CA2717133A1 - Liposome pour une administration au segment posterieur de l'oeil et composition pharmaceutique pour une maladie du segment posterieur de l'oeil - Google Patents

Liposome pour une administration au segment posterieur de l'oeil et composition pharmaceutique pour une maladie du segment posterieur de l'oeil Download PDF

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Publication number
CA2717133A1
CA2717133A1 CA2717133A CA2717133A CA2717133A1 CA 2717133 A1 CA2717133 A1 CA 2717133A1 CA 2717133 A CA2717133 A CA 2717133A CA 2717133 A CA2717133 A CA 2717133A CA 2717133 A1 CA2717133 A1 CA 2717133A1
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CA
Canada
Prior art keywords
liposome
posterior segment
eye
delivery
disease
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
CA2717133A
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English (en)
Other versions
CA2717133C (fr
Inventor
Hideaki Hara
Hirofumi Takeuchi
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Nagoya Industrial Science Research Institute
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Nagoya Industrial Science Research Institute
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
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Publication of CA2717133A1 publication Critical patent/CA2717133A1/fr
Application granted granted Critical
Publication of CA2717133C publication Critical patent/CA2717133C/fr
Expired - Fee Related legal-status Critical Current
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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0048Eye, e.g. artificial tears
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/127Liposomes
    • A61K9/1271Non-conventional liposomes, e.g. PEGylated liposomes, liposomes coated with polymers
    • A61K9/1272Non-conventional liposomes, e.g. PEGylated liposomes, liposomes coated with polymers with substantial amounts of non-phosphatidyl, i.e. non-acylglycerophosphate, surfactants as bilayer-forming substances, e.g. cationic lipids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Biophysics (AREA)
  • Dispersion Chemistry (AREA)
  • Molecular Biology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA2717133A 2008-02-29 2009-02-26 Liposome pour une administration au segment posterieur de l'oeil et composition pharmaceutique pour une maladie du segment posterieur de l'oeil Expired - Fee Related CA2717133C (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2008-051427 2008-02-29
JP2008051427 2008-02-29
PCT/JP2009/053609 WO2009107753A1 (fr) 2008-02-29 2009-02-26 Liposome pour une administration au segment postérieur de l'œil et composition pharmaceutique pour une maladie du segment postérieur de l'œil

Publications (2)

Publication Number Publication Date
CA2717133A1 true CA2717133A1 (fr) 2009-09-03
CA2717133C CA2717133C (fr) 2016-04-26

Family

ID=41016140

Family Applications (1)

Application Number Title Priority Date Filing Date
CA2717133A Expired - Fee Related CA2717133C (fr) 2008-02-29 2009-02-26 Liposome pour une administration au segment posterieur de l'oeil et composition pharmaceutique pour une maladie du segment posterieur de l'oeil

Country Status (7)

Country Link
US (1) US9114070B2 (fr)
EP (1) EP2255788B1 (fr)
JP (1) JP5514098B2 (fr)
CN (1) CN101959503A (fr)
CA (1) CA2717133C (fr)
TW (1) TW200942271A (fr)
WO (1) WO2009107753A1 (fr)

