CH580631A5 - - Google Patents

Info

Publication number
CH580631A5
CH580631A5 CH84871A CH84871A CH580631A5 CH 580631 A5 CH580631 A5 CH 580631A5 CH 84871 A CH84871 A CH 84871A CH 84871 A CH84871 A CH 84871A CH 580631 A5 CH580631 A5 CH 580631A5
Authority
CH
Switzerland
Application number
CH84871A
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Priority to CH84871A priority Critical patent/CH580631A5/xx
Priority to DE19712163600 priority patent/DE2163600A1/de
Priority to ZA718537A priority patent/ZA718537B/xx
Priority to AU37353/71A priority patent/AU460825B2/en
Priority to IL38467A priority patent/IL38467A/xx
Priority to CA131,224A priority patent/CA959834A/en
Priority to US00215187A priority patent/US3839322A/en
Priority to NL7200515A priority patent/NL7200515A/xx
Priority to IS2050A priority patent/IS2050A7/is
Priority to HUHO1449A priority patent/HU162984B/hu
Priority to RO7269395A priority patent/RO70672A/fr
Priority to IE62/72A priority patent/IE35985B1/xx
Priority to IE2001/73*A priority patent/IE35986B1/xx
Priority to PH13213*UA priority patent/PH9500A/en
Priority to SE7200544A priority patent/SE396608B/xx
Priority to OA54470A priority patent/OA03944A/fr
Priority to LU64606A priority patent/LU64606A1/xx
Priority to FI110/72A priority patent/FI55513C/fi
Priority to JP700272A priority patent/JPS551270B1/ja
Priority to ES399014A priority patent/ES399014A1/es
Priority to DK27072AA priority patent/DK141966B/da
Priority to AT42072A priority patent/AT318140B/de
Priority to BG19517A priority patent/BG18851A3/xx
Priority to BR000305/72A priority patent/BR7200305D0/pt
Priority to BE778213A priority patent/BE778213A/fr
Priority to SU7201739249A priority patent/SU583759A3/ru
Priority to PL1972153004A priority patent/PL89650B1/pl
Priority to CS398A priority patent/CS175424B2/cs
Priority to GB282572A priority patent/GB1334035A/en
Priority to GB384873A priority patent/GB1334036A/en
Priority to FR7201882A priority patent/FR2122546B1/fr
Priority to DO1972001956A priority patent/DOP1972001956A/es
Priority to ES404014A priority patent/ES404014A1/es
Priority to SE7411317A priority patent/SE419082B/xx
Priority to MY191/74A priority patent/MY7400191A/xx
Priority to US05/619,128 priority patent/USRE29003E/en
Priority to SE7513806A priority patent/SE7513806L/xx
Publication of CH580631A5 publication Critical patent/CH580631A5/xx
Priority to NO763546A priority patent/NO763546L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24—Oxygen or sulfur atoms
    • C07D207/26—2-Pyrrolidones
    • C07D207/273—2-Pyrrolidones with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to other ring carbon atoms
    • C07D207/277—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D207/28—2-Pyrrolidone-5- carboxylic acids; Functional derivatives thereof, e.g. esters, nitriles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/78—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C07D213/79—Acids; Esters
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/89—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/50—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D217/00—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems
    • C07D217/22—Heterocyclic compounds containing isoquinoline or hydrogenated isoquinoline ring systems with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to carbon atoms of the nitrogen-containing ring
    • C07D217/26—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C07D239/54—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals
    • C07D239/545—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/557—Two oxygen atoms as doubly bound oxygen atoms or as unsubstituted hydroxy radicals with other hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms, e.g. orotic acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
    • C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D261/18—Carbon atoms having three bonds to hetero atoms, with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/06—1,2,3-Thiadiazoles; Hydrogenated 1,2,3-thiadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/68—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/02—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • C07D309/08—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/10—Oxygen atoms
    • C07D309/12—Oxygen atoms only hydrogen atoms and one oxygen atom directly attached to ring carbon atoms, e.g. tetrahydropyranyl ethers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/38—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
CH84871A 1971-01-20 1971-01-20 CH580631A5 (fr)

Priority Applications (38)

