CA2486055C - Amines that inhibit a mammalian anandamide transporter, and methods of use thereof - Google Patents
Amines that inhibit a mammalian anandamide transporter, and methods of use thereof Download PDFInfo
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- CA2486055C CA2486055C CA2486055A CA2486055A CA2486055C CA 2486055 C CA2486055 C CA 2486055C CA 2486055 A CA2486055 A CA 2486055A CA 2486055 A CA2486055 A CA 2486055A CA 2486055 C CA2486055 C CA 2486055C
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| PCT/US2003/015581 WO2003097573A1 (en) | 2002-05-16 | 2003-05-15 | Amines that inhibit a mammalian anandamide transporter, and methods of use thereof |
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| CA2486055A1 CA2486055A1 (en) | 2003-11-27 |
| CA2486055C true CA2486055C (en) | 2012-03-06 |
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| AU2003237882B2 (en) * | 2002-05-16 | 2010-04-08 | Sunovion Pharmaceuticals Inc. | Amines that inhibit a mammalian anandamide transporter, and methods of use thereof |
| FR2864080B1 (fr) * | 2003-12-23 | 2006-02-03 | Sanofi Synthelabo | Derives de 1-piperazine-et-1-homopiperazine-carboxylates, leur preparation et leur application en therapeutique |
| FR2866888B1 (fr) * | 2004-02-26 | 2006-05-05 | Sanofi Synthelabo | Derives de alkylpiperazine- et alkylhomopiperazine- carboxylates, leur preparation et leur application en therapeutique |
| US20060084659A1 (en) * | 2004-10-19 | 2006-04-20 | Michael Davis | Augmentation of psychotherapy with cannabinoid reuptake inhibitors |
| WO2006116773A2 (en) * | 2005-04-28 | 2006-11-02 | The Regents Of The University Of California | Methods, compositions, and compounds for modulation of monoacylglycerol lipase, pain, and stress-related disorders |
| WO2010083532A1 (en) * | 2009-01-19 | 2010-07-22 | The Research Foundaton Of State University Of New York | Fatty acid binding proteins as drug targets for modulation of endocannabinoids |
| ES2708723T3 (es) | 2011-08-19 | 2019-04-10 | Univ California | Inhibidores de FAAH restringidos de forma periférica sustituidos en posición meta por bifenilo |
| ES2908240T3 (es) | 2014-04-07 | 2022-04-28 | Univ California | Inhibidores de la enzima amida hidrolasa de ácidos grasos (FAAH) con biodisponibilidad oral mejorada y su uso como medicamentos |
| FR3071833B1 (fr) * | 2017-09-29 | 2020-01-03 | Universite Paris-Sud | Nouveau procede de synthese d'amines tertiaires dissymetriques |
| US10414721B1 (en) | 2018-06-04 | 2019-09-17 | University Of Bern | Inhibitor of endocannabinoid cellular reuptake |
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| US5688825A (en) | 1996-05-31 | 1997-11-18 | University Of Connecticut | Anandamide amidase inhibitors as analgesic agents |
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| CA2486055A1 (en) | 2003-11-27 |
| US20040048907A1 (en) | 2004-03-11 |
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| EP1509489A1 (en) | 2005-03-02 |
| ATE516263T1 (de) | 2011-07-15 |
| KR20050012246A (ko) | 2005-01-31 |
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| US20060281742A1 (en) | 2006-12-14 |
| EP1509489A4 (en) | 2007-03-21 |
| JP2005526133A (ja) | 2005-09-02 |
| KR101087883B1 (ko) | 2011-11-30 |
| EP1509489B1 (en) | 2011-07-13 |
| US20090163593A1 (en) | 2009-06-25 |
| US7671087B2 (en) | 2010-03-02 |
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