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* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2010256558B2 (en) 2009-06-03 2013-10-03 Forsight Labs, Llc Anterior segment drug delivery
JPWO2011062255A1 (ja) * 2009-11-20 2013-04-11 コニカミノルタホールディングス株式会社 混合有機溶媒を油相として用いる二段階乳化によるリポソームの製造方法
JP2011246464A (ja) * 2010-04-28 2011-12-08 Wakamoto Pharmaceutical Co Ltd ジクロフェナクナトリウムを封入した後眼部到達用ポリマーコーティングリポソーム
WO2012021107A2 (fr) 2010-08-12 2012-02-16 Nanyang Technological University Formulation de liposomes pour l'administration d'un médicament dans l'œil
CN103975202B (zh) * 2012-01-05 2016-09-14 三菱电机株式会社 空调装置
JP6231995B2 (ja) * 2012-02-10 2017-11-15 タイワン リポソーム カンパニー リミテッド 眼の疾患の合併症を低減するための薬学的組成物
CN103860467A (zh) * 2012-11-22 2014-06-18 苏州太湖美药业有限公司 溴芬酸钠脂质体滴眼液
EP3057514A4 (fr) * 2013-10-15 2017-08-02 Forsight Vision5, Inc. Préparations et méthodes permettant d'augmenter ou de réduire le mucus
US9956195B2 (en) 2014-01-07 2018-05-01 Nanyang Technological University Stable liposomal formulations for ocular drug delivery
CN106458920B (zh) * 2014-03-31 2019-02-15 千寿制药株式会社 炔基吲唑衍生物及其用途
KR20170048426A (ko) * 2014-08-22 2017-05-08 광저우 캉루이 바이오로지컬 파마슈티컬 테크놀로지 씨오., 엘티디. 시각 장애를 치료하기 위한 조성물 및 방법
EA201791337A1 (ru) 2014-12-15 2017-11-30 Дзе Джонс Хопкинс Юниверсити Составы сунитиниба и способы их применения в лечении глазных нарушений
WO2016104690A1 (fr) 2014-12-25 2016-06-30 国立大学法人京都大学 Lipoprotéine haute densité et administration de médicament au segment postérieur de l'œil par instillation oculaire de ladite lipoprotéine haute densité fusionnée à un peptide cytophile
EP3283004A4 (fr) 2015-04-13 2018-12-05 Forsight Vision5, Inc. Composition d'insert oculaire d'agent pharmaceutiquement actif cristallin ou semi-cristallin
WO2017027017A1 (fr) * 2015-08-11 2017-02-16 Peregrine Ophthalmic PTE LTD. Formulations liposomales stables d'inhibiteurs de l'anhydrase carbonique pour administration médicamenteuse oculaires
CN109364020B (zh) * 2015-09-02 2021-12-28 盛世泰科生物医药技术(苏州)有限公司 一种用于预防和治疗白内障的眼用制剂及其制备方法
BR112018009644A2 (pt) 2015-11-12 2018-11-06 Graybug Vision Inc micropartículas agregantes sólidas modificadas na superfície, material injetável, processo para preparação de micropartículas agregantes sólidas modificadas na superfície, método para tratamento de um distúrbio ocular, e, uso de micropartículas agregantes sólidas modificadas na superfície
US20190133931A1 (en) * 2016-04-19 2019-05-09 Nanyang Technological University Subconjunctival depot forming formulations for ocular drug delivery
BR112019003160A2 (pt) * 2016-08-18 2019-05-28 Bremer Troy composição farmacêutica, métodos para distribuir ureia na interface vitreorretiniana, para induzir desprendimento vítreo posterior e para tratar retinopatia diabética ou adesão vitreomacular, e, uso da composição farmacêutica.
WO2018209155A1 (fr) 2017-05-10 2018-11-15 Graybug Vision, Inc. Microparticules à libération prolongée et suspensions de celles-ci destinées à une thérapie médicale
WO2020189773A1 (fr) * 2019-03-20 2020-09-24 洋文 竹内 Composition d'administration au segment postérieur

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4938965A (en) * 1987-07-22 1990-07-03 Her Majesty The Queen In Right Of Canada, As Represented By The Minister Of National Defence Of Her Majesty's Canadian Government Ocular delivery of prophylactic agents
JPH04505319A (ja) * 1989-04-04 1992-09-17 アルコン ラボラトリーズ インコーポレイテッド 創傷、切傷および擦傷に対する治療剤のデリバリーとしてのリポソームの使用
CA2205863A1 (fr) * 1994-12-19 1996-06-27 Taisho Pharmaceutical Co., Ltd. Gouttes de collyre aux liposomes
JP3963506B2 (ja) 1996-08-26 2007-08-22 俊彦 松尾 リポソーム点眼剤
AU2001292287A1 (en) 2000-10-26 2002-05-06 Senju Pharmaceutical Co. Ltd. Drug composition comprising dipeptydyl aldehyde derivative
JP4228195B2 (ja) 2002-02-22 2009-02-25 参天製薬株式会社 微粒子結膜下投与ドラッグデリバリーシステム
KR20040084931A (ko) * 2002-02-22 2004-10-06 산텐 세이야꾸 가부시키가이샤 미립자 결막하 투여를 위한 약물 수송 시스템
CN100431525C (zh) 2003-07-17 2008-11-12 台湾东洋药品工业股份有限公司 脂质体悬浮液制造方法及含该法所制脂质体悬浮液的产物
RU2369384C2 (ru) 2003-11-20 2009-10-10 ЙЭм БАЙОСАЙЕНСИЗ ИНК. Стабильные липосомальные композиции
CN1256091C (zh) 2004-06-29 2006-05-17 常州太平洋药物研究所有限公司 阿霉素或盐酸阿霉素脂质体注射剂及其制备工艺
CN100566810C (zh) 2005-01-18 2009-12-09 国立大学法人北海道大学 用脂质膜被覆粒子的方法
WO2007096744A1 (fr) 2006-02-21 2007-08-30 Pfizer Products Inc. Methodes de traitement de la degenerescence maculaire et de pathologies de l'oeil associees

Also Published As

Publication number Publication date
TW200942271A (en) 2009-10-16
EP2255788B1 (fr) 2015-07-22
CA2717133C (fr) 2016-04-26
CN101959503A (zh) 2011-01-26
EP2255788A1 (fr) 2010-12-01
US9114070B2 (en) 2015-08-25
JP5514098B2 (ja) 2014-06-04
EP2255788A4 (fr) 2013-07-10
WO2009107753A1 (fr) 2009-09-03
JPWO2009107753A1 (ja) 2011-07-07
US20110008421A1 (en) 2011-01-13

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