CA2759891A1 - Gpr 119 modulators - Google Patents
Gpr 119 modulators Download PDFInfo
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- CA2759891A1 CA2759891A1 CA2759891A CA2759891A CA2759891A1 CA 2759891 A1 CA2759891 A1 CA 2759891A1 CA 2759891 A CA2759891 A CA 2759891A CA 2759891 A CA2759891 A CA 2759891A CA 2759891 A1 CA2759891 A1 CA 2759891A1
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- mmol
- carboxylate
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- dihydro
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| TW201111361A (en) | 2009-06-24 | 2011-04-01 | Boehringer Ingelheim Int | New compounds, pharmaceutical composition and methods relating thereto |
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| WO2012025811A1 (en) | 2010-08-23 | 2012-03-01 | Lupin Limited | Indolylpyrimidines as modulators of gpr119 |
| CA2815169C (en) | 2010-10-29 | 2015-10-06 | Pfizer Inc. | N1/n2-lactam acetyl-coa carboxylase inhibitors |
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| EP2813505A1 (en) | 2013-06-14 | 2014-12-17 | Asceneuron SA | Tetraaza-cyclopenta[a]indenyl derivatives |
| JP6348582B2 (ja) | 2013-10-09 | 2018-06-27 | ファイザー・インク | プロスタグランジンｅｐ３受容体の拮抗薬 |
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| US20100120807A1 (en) * | 2007-03-08 | 2010-05-13 | Irm Llc | Compounds and compositions as modulators of gpr119 activity |
| WO2008137436A1 (en) * | 2007-05-04 | 2008-11-13 | Bristol-Myers Squibb Company | [6,5]-bicyclic gpr119 g protein-coupled receptor agonists |
| CN101896481B (zh) * | 2007-10-16 | 2014-04-30 | 第一三共株式会社 | 嘧啶基二氢吲哚化合物 |
| AR076024A1 (es) * | 2009-04-03 | 2011-05-11 | Schering Corp | Derivados de heterociclos biciclicos puenteados y metodos de uso de los mismos |
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- 2010-04-12 CA CA2759891A patent/CA2759891A1/en not_active Abandoned
- 2010-04-12 EP EP10717259A patent/EP2427448A1/en not_active Withdrawn
- 2010-04-12 JP JP2012509115A patent/JP2012526096A/ja not_active Withdrawn
- 2010-04-12 WO PCT/IB2010/051567 patent/WO2010128414A1/en not_active Ceased
- 2010-04-12 US US13/318,152 patent/US20120052130A1/en not_active Abandoned
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| WO2010128414A1 (en) | 2010-11-11 |
| EP2427448A1 (en) | 2012-03-14 |
| JP2012526096A (ja) | 2012-10-25 |
| US20120052130A1 (en) | 2012-03-01 |
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