CA3043396A1 - Compounds and pharmaceutical compositions thereof for the treatment of inflammatory diseases - Google Patents
Compounds and pharmaceutical compositions thereof for the treatment of inflammatory diseases Download PDFInfo
- Publication number
- CA3043396A1 CA3043396A1 CA3043396A CA3043396A CA3043396A1 CA 3043396 A1 CA3043396 A1 CA 3043396A1 CA 3043396 A CA3043396 A CA 3043396A CA 3043396 A CA3043396 A CA 3043396A CA 3043396 A1 CA3043396 A1 CA 3043396A1
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- Prior art keywords
- compound
- pharmaceutically acceptable
- acceptable salt
- pharmaceutical composition
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Classifications
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- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/541—Non-condensed thiazines containing further heterocyclic rings
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
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- Neurosurgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Pulmonology (AREA)
- Gastroenterology & Hepatology (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Applications Claiming Priority (13)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB1618961.5 | 2016-11-10 | ||
| GB1618963.1 | 2016-11-10 | ||
| GB201618959 | 2016-11-10 | ||
| GB1618959.9 | 2016-11-10 | ||
| GB201618961 | 2016-11-10 | ||
| GB201618962 | 2016-11-10 | ||
| GB1618964.9 | 2016-11-10 | ||
| GB1618960.7 | 2016-11-10 | ||
| GB201618960 | 2016-11-10 | ||
| GB1618962.3 | 2016-11-10 | ||
| GB201618963 | 2016-11-10 | ||
| GB201618964 | 2016-11-10 | ||
| PCT/EP2017/078701 WO2018087202A1 (en) | 2016-11-10 | 2017-11-09 | Compounds and pharmaceutical compositions thereof for the treatment of inflammatory diseases |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA3043396A1 true CA3043396A1 (en) | 2018-05-17 |
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|---|---|---|---|
| CA3043396A Abandoned CA3043396A1 (en) | 2016-11-10 | 2017-11-09 | Compounds and pharmaceutical compositions thereof for the treatment of inflammatory diseases |
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| US (1) | US20190314382A1 (enExample) |
| EP (1) | EP3538103A1 (enExample) |
| JP (1) | JP2019534304A (enExample) |
| AU (1) | AU2017358703A1 (enExample) |
| CA (1) | CA3043396A1 (enExample) |
| RU (1) | RU2019117562A (enExample) |
| TW (1) | TW201821080A (enExample) |
| WO (1) | WO2018087202A1 (enExample) |
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| WO2019132654A1 (en) * | 2017-12-27 | 2019-07-04 | Erasmus University Medical Center Rotterdam | Methods of treating sarcoidosis |
| US12171764B2 (en) | 2018-06-20 | 2024-12-24 | Biora Therapeutics, Inc. | Treatment of a disease of the gastrointestinal tract with a JAK or other kinase inhibitor |
| WO2020009566A1 (en) * | 2018-07-04 | 2020-01-09 | Erasmus University Medical Center Rotterdam | Methods of treating sarcoidosis |
| EP3941474A2 (en) | 2019-03-19 | 2022-01-26 | Incyte Corporation | Biomarkers for vitiligo |
| MA56215A (fr) | 2019-06-10 | 2022-04-20 | Incyte Corp | Traitement topique du vitiligo par un inhibiteur de jak |
| JP7518900B2 (ja) * | 2019-10-16 | 2024-07-18 | インサイト・コーポレイション | 皮膚エリテマトーデス及び扁平苔癬（ｌｐ）の治療のためのｊａｋ１阻害剤の使用 |
| US11992490B2 (en) | 2019-10-16 | 2024-05-28 | Incyte Corporation | Use of JAK1 inhibitors for the treatment of cutaneous lupus erythematosus and Lichen planus (LP) |
| CN115282168B (zh) * | 2022-08-30 | 2024-05-31 | 马应龙大健康有限公司 | 一种缓解婴幼儿湿疹症状的舒缓润肤霜及其制备方法和应用 |
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| WO2005002623A1 (ja) | 2003-07-03 | 2005-01-13 | Japan Science And Technology Agency | サルコイドーシスの治療薬と治療方法 |
| TWI462920B (zh) | 2009-06-26 | 2014-12-01 | 葛萊伯格有限公司 | 用於治療退化性及發炎疾病之新穎化合物 |
| HUE040127T2 (hu) * | 2012-03-29 | 2019-02-28 | Univ Columbia | Eljárások hajhullási rendellenességek kezelésére |
| UY34855A (es) | 2012-06-22 | 2014-01-31 | Galapagos Nv | Aminotriazolopiridina para usar el tratamiento de la inflamación y composiciones farmacéuticas de ella. |
| CA2926361A1 (en) * | 2013-10-24 | 2015-04-30 | Abbvie Inc. | Jak1 selective inhibitor and uses thereof |
| GB201402071D0 (en) | 2014-02-07 | 2014-03-26 | Galapagos Nv | Novel salts and pharmaceutical compositions thereof for the treatment of inflammatory disorders |
| GB201402070D0 (en) | 2014-02-07 | 2014-03-26 | Galapagos Nv | Pharmaceutical compositions for the treatment of inflammatory disorders |
| WO2016165953A1 (en) | 2015-04-13 | 2016-10-20 | Galapagos Nv | Methods for the treatment of inflammatory disorders |
| WO2016165952A1 (en) | 2015-04-13 | 2016-10-20 | Galapagos Nv | Methods for the treatment of cardiovascular disorders |
| AU2016259023A1 (en) * | 2015-05-07 | 2017-11-30 | The Trustees Of Columbia University In The City Of New York | Methods and compositions for promoting hair growth |
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2017
- 2017-11-09 CA CA3043396A patent/CA3043396A1/en not_active Abandoned
- 2017-11-09 WO PCT/EP2017/078701 patent/WO2018087202A1/en not_active Ceased
- 2017-11-09 US US16/348,799 patent/US20190314382A1/en not_active Abandoned
- 2017-11-09 JP JP2019524273A patent/JP2019534304A/ja not_active Withdrawn
- 2017-11-09 AU AU2017358703A patent/AU2017358703A1/en not_active Abandoned
- 2017-11-09 EP EP17800795.1A patent/EP3538103A1/en not_active Withdrawn
- 2017-11-09 RU RU2019117562A patent/RU2019117562A/ru not_active Application Discontinuation
- 2017-11-10 TW TW106139074A patent/TW201821080A/zh unknown
Also Published As
| Publication number | Publication date |
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| RU2019117562A3 (enExample) | 2021-02-09 |
| US20190314382A1 (en) | 2019-10-17 |
| JP2019534304A (ja) | 2019-11-28 |
| RU2019117562A (ru) | 2020-12-10 |
| WO2018087202A1 (en) | 2018-05-17 |
| TW201821080A (zh) | 2018-06-16 |
| EP3538103A1 (en) | 2019-09-18 |
| AU2017358703A1 (en) | 2019-05-09 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Discontinued |
Effective date: 20230509 |