Application Number Priority Date Filing Date Title
CH84871A CH580631A5 (fr) 1971-01-20 1971-01-20
DE19712163600 DE2163600A1 (de) 1971-01-20 1971-12-21 Acylderivate
ZA718537A ZA718537B (en) 1971-01-20 1971-12-21 Acyl derivatives
AU37353/71A AU460825B2 (en) 1971-01-20 1971-12-24 Acyl derivatives
IL38467A IL38467A (en) 1971-01-20 1971-12-27 Heterocyclylcarbonyloxyalkyl carboxylic acids,heterocyclylcarbonyloxyalkyl penicillins,their manufacture and pharmaceutical compositions containing said penicillins
CA131,224A CA959834A (en) 1971-01-20 1971-12-29 Novel penicillins
US00215187A US3839322A (en) 1971-01-20 1972-01-03 (r)-1-(2-furoyloxy)-3-methylbutyl-pencillin compounds
NL7200515A NL7200515A (fr) 1971-01-20 1972-01-13
IS2050A IS2050A7 (is) 1971-01-20 1972-01-13 Efni afleidd úr acyli og aðferð til að framleiða þau.
HUHO1449A HU162984B (fr) 1971-01-20 1972-01-13
RO7269395A RO70672A (fr) 1971-01-20 1972-01-14 Procede pour la preparation des derives de l'acide 6-aminopenicillanique
IE62/72A IE35985B1 (en) 1971-01-20 1972-01-17 6-aminopenicillanic acid derivatives and a process for the manufacture thereof
IE2001/73*A IE35986B1 (en) 1971-01-20 1972-01-17 Carboxylic acids and a process for the preparation thereof
PH13213*UA PH9500A (en) 1971-01-20 1972-01-18 6-amino-penicillanic acid derivatives
SE7200544A SE396608B (sv) 1971-01-20 1972-01-18 Sett att framstella nya penicilliner
OA54470A OA03944A (fr) 1971-01-20 1972-01-18 Dérivés acylés et leur procédé de préparation.
LU64606A LU64606A1 (fr) 1971-01-20 1972-01-18
FI110/72A FI55513C (fi) 1971-01-20 1972-01-18 Foerfarande foer framstaellning av terapeutiskt anvaendbara alfa-acyloxialkylpenicilliner
ES399014A ES399014A1 (es) 1971-01-20 1972-01-19 Procedimiento para la preparacion de derivados de acido 6-amino-penicilanico.
JP700272A JPS551270B1 (fr) 1971-01-20 1972-01-19
DK27072AA DK141966B (da) 1971-01-20 1972-01-19 Analogifremgangsmåde til fremstilling af penicillinforbindelser eller salte eller hydratiserede former deraf.
AT42072A AT318140B (de) 1971-01-20 1972-01-19 Verfahren zur Herstellung von neuen Penicillinen
BG19517A BG18851A3 (fr) 1971-01-20 1972-01-19
BR000305/72A BR7200305D0 (pt) 1971-01-20 1972-01-19 Processo para preparacao de novos derivados de acido 6'-a-mino-penicilanico
BE778213A BE778213A (fr) 1971-01-20 1972-01-19 Derives acyles
SU7201739249A SU583759A3 (ru) 1971-01-20 1972-01-19 Способ получени пенициллинов или их солей или гидратированных форм
GB384873A GB1334036A (en) 1971-01-20 1972-01-20 Carboxylic acids and a process for the preparation thereof
CS398A CS175424B2 (fr) 1971-01-20 1972-01-20
GB282572A GB1334035A (en) 1971-01-20 1972-01-20 6-aminopenicillanic acid derivatives and a process for the manufacture thereof
PL1972153004A PL89650B1 (fr) 1971-01-20 1972-01-20
FR7201882A FR2122546B1 (fr) 1971-01-20 1972-01-20
DO1972001956A DOP1972001956A (es) 1971-01-20 1972-01-24 Derivados de acilo.
ES404014A ES404014A1 (es) 1971-01-20 1972-06-19 Procedimiento para la preparacion de acidos carboniloxicar-boxilicos sustituidos.
SE7411317A SE419082B (sv) 1971-01-20 1974-09-06 Acyloxialkylkarboxylsyror till anvendning for framstellning av alfa-acyloxialkyl-penicilliner
MY191/74A MY7400191A (en) 1971-01-20 1974-12-30 6-amino penicillanic and derivatives and a process for the manufacture thereof
US05/619,128 USRE29003E (en) 1971-01-20 1975-10-02 (R)-1-(2-furoyloxy)-3-methylbutyl-penicillin
SE7513806A SE7513806L (sv) 1971-01-20 1975-12-08 Acylderivat
NO763546A NO763546L (fr) 1971-01-20 1976-10-18

