CA2543338A1 - Novel medical uses of compounds showing cb1-antagonistic activity and combination treatment involving said compounds - Google Patents

Novel medical uses of compounds showing cb1-antagonistic activity and combination treatment involving said compounds Download PDF

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Publication number
CA2543338A1
CA2543338A1 CA002543338A CA2543338A CA2543338A1 CA 2543338 A1 CA2543338 A1 CA 2543338A1 CA 002543338 A CA002543338 A CA 002543338A CA 2543338 A CA2543338 A CA 2543338A CA 2543338 A1 CA2543338 A1 CA 2543338A1
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Canada
Prior art keywords
group
alkyl
substituted
compound
treatment
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Abandoned
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CA002543338A
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English (en)
French (fr)
Inventor
Jochen Antel
Peter-Colin Gregory
Harald Waldeck
Guenter Krause
Josephus Hubertus Maria Lange
Chris Kruse
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Abbott Products GmbH
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Individual
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Publication of CA2543338A1 publication Critical patent/CA2543338A1/en
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    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/365—Lactones
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  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Pulmonology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Psychology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Hematology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Addiction (AREA)
  • Virology (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Toxicology (AREA)
CA002543338A 2003-10-24 2004-10-22 Novel medical uses of compounds showing cb1-antagonistic activity and combination treatment involving said compounds Abandoned CA2543338A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
EP03103961.3 2003-10-24
EP03103961 2003-10-24
EP03103967.0 2003-10-27
EP03103967 2003-10-27
PCT/EP2004/052639 WO2005039550A2 (en) 2003-10-24 2004-10-22 Novel medical uses of compounds showing cb1-antagonistic activity and combination treatment involving said compounds

Publications (1)

Publication Number Publication Date
CA2543338A1 true CA2543338A1 (en) 2005-05-06

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Application Number Title Priority Date Filing Date
CA002543338A Abandoned CA2543338A1 (en) 2003-10-24 2004-10-22 Novel medical uses of compounds showing cb1-antagonistic activity and combination treatment involving said compounds

Country Status (8)

Country Link
EP (1) EP1753413A2 (de)
JP (1) JP2007513872A (de)
AU (1) AU2004283056A1 (de)
BR (1) BRPI0415851A (de)
CA (1) CA2543338A1 (de)
MX (1) MXPA06004434A (de)
RU (1) RU2006117627A (de)
WO (1) WO2005039550A2 (de)

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WO2004058145A2 (en) 2002-12-19 2004-07-15 Merck & Co., Inc. Substituted amides
AR046132A1 (es) * 2003-10-24 2005-11-23 Solvay Pharm Gmbh Composicin farmaceutica que contiene al menos un compuesto con actividad de receptor de cb1, o un profarmaco , tautomero o sal del mismo, como componente activo adecuado para el tratamiento y/o profilaxis de enfermedades relacionadas con el receptor cb1 en pacientes juveniles y/o para el tratamiento
CN101084207A (zh) 2004-09-20 2007-12-05 泽农医药公司 杂环衍生物及其作为硬脂酰CoA去饱和酶抑制剂的用途
MX2007003321A (es) 2004-09-20 2007-06-05 Xenon Pharmaceuticals Inc Derivados heterociclicos y su uso como agentes terapeuticos.
EP2316458A1 (de) 2004-09-20 2011-05-04 Xenon Pharmaceuticals Inc. Pyridazin-Derivate zur Verhinderung menschlicher Stearoyl-coa-desaturas
US7592343B2 (en) 2004-09-20 2009-09-22 Xenon Pharmaceuticals Inc. Pyridazine-piperazine compounds and their use as stearoyl-CoA desaturase inhibitors
CN101084212A (zh) 2004-09-20 2007-12-05 泽农医药公司 杂环衍生物及其作为硬脂酰CoA去饱和酶介导剂的用途
EP2289510A1 (de) 2004-09-20 2011-03-02 Xenon Pharmaceuticals Inc. Heterozyklische Derivate zur Behandlung von durch Stearoyl-Coa-Desaturase-Enzyme verursachten Krankheiten
WO2006034440A2 (en) 2004-09-20 2006-03-30 Xenon Pharmaceuticals Inc. Heterocyclic derivatives and their use as stearoyl-coa desaturase inhibitors
CN101208089A (zh) 2005-06-03 2008-06-25 泽农医药公司 氨基噻唑衍生物作为人硬酯酰-CoA去饱和酶抑制剂
EP1921073A1 (de) 2006-11-10 2008-05-14 Laboratorios del Dr. Esteve S.A. 1,2,4-Triazole als Sigma Rezeptoren Hemmstoffe

Family Cites Families (16)

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EP1753413A2 (de) 2007-02-21
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MXPA06004434A (es) 2006-06-20
BRPI0415851A (pt) 2007-01-02

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