AR045223A1 - Compuestos derivados de pirimidina y composiciones antihelminticas e insecticidas que los contienen como principios activos. - Google Patents
Compuestos derivados de pirimidina y composiciones antihelminticas e insecticidas que los contienen como principios activos.Info
- Publication number
- AR045223A1 AR045223A1 ARP040102787A ARP040102787A AR045223A1 AR 045223 A1 AR045223 A1 AR 045223A1 AR P040102787 A ARP040102787 A AR P040102787A AR P040102787 A ARP040102787 A AR P040102787A AR 045223 A1 AR045223 A1 AR 045223A1
- Authority
- AR
- Argentina
- Prior art keywords
- pyrimidine
- compounds derived
- alkyl
- antihelmintic
- compositions containing
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
- A61P33/06—Antimalarials
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
- A61P33/12—Schistosomicides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/14—Ectoparasiticides, e.g. scabicides
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/50—Three nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Tropical Medicine & Parasitology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Abstract
Compuestos derivados de pirimidina como ingredientes activos de composiciones antihelmínticas e insecticidas utilizables para el tratamiento de enfermedades parasitarias como así también el control de parásitos en una planta o cosecha agrícola. Reivindicación 1: Un compuesto de fórmula (1) que comprende: en la A y B se seleccionan independientemente del grupo comprendido por H, alquilo C1-6, NRR´, y alcoxi C1-6; X es uno a tres sustituyentes seleccionados del grupo que comprende halógeno, alquilo C1-6, -OH, alcoxi C1-6, tioalcoxi C1-6, -NRR´, -CO2R, -CONRR´, -CN, -NO2 y -SO2NRR´; R y R´ son independientemente H, alquilo C1-6 o, tomados conjuntamente, forman un anillo de 5 a 7 miembros que contiene opcionalmente un heteroátomo adicional de NR, O o S; m es 1 o 2; n es 1, 2 o 3; cuando m y n son 2, Z es -N-, -CH- o -COR-; cuando m es 1 o 2 y n es 1 o 3, Z es -CH- o -COR-.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US49329603P | 2003-08-07 | 2003-08-07 |
Publications (1)
Publication Number | Publication Date |
---|---|
AR045223A1 true AR045223A1 (es) | 2005-10-19 |
Family
ID=34135225
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
ARP040102787A AR045223A1 (es) | 2003-08-07 | 2004-08-05 | Compuestos derivados de pirimidina y composiciones antihelminticas e insecticidas que los contienen como principios activos. |
Country Status (9)
Country | Link |
---|---|
US (1) | US20050032810A1 (es) |
EP (1) | EP1654249A1 (es) |
JP (1) | JP2007501781A (es) |
AR (1) | AR045223A1 (es) |
AU (1) | AU2004263373A1 (es) |
CA (1) | CA2534975A1 (es) |
CL (1) | CL2004001921A1 (es) |
TW (1) | TW200509794A (es) |
WO (1) | WO2005014573A1 (es) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1692939A1 (en) * | 2005-02-19 | 2006-08-23 | Bayer CropScience S.A. | Pesticidal substituted piperidines |
EP1869007A1 (en) * | 2005-04-14 | 2007-12-26 | Teva Pharmaceutical Industries Ltd | Process for preparing quetiapine fumarate |
CN101597278B (zh) | 2008-06-04 | 2013-04-17 | 中国中化股份有限公司 | 酰胺类化合物及其制备与应用 |
JP2014237589A (ja) * | 2011-09-28 | 2014-12-18 | 日本曹達株式会社 | 環状アミン化合物および有害生物防除剤 |
PL2814825T3 (pl) * | 2012-02-03 | 2016-08-31 | Zoetis Services Llc | Dihydrofuranowe pochodne azetydyny jako środki przeciwpasożytnicze |
WO2014023723A1 (en) * | 2012-08-08 | 2014-02-13 | Novartis Ag | Subtituted azines as pesticides |
KR20220004671A (ko) * | 2019-05-02 | 2022-01-11 | 콘스텔레이션 파마슈티칼스, 인크. | Trex1의 조절제 |
WO2024073502A1 (en) * | 2022-09-28 | 2024-04-04 | Accutar Biotechnology Inc. | Heterocyclic compounds as e3 ligase inhibitors |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8929022D0 (en) * | 1989-12-22 | 1990-02-28 | Ici Plc | Diazine derivatives |
GB9205484D0 (en) * | 1991-03-28 | 1992-04-29 | Ici Plc | Heterocyclic compounds |
GB9219635D0 (en) * | 1992-09-16 | 1992-10-28 | Ici Plc | Heterocyclic compounds |
RU2136661C1 (ru) * | 1993-10-21 | 1999-09-10 | Джи Ди Сирл энд Ко. | Амидинопроизводные, их применение и фармацевтическая композиция |
IL116893A (en) * | 1995-02-10 | 2000-02-29 | Yamanouchi Pharma Co Ltd | Piperazine derivatives and pharmaceutical compositions containing them |
ZA974584B (en) * | 1996-06-07 | 1998-11-26 | Upjohn Co | Method for discovering novel anthelmintic compounds |
FR2783519B1 (fr) * | 1998-09-23 | 2003-01-24 | Sod Conseils Rech Applic | Nouveaux derives d'amidines, leur preparation, leur application a titre de medicaments et les compositions pharmaceutiques les contenant |
EP1437348A1 (fr) * | 2003-01-13 | 2004-07-14 | L'oreal | Dérivés de de la 6-méthyl-pyrimidine-2,4-diamine, procédé de synthèse, compositions les comprenant et utilisations comme agents neutralisants basiques |
-
2004
- 2004-07-26 EP EP04744133A patent/EP1654249A1/en not_active Withdrawn
- 2004-07-26 WO PCT/IB2004/002482 patent/WO2005014573A1/en not_active Application Discontinuation
- 2004-07-26 JP JP2006522428A patent/JP2007501781A/ja not_active Withdrawn
- 2004-07-26 AU AU2004263373A patent/AU2004263373A1/en not_active Abandoned
- 2004-07-26 CA CA002534975A patent/CA2534975A1/en not_active Abandoned
- 2004-07-29 CL CL200401921A patent/CL2004001921A1/es unknown
- 2004-08-05 US US10/912,513 patent/US20050032810A1/en not_active Abandoned
- 2004-08-05 AR ARP040102787A patent/AR045223A1/es unknown
- 2004-08-06 TW TW093123651A patent/TW200509794A/zh unknown
Also Published As
Publication number | Publication date |
---|---|
JP2007501781A (ja) | 2007-02-01 |
CL2004001921A1 (es) | 2005-06-03 |
TW200509794A (en) | 2005-03-16 |
CA2534975A1 (en) | 2005-02-17 |
US20050032810A1 (en) | 2005-02-10 |
WO2005014573A1 (en) | 2005-02-17 |
EP1654249A1 (en) | 2006-05-10 |
AU2004263373A1 (en) | 2005-02-17 |
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Legal Events
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