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH84871A CH580631A5 (fr) 1971-01-20 1971-01-20

Publications (1)

Publication Number Publication Date
CH580631A5 true CH580631A5 (fr) 1976-10-15

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Application Number Title Priority Date Filing Date
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Country Status (31)

Country Link
US (1) US3839322A (fr)
JP (1) JPS551270B1 (fr)
AT (1) AT318140B (fr)
AU (1) AU460825B2 (fr)
BE (1) BE778213A (fr)
BG (1) BG18851A3 (fr)
BR (1) BR7200305D0 (fr)
CA (1) CA959834A (fr)
CH (1) CH580631A5 (fr)
CS (1) CS175424B2 (fr)
DE (1) DE2163600A1 (fr)
DK (1) DK141966B (fr)
DO (1) DOP1972001956A (fr)
ES (2) ES399014A1 (fr)
FI (1) FI55513C (fr)
FR (1) FR2122546B1 (fr)
GB (2) GB1334035A (fr)
HU (1) HU162984B (fr)
IE (2) IE35986B1 (fr)
IL (1) IL38467A (fr)
IS (1) IS2050A7 (fr)
LU (1) LU64606A1 (fr)
MY (1) MY7400191A (fr)
NL (1) NL7200515A (fr)
OA (1) OA03944A (fr)
PH (1) PH9500A (fr)
PL (1) PL89650B1 (fr)
RO (1) RO70672A (fr)
SE (3) SE396608B (fr)
SU (1) SU583759A3 (fr)
ZA (1) ZA718537B (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3957758A (en) * 1972-01-03 1976-05-18 Hoffmann-La Roche Inc. 6-acyl derivatives of aminopenicillanic acid
GB8421112D0 (en) * 1984-08-20 1984-09-26 Unilever Plc Pyroglutamic acid esters
US5190980A (en) * 1984-08-20 1993-03-02 Lever Brothers Company, Division Of Conopco, Inc. Pyroglutamic acid esters, their synthesis and use in topical products
IL83978A (en) * 1986-09-26 1992-05-25 Ciba Geigy Process and compositions containing dihalopyridine derivatives for protecting plants against diseases,certain such novel derivatives and their preparation
DE4221605A1 (de) * 1992-07-01 1994-01-05 Basf Ag Verfahren zur Herstellung von 7,16-Dichlor-dianthrachinon-N,N'-dihydroazin

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1125557A (en) * 1966-05-13 1968-08-28 Beecham Group Ltd Penicillins

Also Published As

Publication number Publication date
ES399014A1 (es) 1974-11-01
AU3735371A (en) 1973-06-28
AU460825B2 (en) 1975-05-08
US3839322A (en) 1974-10-01
SU583759A3 (ru) 1977-12-05
SE7513806L (sv) 1975-12-08
BG18851A3 (fr) 1975-03-20
BE778213A (fr) 1972-07-19
PL89650B1 (fr) 1976-12-31
HU162984B (fr) 1973-05-28
GB1334036A (en) 1973-10-17
FI55513B (fi) 1979-04-30
BR7200305D0 (pt) 1973-12-18
SE7411317L (fr) 1974-09-06
JPS551270B1 (fr) 1980-01-12
NL7200515A (fr) 1972-07-24
FR2122546B1 (fr) 1975-06-13
IS2050A7 (is) 1972-02-16
CS175424B2 (fr) 1977-05-31
PH9500A (en) 1976-01-09
FR2122546A1 (fr) 1972-09-01
LU64606A1 (fr) 1973-08-03
SE419082B (sv) 1981-07-13
OA03944A (fr) 1975-08-14
DK141966C (fr) 1981-01-26
AT318140B (de) 1974-09-25
CA959834A (en) 1974-12-24
ZA718537B (en) 1972-09-27
IL38467A (en) 1975-12-31
FI55513C (fi) 1979-08-10
RO70672A (fr) 1982-08-17
IE35985B1 (en) 1976-07-21
DE2163600A1 (de) 1972-08-17
IE35985L (en) 1972-07-20
MY7400191A (en) 1974-12-31
ES404014A1 (es) 1975-05-16
IE35986B1 (en) 1976-07-21
IL38467A0 (en) 1972-02-29
DK141966B (da) 1980-07-28
GB1334035A (en) 1973-10-17
SE396608B (sv) 1977-09-26
DOP1972001956A (es) 1977-01-27

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