CA2689987A1 - Composition pharmaceutique d'un nouveau systeme destine a la liberation de steroides dans le vagin - Google Patents
Composition pharmaceutique d'un nouveau systeme destine a la liberation de steroides dans le vagin Download PDFInfo
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- CA2689987A1 CA2689987A1 CA2689987A CA2689987A CA2689987A1 CA 2689987 A1 CA2689987 A1 CA 2689987A1 CA 2689987 A CA2689987 A CA 2689987A CA 2689987 A CA2689987 A CA 2689987A CA 2689987 A1 CA2689987 A1 CA 2689987A1
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- LYCAIKOWRPUZTN-UHFFFAOYSA-N ethylene glycol Natural products OCCO LYCAIKOWRPUZTN-UHFFFAOYSA-N 0.000 description 1
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- 238000010874 in vitro model Methods 0.000 description 1
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- 229940039696 lactobacillus Drugs 0.000 description 1
- 229940039695 lactobacillus acidophilus Drugs 0.000 description 1
- GFIJNRVAKGFPGQ-LIJARHBVSA-N leuprolide Chemical compound CCNC(=O)[C@@H]1CCCN1C(=O)[C@H](CCCNC(N)=N)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](CO)NC(=O)[C@H](CC=1C2=CC=CC=C2NC=1)NC(=O)[C@H](CC=1N=CNC=1)NC(=O)[C@H]1NC(=O)CC1)CC1=CC=C(O)C=C1 GFIJNRVAKGFPGQ-LIJARHBVSA-N 0.000 description 1
- 229960004338 leuprorelin Drugs 0.000 description 1
- 150000002634 lipophilic molecules Chemical class 0.000 description 1
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- 239000007935 oral tablet Substances 0.000 description 1
- 210000001672 ovary Anatomy 0.000 description 1
- 230000027758 ovulation cycle Effects 0.000 description 1
- 239000000813 peptide hormone Substances 0.000 description 1
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- 239000010452 phosphate Substances 0.000 description 1
- NBIIXXVUZAFLBC-UHFFFAOYSA-K phosphate Chemical compound [O-]P([O-])([O-])=O NBIIXXVUZAFLBC-UHFFFAOYSA-K 0.000 description 1
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- 208000016685 primary ovarian failure Diseases 0.000 description 1
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- 230000008569 process Effects 0.000 description 1
- 108090000765 processed proteins & peptides Proteins 0.000 description 1
- 108090000623 proteins and genes Proteins 0.000 description 1
- 102000004169 proteins and genes Human genes 0.000 description 1
- 239000008213 purified water Substances 0.000 description 1
- 210000002321 radial artery Anatomy 0.000 description 1
- 239000003488 releasing hormone Substances 0.000 description 1
- 238000012552 review Methods 0.000 description 1
- 239000000932 sedative agent Substances 0.000 description 1
- 230000001624 sedative effect Effects 0.000 description 1
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- FBWNMEQMRUMQSO-UHFFFAOYSA-N tergitol NP-9 Chemical compound CCCCCCCCCC1=CC=C(OCCOCCOCCOCCOCCOCCOCCOCCOCCO)C=C1 FBWNMEQMRUMQSO-UHFFFAOYSA-N 0.000 description 1
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Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0034—Urogenital system, e.g. vagina, uterus, cervix, penis, scrotum, urethra, bladder; Personal lubricants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Diabetes (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Gynecology & Obstetrics (AREA)
- Reproductive Health (AREA)
- Urology & Nephrology (AREA)
- Endocrinology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CL2007001634 | 2007-06-06 | ||
| CL1634-2007 | 2007-06-06 | ||
| PCT/US2008/065722 WO2008154240A1 (fr) | 2007-06-06 | 2008-06-04 | Composition pharmaceutique d'un nouveau système destiné à la libération de stéroïdes dans le vagin |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2689987A1 true CA2689987A1 (fr) | 2008-12-18 |
Family
ID=40951496
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2689987A Abandoned CA2689987A1 (fr) | 2007-06-06 | 2008-06-04 | Composition pharmaceutique d'un nouveau systeme destine a la liberation de steroides dans le vagin |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP2157946A1 (fr) |
| CN (1) | CN101730514A (fr) |
| AR (1) | AR070302A1 (fr) |
| BR (1) | BRPI0812578A2 (fr) |
| CA (1) | CA2689987A1 (fr) |
| CO (1) | CO6270199A2 (fr) |
| MX (1) | MX2009013305A (fr) |
| PE (1) | PE20090324A1 (fr) |
| WO (1) | WO2008154240A1 (fr) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2011073995A2 (fr) | 2009-12-14 | 2011-06-23 | Lincoln Pharmaceuticals Limited | Liquide contenant de la progestérone à pulvériser dans le vagin |
| WO2015073066A1 (fr) | 2013-11-12 | 2015-05-21 | University Of Utah Research Foundation | Hydrogel thermosensible à base de glycol-chitine pour administration de progestérone par voie vaginale |
| CN114129530A (zh) * | 2021-12-08 | 2022-03-04 | 南京康川济医药科技有限公司 | 一种黄体酮缓释组合物及其制备方法 |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1997040792A1 (fr) * | 1996-04-30 | 1997-11-06 | Theratech, Inc. | Administration transdermique d'hormones steroidiennes au moyen de diethanolamides d'acides gras c12-c18 utilises comme activateurs de l'infiltration |
| ITMI20010913A1 (it) * | 2001-05-04 | 2002-11-04 | Univ Pavia | Composizioni a rilascio controllato di acido lattico a livello vaginale |
-
2008
- 2008-06-04 CA CA2689987A patent/CA2689987A1/fr not_active Abandoned
- 2008-06-04 CN CN200880019113A patent/CN101730514A/zh active Pending
- 2008-06-04 WO PCT/US2008/065722 patent/WO2008154240A1/fr active Application Filing
- 2008-06-04 EP EP08770092A patent/EP2157946A1/fr not_active Withdrawn
- 2008-06-04 MX MX2009013305A patent/MX2009013305A/es not_active Application Discontinuation
- 2008-06-04 BR BRPI0812578A patent/BRPI0812578A2/pt not_active IP Right Cessation
- 2008-06-05 AR ARP080102407A patent/AR070302A1/es not_active Application Discontinuation
- 2008-06-05 PE PE2008000954A patent/PE20090324A1/es not_active Application Discontinuation
-
2010
- 2010-01-06 CO CO10001028A patent/CO6270199A2/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| MX2009013305A (es) | 2010-04-21 |
| AR070302A1 (es) | 2010-03-31 |
| EP2157946A1 (fr) | 2010-03-03 |
| CN101730514A (zh) | 2010-06-09 |
| CO6270199A2 (es) | 2011-04-20 |
| BRPI0812578A2 (pt) | 2015-09-29 |
| PE20090324A1 (es) | 2009-04-09 |
| WO2008154240A1 (fr) | 2008-12-18 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request | ||
| FZDE | Dead |
Effective date: 20130516 |