CA2477832A1 - Methods of treating diabetes using pde 11a inhibitors - Google Patents
Methods of treating diabetes using pde 11a inhibitors Download PDFInfo
- Publication number
- CA2477832A1 CA2477832A1 CA002477832A CA2477832A CA2477832A1 CA 2477832 A1 CA2477832 A1 CA 2477832A1 CA 002477832 A CA002477832 A CA 002477832A CA 2477832 A CA2477832 A CA 2477832A CA 2477832 A1 CA2477832 A1 CA 2477832A1
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- Prior art keywords
- inhibitor
- diabetes
- pde11a
- insulin
- administering
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
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- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
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- Epidemiology (AREA)
- Urology & Nephrology (AREA)
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- Heart & Thoracic Surgery (AREA)
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- Emergency Medicine (AREA)
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- Pregnancy & Childbirth (AREA)
- Obesity (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US36469702P | 2002-03-14 | 2002-03-14 | |
| US60/364,697 | 2002-03-14 | ||
| US38903602P | 2002-06-13 | 2002-06-13 | |
| US60/389,036 | 2002-06-13 | ||
| PCT/US2003/008132 WO2003077949A2 (en) | 2002-03-14 | 2003-03-14 | Methods of treating diabetes using pde 11a inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2477832A1 true CA2477832A1 (en) | 2003-09-25 |
Family
ID=28045431
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002477832A Abandoned CA2477832A1 (en) | 2002-03-14 | 2003-03-14 | Methods of treating diabetes using pde 11a inhibitors |
Country Status (7)
| Country | Link |
|---|---|
| EP (1) | EP1496940A2 (de) |
| JP (1) | JP2005527524A (de) |
| AU (1) | AU2003220342B2 (de) |
| BR (1) | BR0308415A (de) |
| CA (1) | CA2477832A1 (de) |
| MX (1) | MXPA04008195A (de) |
| WO (1) | WO2003077949A2 (de) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2008502909A (ja) * | 2004-06-15 | 2008-01-31 | メタボレックス インコーポレーティッド | 糖尿病およびインスリン抵抗性の診断および治療の方法 |
| MEP8509A (en) | 2006-09-07 | 2011-12-20 | Combination treatment for diabetes mellitus | |
| KR101560844B1 (ko) | 2007-06-04 | 2015-10-15 | 벤-구리온 유니버시티 오브 더 네게브 리서치 앤드 디벨럽먼트 어쏘러티 | 트라이-아릴계 화합물 및 이를 포함하는 조성물 |
| EP3199203B1 (de) | 2008-02-29 | 2020-02-05 | Concert Pharmaceuticals Inc. | Substituierte xanthinderivate |
| US20110053961A1 (en) | 2009-02-27 | 2011-03-03 | Concert Pharmaceuticals, Inc. | Substituted xanthine derivatives |
| JP2012520342A (ja) * | 2009-03-16 | 2012-09-06 | ジェンメディカ・セラピューティックス・ソシエダッド・リミターダ | 代謝障害を処置するのに有用な抗炎症剤および抗酸化剤のコンジュゲート |
| WO2013013052A1 (en) | 2011-07-19 | 2013-01-24 | Concert Pharmaceuticals, Inc. | Substituted xanthine derivatives |
| JP2015067538A (ja) * | 2013-09-26 | 2015-04-13 | 株式会社アイエイアイ | 血糖値降下剤 |
| CN106061940A (zh) | 2013-11-05 | 2016-10-26 | 本古里安大学内盖夫研究发展局 | 治疗糖尿病和由其引发的并发疾病的化合物 |
| WO2015160913A1 (en) | 2014-04-18 | 2015-10-22 | Concert Pharmaceuticals, Inc. | Methods of treating hyperglycemia |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6414002B1 (en) * | 1999-09-22 | 2002-07-02 | Bristol-Myers Squibb Company | Substituted acid derivatives useful as antidiabetic and antiobesity agents and method |
| EP1297115A2 (de) * | 2000-06-26 | 2003-04-02 | Bayer Aktiengesellschaft | Regulation eines menschlichen phosphodiesterase-ähnlichen enzyms |
| EP1211313A3 (de) * | 2000-11-01 | 2003-04-23 | Pfizer Limited | Modulation der PDE11A-AKtivität |
-
2003
- 2003-03-14 MX MXPA04008195A patent/MXPA04008195A/es not_active Application Discontinuation
- 2003-03-14 BR BR0308415-9A patent/BR0308415A/pt not_active IP Right Cessation
- 2003-03-14 AU AU2003220342A patent/AU2003220342B2/en not_active Expired - Fee Related
- 2003-03-14 WO PCT/US2003/008132 patent/WO2003077949A2/en not_active Ceased
- 2003-03-14 CA CA002477832A patent/CA2477832A1/en not_active Abandoned
- 2003-03-14 JP JP2003576002A patent/JP2005527524A/ja not_active Withdrawn
- 2003-03-14 EP EP03716641A patent/EP1496940A2/de not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| WO2003077949A2 (en) | 2003-09-25 |
| WO2003077949A3 (en) | 2004-03-25 |
| AU2003220342B2 (en) | 2007-06-07 |
| AU2003220342A1 (en) | 2003-09-29 |
| EP1496940A2 (de) | 2005-01-19 |
| BR0308415A (pt) | 2005-02-15 |
| MXPA04008195A (es) | 2004-11-26 |
| JP2005527524A (ja) | 2005-09-15 |
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