CH459239A - Verfahren zur Herstellung von Benzodiazepin-Derivaten - Google Patents
Verfahren zur Herstellung von Benzodiazepin-DerivatenInfo
- Publication number
- CH459239A CH459239A CH551966A CH551966A CH459239A CH 459239 A CH459239 A CH 459239A CH 551966 A CH551966 A CH 551966A CH 551966 A CH551966 A CH 551966A CH 459239 A CH459239 A CH 459239A
- Authority
- CH
- Switzerland
- Prior art keywords
- preparation
- benzodiazepine derivatives
- benzodiazepine
- derivatives
- Prior art date
Links
- 229940053197 benzodiazepine derivative antiepileptics Drugs 0.000 title 1
- 125000003310 benzodiazepinyl group Chemical class N1N=C(C=CC2=C1C=CC=C2)* 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
- C07D243/24—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
- C07D243/24—Oxygen atoms
- C07D243/28—Preparation including building-up the benzodiazepine skeleton from compounds containing no hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US9666361A | 1961-03-20 | 1961-03-20 | |
| US114038A US3153082A (en) | 1961-06-01 | 1961-06-01 | 2-amino-benzophenones |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CH459239A true CH459239A (de) | 1968-07-15 |
Family
ID=26791934
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CH288462A CH445500A (de) | 1961-03-20 | 1962-03-09 | Verfahren zur Herstellung von Benzodiazepin-Derivaten |
| CH551966A CH459239A (de) | 1961-03-20 | 1962-03-09 | Verfahren zur Herstellung von Benzodiazepin-Derivaten |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CH288462A CH445500A (de) | 1961-03-20 | 1962-03-09 | Verfahren zur Herstellung von Benzodiazepin-Derivaten |
Country Status (5)
| Country | Link |
|---|---|
| BE (1) | BE615194A (de) |
| CH (2) | CH445500A (de) |
| ES (1) | ES275601A1 (de) |
| GB (2) | GB985658A (de) |
| SE (1) | SE301974B (de) |
-
1962
- 1962-03-09 CH CH288462A patent/CH445500A/de unknown
- 1962-03-09 CH CH551966A patent/CH459239A/de unknown
- 1962-03-16 GB GB1281964A patent/GB985658A/en not_active Expired
- 1962-03-16 GB GB1012062A patent/GB985657A/en not_active Expired
- 1962-03-16 BE BE615194A patent/BE615194A/fr unknown
- 1962-03-17 ES ES275601A patent/ES275601A1/es not_active Expired
- 1962-03-19 SE SE303062A patent/SE301974B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| GB985657A (en) | 1965-03-10 |
| CH445500A (de) | 1967-10-31 |
| GB985658A (en) | 1965-03-10 |
| DE1445858B2 (de) | 1975-07-03 |
| BE615194A (fr) | 1962-09-17 |
| SE301974B (de) | 1968-07-01 |
| ES275601A1 (es) | 1962-09-16 |
| DE1445858A1 (de) | 1969-01-16 |
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