CA2542909C - 2-aminoaryloxazole compounds as tyrosine kinase inhibitors - Google Patents
2-aminoaryloxazole compounds as tyrosine kinase inhibitors Download PDFInfo
- Publication number
- CA2542909C CA2542909C CA2542909A CA2542909A CA2542909C CA 2542909 C CA2542909 C CA 2542909C CA 2542909 A CA2542909 A CA 2542909A CA 2542909 A CA2542909 A CA 2542909A CA 2542909 C CA2542909 C CA 2542909C
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- Prior art keywords
- phenyl
- oxazol
- methyl
- pyridin
- ylamino
- Prior art date
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Classifications
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- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
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- Pharmacology & Pharmacy (AREA)
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- Biomedical Technology (AREA)
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- Transplantation (AREA)
- Urology & Nephrology (AREA)
- Heart & Thoracic Surgery (AREA)
- Vascular Medicine (AREA)
- Surgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicinal Preparation (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US51321403P | 2003-10-23 | 2003-10-23 | |
| US60/513,214 | 2003-10-23 | ||
| PCT/IB2004/003698 WO2005040139A2 (en) | 2003-10-23 | 2004-10-22 | 2-aminoaryloxazole compounds as tyrosine kinase inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CA2542909A1 CA2542909A1 (en) | 2005-05-06 |
| CA2542909C true CA2542909C (en) | 2012-07-10 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2542909A Expired - Fee Related CA2542909C (en) | 2003-10-23 | 2004-10-22 | 2-aminoaryloxazole compounds as tyrosine kinase inhibitors |
Country Status (15)
| Country | Link |
|---|---|
| US (2) | US7718676B2 (https=) |
| EP (1) | EP1684750B1 (https=) |
| JP (1) | JP4971797B2 (https=) |
| CN (1) | CN1950347B (https=) |
| AT (1) | ATE465731T1 (https=) |
| AU (1) | AU2004283162B2 (https=) |
| BR (1) | BRPI0415467A (https=) |
| CA (1) | CA2542909C (https=) |
| DK (1) | DK1684750T3 (https=) |
| HR (1) | HRP20100326T1 (https=) |
| IL (1) | IL175028A (https=) |
| NO (1) | NO20062308L (https=) |
| NZ (1) | NZ546645A (https=) |
| PL (1) | PL1684750T3 (https=) |
| WO (1) | WO2005040139A2 (https=) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8272435B2 (en) | 2003-05-31 | 2012-09-25 | Cameron Systems (Ireland) Limited | Apparatus and method for recovering fluids from a well and/or injecting fluids into a well |
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| US7652044B2 (en) * | 2003-06-03 | 2010-01-26 | Novartis A.G. | P-38 inhibitors |
| EP1684750B1 (en) * | 2003-10-23 | 2010-04-28 | AB Science | 2-aminoaryloxazole compounds as tyrosine kinase inhibitors |
| CA2555403C (en) | 2004-02-26 | 2012-08-21 | Des Enhanced Recovery Limited | Connection system for subsea flow interface equipment |
| WO2005102318A1 (en) * | 2004-04-20 | 2005-11-03 | Ab Science | Use of c-kit inhibitors for treating hiv related diseases |
| CA2564568A1 (en) * | 2004-04-20 | 2005-11-03 | Ab Science | Use of c-kit inhibitors for treating inflammatory muscle disorders including myositis and muscular dystrophy |
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| US8272435B2 (en) | 2003-05-31 | 2012-09-25 | Cameron Systems (Ireland) Limited | Apparatus and method for recovering fluids from a well and/or injecting fluids into a well |
Also Published As
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| US7718676B2 (en) | 2010-05-18 |
| BRPI0415467A (pt) | 2006-12-19 |
| JP2007509130A (ja) | 2007-04-12 |
| WO2005040139A3 (en) | 2005-10-13 |
| IL175028A (en) | 2011-02-28 |
| AU2004283162B2 (en) | 2011-12-15 |
| CA2542909A1 (en) | 2005-05-06 |
| DK1684750T3 (da) | 2010-08-09 |
| EP1684750A2 (en) | 2006-08-02 |
| CN1950347A (zh) | 2007-04-18 |
| US8110591B2 (en) | 2012-02-07 |
| ATE465731T1 (de) | 2010-05-15 |
| US20070142390A1 (en) | 2007-06-21 |
| PL1684750T3 (pl) | 2010-10-29 |
| WO2005040139A8 (en) | 2006-06-01 |
| IL175028A0 (en) | 2006-08-20 |
| HRP20100326T1 (hr) | 2010-10-31 |
| NZ546645A (en) | 2010-02-26 |
| EP1684750B1 (en) | 2010-04-28 |
| NO20062308L (no) | 2006-05-22 |
| CN1950347B (zh) | 2012-04-04 |
| AU2004283162A1 (en) | 2005-05-06 |
| WO2005040139A2 (en) | 2005-05-06 |
| US20100113471A1 (en) | 2010-05-06 |
| JP4971797B2 (ja) | 2012-07-11 |
| HK1091134A1 (en) | 2007-01-12 |
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