CA2570386A1 - Methods of using albuterol and calcium activated potassium channel openers - Google Patents
Methods of using albuterol and calcium activated potassium channel openers Download PDFInfo
- Publication number
- CA2570386A1 CA2570386A1 CA002570386A CA2570386A CA2570386A1 CA 2570386 A1 CA2570386 A1 CA 2570386A1 CA 002570386 A CA002570386 A CA 002570386A CA 2570386 A CA2570386 A CA 2570386A CA 2570386 A1 CA2570386 A1 CA 2570386A1
- Authority
- CA
- Canada
- Prior art keywords
- albuterol
- potassium channel
- pharmaceutically acceptable
- solvate
- dosage form
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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- 229960002052 salbutamol Drugs 0.000 title claims abstract description 45
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Classifications
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pulmonology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Molecular Biology (AREA)
- Immunology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US57882704P | 2004-06-14 | 2004-06-14 | |
| US60/578,827 | 2004-06-14 | ||
| US59902704P | 2004-08-06 | 2004-08-06 | |
| US60/599,027 | 2004-08-06 | ||
| US60729004P | 2004-09-07 | 2004-09-07 | |
| US60/607,290 | 2004-09-07 | ||
| PCT/US2005/021171 WO2005123071A1 (en) | 2004-06-14 | 2005-06-14 | Methods of using albuterol and calcium activated potassium channel openers |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2570386A1 true CA2570386A1 (en) | 2005-12-29 |
Family
ID=35509445
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002570386A Abandoned CA2570386A1 (en) | 2004-06-14 | 2005-06-14 | Methods of using albuterol and calcium activated potassium channel openers |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20090035224A1 (enExample) |
| EP (1) | EP1773325A4 (enExample) |
| JP (1) | JP2008502698A (enExample) |
| AU (1) | AU2005254096A1 (enExample) |
| CA (1) | CA2570386A1 (enExample) |
| WO (1) | WO2005123071A1 (enExample) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SI1634595T1 (sl) * | 2004-08-19 | 2008-12-31 | Rottapharm Spa | N-fenilbenzamidni derivati kot zdravila za zdravljenje kronične obstruktivne pljučne bolezni (KOPB) |
| US20100015061A1 (en) * | 2006-01-06 | 2010-01-21 | Boehringer Ingeheim International GmnH | Pharmaceutical Compositions Based on Anticholinergics and Andolast |
| ES2365533T3 (es) * | 2006-07-31 | 2011-10-06 | Rottapharm S.P.A. | Combinación de andolast / glucocorticoides. |
| JP6211380B2 (ja) * | 2012-10-17 | 2017-10-11 | 丸善製薬株式会社 | Tie2活性化剤、血管新生抑制剤、血管の成熟化剤、血管の正常化剤、及び血管の安定化剤 |
| JP2013056925A (ja) * | 2012-11-21 | 2013-03-28 | Rottapharm Spa | アンドラスト/グルココルチコイドの併用 |
| CN112535668B (zh) * | 2020-10-29 | 2023-08-18 | 苏州君宁新药开发中心有限公司 | 一种左旋硫酸沙丁胺醇颗粒剂及其用途 |
| CN113476428B (zh) * | 2021-01-28 | 2022-03-29 | 朗天药业(湖北)有限公司 | 一种吸入用硫酸沙丁胺醇溶液及其制备方法 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU7174191A (en) * | 1990-01-05 | 1991-07-24 | Sepracor, Inc. | Optically pure r(-) albuterol for treating asthma |
| US5200422A (en) * | 1990-09-24 | 1993-04-06 | Neurosearch A/S | Benzimidazole derivatives, their preparation and use |
| US5637470A (en) * | 1994-05-13 | 1997-06-10 | Merck & Co., Inc. | Screening array using cells expressing recombinant α and β subunits of the mammalian large-conductance (maxi-K) potassium channel |
| ES2199336T3 (es) * | 1997-08-08 | 2004-02-16 | Rotta Research Laboratorium S.P.A. | Una composicion farmaceutica novedosa para inhalacion que contiene cr 2039 (andolast). |
| EP1107747A4 (en) * | 1998-08-26 | 2003-04-23 | Smithkline Beecham Corp | COMPOSITIONS FOR THE TREATMENT OF PULMONARY DISEASES |
| US6656461B1 (en) * | 2000-02-29 | 2003-12-02 | The Trustees Of Columbia University In The City Of New York | Therapeutic treatment of chronic obstructive pulmonary disease |
| US7713964B2 (en) * | 2001-12-03 | 2010-05-11 | Wyeth Llc | Methods for treating asthmatic conditions |
| TWI271402B (en) * | 2002-10-15 | 2007-01-21 | Tanabe Seiyaku Co | Large conductance calcium-activated K channel opener |
| US20040109826A1 (en) * | 2002-12-06 | 2004-06-10 | Dey, L.P. | Stabilized albuterol compositions and method of preparation thereof |
-
2005
- 2005-06-14 US US11/629,686 patent/US20090035224A1/en not_active Abandoned
- 2005-06-14 CA CA002570386A patent/CA2570386A1/en not_active Abandoned
- 2005-06-14 WO PCT/US2005/021171 patent/WO2005123071A1/en not_active Ceased
- 2005-06-14 EP EP05766071A patent/EP1773325A4/en not_active Withdrawn
- 2005-06-14 AU AU2005254096A patent/AU2005254096A1/en not_active Abandoned
- 2005-06-14 JP JP2007516693A patent/JP2008502698A/ja not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| JP2008502698A (ja) | 2008-01-31 |
| AU2005254096A1 (en) | 2005-12-29 |
| EP1773325A4 (en) | 2007-11-07 |
| US20090035224A1 (en) | 2009-02-05 |
| EP1773325A1 (en) | 2007-04-18 |
| WO2005123071A1 (en) | 2005-12-29 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Discontinued | ||
| FZDE | Discontinued |
Effective date: 20110614 |