CA2758965C - Method for the preparation of amphiphilic imidazolinium compounds - Google Patents

Method for the preparation of amphiphilic imidazolinium compounds Download PDF

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Publication number
CA2758965C
CA2758965C CA2758965A CA2758965A CA2758965C CA 2758965 C CA2758965 C CA 2758965C CA 2758965 A CA2758965 A CA 2758965A CA 2758965 A CA2758965 A CA 2758965A CA 2758965 C CA2758965 C CA 2758965C
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CA
Canada
Prior art keywords
compound
formula
molecular sieves
groups
trihaloalkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
CA2758965A
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English (en)
French (fr)
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CA2758965A1 (en
Inventor
Cheng-Sein Yu
Lee B. Bussey
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Juvaris Biotherapeutics Inc
Original Assignee
Juvaris Biotherapeutics Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Juvaris Biotherapeutics Inc filed Critical Juvaris Biotherapeutics Inc
Publication of CA2758965A1 publication Critical patent/CA2758965A1/en
Application granted granted Critical
Publication of CA2758965C publication Critical patent/CA2758965C/en
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C07D233/60—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms with hydrocarbon radicals, substituted by oxygen or sulfur atoms, attached to ring nitrogen atoms
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
CA2758965A 2009-04-29 2010-04-28 Method for the preparation of amphiphilic imidazolinium compounds Active CA2758965C (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US12/432,660 US8044215B2 (en) 2009-04-29 2009-04-29 Methods for the preparation of amphillic nitrogen containing imidazolinium derivative compounds
US12/432,660 2009-04-29
PCT/US2010/032723 WO2010126978A1 (en) 2009-04-29 2010-04-28 Methods for the preparation of amphiphilic nitrogen containing imidazolinium derivative compounds

Publications (2)

Publication Number Publication Date
CA2758965A1 CA2758965A1 (en) 2010-11-04
CA2758965C true CA2758965C (en) 2017-07-11

Family

ID=42235194

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2758965A Active CA2758965C (en) 2009-04-29 2010-04-28 Method for the preparation of amphiphilic imidazolinium compounds

Country Status (7)

Country Link
US (1) US8044215B2 (enExample)
EP (1) EP2430001B1 (enExample)
JP (1) JP5647231B2 (enExample)
AU (1) AU2010241712B2 (enExample)
BR (1) BRPI1015376A2 (enExample)
CA (1) CA2758965C (enExample)
WO (1) WO2010126978A1 (enExample)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1811202A1 (en) 2005-12-30 2007-07-25 Fallbrook Technologies, Inc. A continuously variable gear transmission
US8996263B2 (en) 2007-11-16 2015-03-31 Fallbrook Intellectual Property Company Llc Controller for variable transmission
EP3292106B1 (en) * 2015-05-04 2021-10-27 Bayer Animal Health GmbH Process for the preparation of amphiphilic imidazolinium compounds
US10047861B2 (en) 2016-01-15 2018-08-14 Fallbrook Intellectual Property Company Llc Systems and methods for controlling rollback in continuously variable transmissions
US10023266B2 (en) 2016-05-11 2018-07-17 Fallbrook Intellectual Property Company Llc Systems and methods for automatic configuration and automatic calibration of continuously variable transmissions and bicycles having continuously variable transmissions
US11215268B2 (en) 2018-11-06 2022-01-04 Fallbrook Intellectual Property Company Llc Continuously variable transmissions, synchronous shifting, twin countershafts and methods for control of same
US11174922B2 (en) 2019-02-26 2021-11-16 Fallbrook Intellectual Property Company Llc Reversible variable drives and systems and methods for control in forward and reverse directions

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5264618A (en) * 1990-04-19 1993-11-23 Vical, Inc. Cationic lipids for intracellular delivery of biologically active molecules
US5705655A (en) * 1992-12-17 1998-01-06 Megabios Corporation Amphiphilic nitrogen containing imidazolinium derivative compounds and uses
FR2711525B1 (fr) * 1993-10-29 1996-01-12 Virbac Laboratoires Forme Galénique à administration orale pour animaux, son procédé de préparation et ses applications.
US5830878A (en) * 1995-06-07 1998-11-03 Megabios Corporation Cationic lipid: DNA complexes for gene targeting
US6121457A (en) 1997-11-14 2000-09-19 Megabios Corporation Compositions and methods using novel substituted imidazolium lipids

Also Published As

Publication number Publication date
WO2010126978A1 (en) 2010-11-04
AU2010241712A1 (en) 2011-11-24
EP2430001B1 (en) 2013-12-11
AU2010241712B2 (en) 2014-10-23
US8044215B2 (en) 2011-10-25
US20100280258A1 (en) 2010-11-04
JP2012525406A (ja) 2012-10-22
CA2758965A1 (en) 2010-11-04
EP2430001A1 (en) 2012-03-21
BRPI1015376A2 (pt) 2015-09-01
JP5647231B2 (ja) 2014-12-24

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Effective date: 20150320

H11 Ip right ceased following rejected request for revival

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Effective date: 20241030