CA2797560A1 - Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives for the treatment of males - Google Patents
Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives for the treatment of males Download PDFInfo
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- CA2797560A1 CA2797560A1 CA2797560A CA2797560A CA2797560A1 CA 2797560 A1 CA2797560 A1 CA 2797560A1 CA 2797560 A CA2797560 A CA 2797560A CA 2797560 A CA2797560 A CA 2797560A CA 2797560 A1 CA2797560 A1 CA 2797560A1
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- balsalazide
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- therapeutically effective
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Classifications
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/655—Azo (—N=N—), diazo (=N2), azoxy (>N—O—N< or N(=O)—N<), azido (—N3) or diazoamino (—N=N—N<) compounds
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
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| US32815110P | 2010-04-26 | 2010-04-26 | |
| US61/328,151 | 2010-04-26 | ||
| PCT/US2011/033905 WO2011137103A1 (en) | 2010-04-26 | 2011-04-26 | Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives for the treatment of males |
Publications (1)
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| CA2797560A1 true CA2797560A1 (en) | 2011-11-03 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
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| CA2797560A Withdrawn CA2797560A1 (en) | 2010-04-26 | 2011-04-26 | Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives for the treatment of males |
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| US (3) | US8497256B2 (enExample) |
| EP (1) | EP2563117B1 (enExample) |
| JP (1) | JP2013525440A (enExample) |
| AU (1) | AU2011245455A1 (enExample) |
| BR (2) | BR122014009845A2 (enExample) |
| CA (1) | CA2797560A1 (enExample) |
| IL (1) | IL222642A0 (enExample) |
| MX (1) | MX358142B (enExample) |
| WO (1) | WO2011137103A1 (enExample) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2021528385A (ja) | 2018-06-05 | 2021-10-21 | フラッグシップ パイオニアリング イノベーションズ ブイ， インコーポレイテッド | 自己免疫障害を治療するためのアシル化活性剤およびその使用方法 |
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| US326364A (en) | 1885-09-15 | Electric-lamp hanger | ||
| US4298595A (en) | 1978-12-20 | 1981-11-03 | Dynapol | Pharmaceutical preparations containing a polymeric agent for releasing 5-aminosalicylic acid or its salts into the gastrointestinal tract |
| EP0439453B1 (en) | 1987-10-12 | 1994-01-19 | Exomed Australia Pty. Ltd. (ACN 051 976 446) | Improved method for treatment of gastrointestinal disorders |
| US5443826A (en) | 1988-08-02 | 1995-08-22 | Borody; Thomas J. | Treatment of gastro-intestinal disorders with a fecal composition or a composition of bacteroides and E. Coli |
| US5519014A (en) | 1990-10-22 | 1996-05-21 | Borody; Thomas J. | Treatment of non-inflammatory and non-infectious bowel disorders |
| US5498608A (en) | 1994-01-07 | 1996-03-12 | Salix Pharmaceuticals | Use of 2-hydroxy-5-phenylazobenzoic acid derivatives as colon cancer chemopreventative and chemotherapeutic agents |
| US5905073A (en) | 1995-01-06 | 1999-05-18 | Salix Pharmaceuticals, Inc. | Use of 2-hydroxy-5-phenylazobenzoic acid derivatives as colon cancer chemopreventative and chemotherapeutic agents |
| SE9700934D0 (sv) | 1997-03-14 | 1997-03-14 | Astra Ab | New formulation |
| US6551632B2 (en) | 1997-04-01 | 2003-04-22 | Thomas Julius Borody | Methods and compositions for treating inflammatory bowel disease |
| DE69839261T2 (de) | 1997-04-01 | 2009-03-26 | Borody, Thomas Julius, Five Dock | Verfahren und zusammensetzungen zur behandlung entzündlicher darmerkrankungen |
| AUPO665397A0 (en) | 1997-05-07 | 1997-05-29 | Borody, Thomas Julius | Novel therapy for constipation |
| AUPP437698A0 (en) | 1998-06-30 | 1998-07-23 | Baumgart, Karl | Methods for treatment of coronary, carotid and other vascular disease |
| US6326364B1 (en) | 1999-02-08 | 2001-12-04 | Cedars-Sinai Medical Center | Use of 5-aminosalicylates as antimicrobial agents |
| EP2529729A1 (en) | 2005-08-24 | 2012-12-05 | Salix Pharmaceuticals, Inc. | Balsalazide formulations and manufacture thereof |
| US7452872B2 (en) * | 2005-08-24 | 2008-11-18 | Salix Pharmaceuticals, Inc. | Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives |
| US8921344B2 (en) * | 2006-11-03 | 2014-12-30 | Salix Pharmaceuticals, Inc. | Formulations and uses of 2-hydroxy-5-phenylazobenzoic acid derivatives |
| US20100048519A1 (en) | 2006-09-13 | 2010-02-25 | Chyon-Hwa Yeh | Methods of treatment for ulcerative colitis using aminosalicylate |
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2011
- 2011-04-26 AU AU2011245455A patent/AU2011245455A1/en not_active Abandoned
- 2011-04-26 EP EP11775497.8A patent/EP2563117B1/en active Active
- 2011-04-26 CA CA2797560A patent/CA2797560A1/en not_active Withdrawn
- 2011-04-26 US US13/094,261 patent/US8497256B2/en active Active
- 2011-04-26 JP JP2013508147A patent/JP2013525440A/ja active Pending
- 2011-04-26 WO PCT/US2011/033905 patent/WO2011137103A1/en not_active Ceased
- 2011-04-26 BR BR122014009845A patent/BR122014009845A2/pt not_active Application Discontinuation
- 2011-04-26 MX MX2012012324A patent/MX358142B/es active IP Right Grant
- 2011-04-26 BR BR112012027520A patent/BR112012027520A2/pt not_active IP Right Cessation
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2012
- 2012-10-23 IL IL222642A patent/IL222642A0/en unknown
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2013
- 2013-07-10 US US13/938,777 patent/US20130295178A1/en not_active Abandoned
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2014
- 2014-10-08 US US14/509,446 patent/US20150132381A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| BR112012027520A2 (pt) | 2015-09-15 |
| EP2563117A1 (en) | 2013-03-06 |
| WO2011137103A1 (en) | 2011-11-03 |
| US20120058184A1 (en) | 2012-03-08 |
| EP2563117A4 (en) | 2013-09-04 |
| US20130295178A1 (en) | 2013-11-07 |
| IL222642A0 (en) | 2012-12-31 |
| JP2013525440A (ja) | 2013-06-20 |
| US8497256B2 (en) | 2013-07-30 |
| US20150132381A1 (en) | 2015-05-14 |
| EP2563117B1 (en) | 2018-02-21 |
| BR122014009845A2 (pt) | 2015-12-29 |
| MX2012012324A (es) | 2013-01-29 |
| MX358142B (es) | 2018-08-06 |
| AU2011245455A1 (en) | 2012-11-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request |
Effective date: 20160413 |
|
| AZWI | Withdrawn application |
Effective date: 20200422 |