CA3063322A1 - Enhanced solubility drug-containing formulations - Google Patents
Enhanced solubility drug-containing formulations Download PDFInfo
- Publication number
- CA3063322A1 CA3063322A1 CA3063322A CA3063322A CA3063322A1 CA 3063322 A1 CA3063322 A1 CA 3063322A1 CA 3063322 A CA3063322 A CA 3063322A CA 3063322 A CA3063322 A CA 3063322A CA 3063322 A1 CA3063322 A1 CA 3063322A1
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/12—Carboxylic acids; Salts or anhydrides thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/02—Inorganic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P23/00—Anaesthetics
- A61P23/02—Local anaesthetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Anesthesiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Inorganic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201762504546P | 2017-05-11 | 2017-05-11 | |
| US62/504,546 | 2017-05-11 | ||
| PCT/IL2018/050511 WO2018207188A1 (en) | 2017-05-11 | 2018-05-10 | Enhanced solubility drug-containing formulations |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA3063322A1 true CA3063322A1 (en) | 2018-11-15 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA3063322A Pending CA3063322A1 (en) | 2017-05-11 | 2018-05-10 | Enhanced solubility drug-containing formulations |
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|---|---|
| US (1) | US11672863B2 (enExample) |
| EP (1) | EP3621591A1 (enExample) |
| JP (1) | JP2020519593A (enExample) |
| KR (1) | KR20200018438A (enExample) |
| CN (1) | CN110869000A (enExample) |
| AU (1) | AU2018265624A1 (enExample) |
| CA (1) | CA3063322A1 (enExample) |
| IL (1) | IL271673A (enExample) |
| WO (1) | WO2018207188A1 (enExample) |
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| KR20200018438A (ko) | 2017-05-11 | 2020-02-19 | 스테디메드 리미티드 | 향상된 용해도의 약물-함유 제형 |
| JP7190077B2 (ja) * | 2019-08-01 | 2022-12-14 | インカーダ セラピューティクス， インコーポレイテッド | 抗不整脈製剤 |
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| US3910260A (en) | 1972-03-01 | 1975-10-07 | Survival Technology | Method and apparatus of treating heart attack patients prior to the establishment of qualified direct contact personal care |
| US4004577A (en) | 1972-12-04 | 1977-01-25 | Survival Technology, Inc. | Method of treating heart attack patients prior to the establishment of qualified direct contact personal care |
| US3941130A (en) | 1975-03-18 | 1976-03-02 | Tibbs Robert C | Sequential trigger release for injection device |
| US4261358A (en) | 1979-10-01 | 1981-04-14 | Walter Vargas | Automatic syringe plunger |
| US4795433A (en) | 1985-05-20 | 1989-01-03 | Survival Technology, Inc. | Automatic injector for emergency treatment |
| US4689042A (en) | 1985-05-20 | 1987-08-25 | Survival Technology, Inc. | Automatic medicament ingredient mixing and injecting apparatus |
| US4902692A (en) * | 1988-03-18 | 1990-02-20 | Iolab Corporation | Method and composition for ophthalmic anesthesia using rodocaine |
| US5085642A (en) | 1989-07-17 | 1992-02-04 | Survival Technology, Inc. | Conveniently carried frequent use autoinjector |
| US5102393A (en) | 1989-07-17 | 1992-04-07 | Survival Technology, Inc. | Autoinjector converted from intramuscular to subcutaneous mode of injection |
| US5092843A (en) | 1990-04-12 | 1992-03-03 | Survival Technology, Inc. | Dispersion multichamber auto-injector |
| US5267963A (en) | 1992-08-21 | 1993-12-07 | Nicholas Bachynsky | Medication injection device |
| US5922340A (en) * | 1992-09-10 | 1999-07-13 | Children's Medical Center Corporation | High load formulations and methods for providing prolonged local anesthesia |
| US5618563A (en) * | 1992-09-10 | 1997-04-08 | Children's Medical Center Corporation | Biodegradable polymer matrices for sustained delivery of local anesthetic agents |
| US5705190A (en) * | 1995-12-19 | 1998-01-06 | Abbott Laboratories | Controlled release formulation for poorly soluble basic drugs |
| US5747060A (en) * | 1996-03-26 | 1998-05-05 | Euro-Celtique, S.A. | Prolonged local anesthesia with colchicine |
| EP1014946B1 (en) * | 1997-09-18 | 2010-04-07 | Pacira Pharmaceuticals, Inc. | Sustained-release liposomal anesthetic compositions |
| US6149626A (en) | 1997-10-03 | 2000-11-21 | Bachynsky; Nicholas | Automatic injecting syringe apparatus |
| SE9803662D0 (sv) | 1998-10-26 | 1998-10-26 | Pharmacia & Upjohn Ab | Autoinjector |
| JP4775807B2 (ja) * | 2004-12-02 | 2011-09-21 | 株式会社 メドレックス | 局所麻酔薬物含有ゼリー剤 |
| US20060270708A1 (en) * | 2005-05-25 | 2006-11-30 | Navinta Llc | Novel process for preparation of isotonic aqueous injection of ropivacaine |
| JP5535623B2 (ja) | 2006-06-30 | 2014-07-02 | アッヴィ バイオテクノロジー リミテッド | 自動注射装置 |
| CN101744760A (zh) * | 2008-12-18 | 2010-06-23 | 梁颖 | 用于难溶性或易分解性药物的缓释体 |
| CN102106806B (zh) * | 2009-12-29 | 2013-04-17 | 上海中西制药有限公司 | 一种固体制剂的制备方法及所得固体制剂 |
| EP3169316A4 (en) * | 2014-07-15 | 2018-01-24 | Isa Odidi | Compositions and methods for reducing overdose |
| AU2016352007B2 (en) * | 2015-11-12 | 2022-03-17 | Terumo Kabushiki Kaisha | Sustained-release topically administered agent |
| KR20200018438A (ko) | 2017-05-11 | 2020-02-19 | 스테디메드 리미티드 | 향상된 용해도의 약물-함유 제형 |
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2018
- 2018-05-10 KR KR1020197036432A patent/KR20200018438A/ko not_active Ceased
- 2018-05-10 US US16/609,544 patent/US11672863B2/en active Active
- 2018-05-10 WO PCT/IL2018/050511 patent/WO2018207188A1/en not_active Ceased
- 2018-05-10 CN CN201880036754.9A patent/CN110869000A/zh active Pending
- 2018-05-10 JP JP2019561320A patent/JP2020519593A/ja active Pending
- 2018-05-10 EP EP18731194.9A patent/EP3621591A1/en not_active Withdrawn
- 2018-05-10 CA CA3063322A patent/CA3063322A1/en active Pending
- 2018-05-10 AU AU2018265624A patent/AU2018265624A1/en not_active Abandoned
-
2019
- 2019-12-23 IL IL271673A patent/IL271673A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL271673A (en) | 2020-02-27 |
| JP2020519593A (ja) | 2020-07-02 |
| US11672863B2 (en) | 2023-06-13 |
| EP3621591A1 (en) | 2020-03-18 |
| KR20200018438A (ko) | 2020-02-19 |
| US20200054754A1 (en) | 2020-02-20 |
| CN110869000A (zh) | 2020-03-06 |
| AU2018265624A1 (en) | 2019-12-05 |
| WO2018207188A1 (en) | 2018-11-15 |
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