicidas de n-heteroarilpirazol
UY34476A (es) ?mezclas pesticidas que incluyen pirrolidindionas espiroheterocíclicas?.
UY38575A (es) Compuestos de diona cíclicos activos como herbicidas que comprenden un grupo sulfonimidamida
CL2020002099A1 (es) Compuestos herbicidas de 3-azaspiro (5.5) undecano - 8.10 - diona.
AR045223A1 (es) Compuestos derivados de pirimidina y composiciones antihelminticas e insecticidas que los contienen como principios activos.
CL2020002324A1 (es) Derivados de la ciclohexanediona de espiro como herbicidas.
UY38591A (es) Compuestos de diona cíclica herbicidamente activos que comprenden un grupo oxima o hidrazona.
CL2020003349A1 (es) Derivados heterocíclicos como plaguicidas
AR124173A1 (es) Derivados herbicidas

Legal Events

Date Code Title Description
FB Suspension of granting procedure