CA3042877A1 - Tricyclic sulfones as ror gamma modulators - Google Patents

Tricyclic sulfones as ror gamma modulators Download PDF

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Publication number
CA3042877A1
CA3042877A1 CA3042877A CA3042877A CA3042877A1 CA 3042877 A1 CA3042877 A1 CA 3042877A1 CA 3042877 A CA3042877 A CA 3042877A CA 3042877 A CA3042877 A CA 3042877A CA 3042877 A1 CA3042877 A1 CA 3042877A1
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Prior art keywords
substituted
alkyl
cr1b
independently
hydrogen
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CA3042877A
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English (en)
French (fr)
Inventor
David MARCOUX
Myra Beaudoin Bertrand
T.G. Murali Dhar
Michael G. Yang
Zili Xiao
Hai-Yun Xiao
Yeheng Zhu
Carolyn A. WEIGELT
Douglas G. Batt
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Bristol Myers Squibb Co
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Bristol Myers Squibb Co
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Publication of CA3042877A1 publication Critical patent/CA3042877A1/en
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    • C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07C2603/06—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
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    • C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/06—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
    • C07C2603/12—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
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AU2017356911A1 (en) 2019-06-20
EP3541786A1 (en) 2019-09-25
KR102599437B1 (ko) 2023-11-07
EA201991128A1 (ru) 2019-10-31
US20180127368A1 (en) 2018-05-10
CN110278711A (zh) 2019-09-24
KR20190084270A (ko) 2019-07-16
IL266474A (en) 2019-07-31
MX2019005384A (es) 2019-08-12
EP3541786B1 (en) 2020-08-05
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US10435369B2 (en) 2019-10-08

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