CH441342A - Verfahren zur Herstellung von Benzodiazepin-Derivaten - Google Patents

Verfahren zur Herstellung von Benzodiazepin-Derivaten

Info

Publication number
CH441342A
CH441342A CH175363A CH175363A CH441342A CH 441342 A CH441342 A CH 441342A CH 175363 A CH175363 A CH 175363A CH 175363 A CH175363 A CH 175363A CH 441342 A CH441342 A CH 441342A
Authority
CH
Switzerland
Prior art keywords
preparation
benzodiazepine derivatives
benzodiazepine
derivatives
Prior art date
Application number
CH175363A
Other languages
English (en)
Inventor
Keller Oscar
Steiger Norbert
Henryk Sternbach Leo
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of CH441342A publication Critical patent/CH441342A/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D243/00Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/141,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/161,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
    • C07D243/181,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
    • C07D243/24Oxygen atoms
    • C07D243/28Preparation including building-up the benzodiazepine skeleton from compounds containing no hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CH175363A 1962-03-21 1963-02-12 Verfahren zur Herstellung von Benzodiazepin-Derivaten CH441342A (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US18144062A 1962-03-21 1962-03-21

Publications (1)

Publication Number Publication Date
CH441342A true CH441342A (de) 1967-08-15

Family

ID=22664289

Family Applications (3)

Application Number Title Priority Date Filing Date
CH175363A CH441342A (de) 1962-03-21 1963-02-12 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH1719666A CH455814A (de) 1962-03-21 1963-02-12 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH1719566A CH454888A (de) 1962-03-21 1963-02-12 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Family Applications After (2)

Application Number Title Priority Date Filing Date
CH1719666A CH455814A (de) 1962-03-21 1963-02-12 Verfahren zur Herstellung von Benzodiazepin-Derivaten
CH1719566A CH454888A (de) 1962-03-21 1963-02-12 Verfahren zur Herstellung von Benzodiazepin-Derivaten

Country Status (7)

Country Link
BR (1) BR6347165D0 (de)
CH (3) CH441342A (de)
DE (1) DE1445872A1 (de)
DK (1) DK107100C (de)
ES (1) ES286241A1 (de)
GB (1) GB1039372A (de)
SE (1) SE312808B (de)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2529203A1 (fr) * 1982-06-24 1983-12-30 Fabre Sa Pierre Procede industriel d'obtention et de purification de flunitrazepam de qualite pharmaceutique

Also Published As

Publication number Publication date
DE1445872A1 (de) 1969-04-10
CH455814A (de) 1968-05-15
SE312808B (de) 1969-07-28
ES286241A1 (es) 1963-11-16
CH454888A (de) 1968-04-30
DK107100C (da) 1967-04-24
BR6347165D0 (pt) 1973-07-19
GB1039372A (en) 1966-08-17

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