CA2476630A1 - Compositions and formulations of 9-nitrocamptothecin polymorphs and methods of use thereof - Google Patents
Compositions and formulations of 9-nitrocamptothecin polymorphs and methods of use thereof Download PDFInfo
- Publication number
- CA2476630A1 CA2476630A1 CA002476630A CA2476630A CA2476630A1 CA 2476630 A1 CA2476630 A1 CA 2476630A1 CA 002476630 A CA002476630 A CA 002476630A CA 2476630 A CA2476630 A CA 2476630A CA 2476630 A1 CA2476630 A1 CA 2476630A1
- Authority
- CA
- Canada
- Prior art keywords
- nitrocamptothecin
- characterizable
- polymorph
- polymorphic form
- exotherm
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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Landscapes
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Applications Claiming Priority (13)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US10/081,745 US6482830B1 (en) | 2002-02-21 | 2002-02-21 | Compositions and formulations of 9-nitrocamptothecin polymorphs and methods of use therefor |
| US10/081,998 US6492379B1 (en) | 2002-02-21 | 2002-02-21 | Compositions and formulations of 9-nitrocamptothecin polymorphs and methods of use therefor |
| US10/082,003 | 2002-02-21 | ||
| US10/082,003 US7049322B2 (en) | 2002-02-21 | 2002-02-21 | Compositions and formulations of 9-nitrocamptothecin polymorphs and methods of use therefor |
| US10/080,530 | 2002-02-21 | ||
| US10/081,998 | 2002-02-21 | ||
| US10/081,991 | 2002-02-21 | ||
| US10/081,745 | 2002-02-21 | ||
| US10/081,991 US6756381B2 (en) | 2002-02-21 | 2002-02-21 | Compositions and formulations of 9-nitrocamptothecin polymorphs and methods of use thereof |
| US10/080,530 US7071202B2 (en) | 2002-02-21 | 2002-02-21 | Compositions and formulations of 9-nitrocamptothecin polymorphs and methods of use therefor |
| US10/267,909 US6696458B2 (en) | 2002-02-21 | 2002-10-08 | Compositions and formulations of 9-nitrocamptothecin polymorphs and methods of use thereof |
| US10/267,909 | 2002-10-08 | ||
| PCT/US2003/005118 WO2003072027A2 (en) | 2002-02-21 | 2003-02-19 | Compositions and formulations of 9- nitrocamptothecin polymorphs and methods of use thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2476630A1 true CA2476630A1 (en) | 2003-09-04 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002476630A Abandoned CA2476630A1 (en) | 2002-02-21 | 2003-02-19 | Compositions and formulations of 9-nitrocamptothecin polymorphs and methods of use thereof |
Country Status (6)
| Country | Link |
|---|---|
| US (7) | US6482830B1 (enExample) |
| EP (1) | EP1476159A4 (enExample) |
| JP (1) | JP2005520819A (enExample) |
| AU (1) | AU2003215336A1 (enExample) |
| CA (1) | CA2476630A1 (enExample) |
| WO (1) | WO2003072027A2 (enExample) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
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| WO2002068398A1 (en) * | 2001-02-27 | 2002-09-06 | Teva Pharmaceutical Industries Ltd. | New crystal forms of lamotrigine and processes for their preparations |
| US8133501B2 (en) | 2002-02-08 | 2012-03-13 | Boston Scientific Scimed, Inc. | Implantable or insertable medical devices for controlled drug delivery |
| US6887270B2 (en) | 2002-02-08 | 2005-05-03 | Boston Scientific Scimed, Inc. | Implantable or insertable medical device resistant to microbial growth and biofilm formation |
| US7993390B2 (en) * | 2002-02-08 | 2011-08-09 | Boston Scientific Scimed, Inc. | Implantable or insertable medical device resistant to microbial growth and biofilm formation |
| US8685427B2 (en) | 2002-07-31 | 2014-04-01 | Boston Scientific Scimed, Inc. | Controlled drug delivery |
| US6482830B1 (en) * | 2002-02-21 | 2002-11-19 | Supergen, Inc. | Compositions and formulations of 9-nitrocamptothecin polymorphs and methods of use therefor |
| CA2483103A1 (en) * | 2002-04-23 | 2003-11-06 | Teva Pharmaceutical Industries Ltd. | Pharmaceutical composition containing lamotrigine particles of defined morphology |
| US8920826B2 (en) | 2002-07-31 | 2014-12-30 | Boston Scientific Scimed, Inc. | Medical imaging reference devices |
| US20040121003A1 (en) * | 2002-12-19 | 2004-06-24 | Acusphere, Inc. | Methods for making pharmaceutical formulations comprising deagglomerated microparticles |
| EP1699435A4 (en) * | 2003-09-18 | 2009-05-20 | Norton Healthcare Ltd | PARTICLE |
| US20050100529A1 (en) * | 2003-11-06 | 2005-05-12 | Zeldis Jerome B. | Methods of using and compositions comprising immunomodulatory compounds for the treatment and management of asbestos-related diseases and disorders |
| AR046579A1 (es) * | 2003-11-12 | 2005-12-14 | Smithkline Beecham Corp | Compuesto cristalino de topotecan, composicion farmaceutica que lo comprende, procedimiento para prepararlo y su uso para preparar dicha composicion farmaceutica |
| CN1324032C (zh) * | 2004-01-07 | 2007-07-04 | 重庆医药工业研究院有限责任公司 | 一种新的9－硝基喜树碱晶型和药物组合物 |
| US7371906B2 (en) * | 2004-08-24 | 2008-05-13 | Eastman Kodak Company | Process for photo-oxidative stability improvements |
| ITFI20050087A1 (it) * | 2005-05-02 | 2006-11-03 | Perini Fabio Spa | Metodo e dispositivo per produrre rotoli di materiale nastriforme con una fasciatura esterna |
| IL168603A (en) * | 2005-05-16 | 2011-05-31 | Resdevco Res And Dev Co | Pharmaceutical or cosmetic composition for the prevention and treatment of irritation of mucous cells or skin cells |
| US20070123539A1 (en) * | 2005-10-20 | 2007-05-31 | University Of South Florida | Treatment of Restenosis and Stenosis with Dasatinib |
| US20070099992A1 (en) * | 2005-11-03 | 2007-05-03 | Kane Lynn C N | Direct application of vitamin C to the lung tissue and respiratory passages by use of an asthma medication-type inhaler or similar inhaler |
| US20100038816A1 (en) * | 2006-08-16 | 2010-02-18 | Novartis Ag | Method of making solid dispersions of highly crystalline therapeutic compounds |
| US8307341B2 (en) * | 2007-04-25 | 2012-11-06 | International Business Machines Corporation | Generating customized documentation for a software product |
| CN103130814B (zh) * | 2011-11-25 | 2016-03-09 | 上海医药工业研究院 | 两种9-硝基喜树碱新晶型及其制备方法 |
| GB201700555D0 (en) | 2017-01-12 | 2017-03-01 | Peptinnovate Ltd | Method for the treatment of a relapsing-remitting condition |
| US12331088B2 (en) | 2017-01-12 | 2025-06-17 | Revolo Biotherapeutics Limited | Method for the treatment of a relapsing-remitting condition |
| US12358957B2 (en) | 2017-01-12 | 2025-07-15 | Revolo Biotherapeutics Limited | Method for the acute treatment of atopic dermatitis and allergic skin hypersensitivity |
Family Cites Families (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3700819A (en) | 1970-12-07 | 1972-10-24 | Bell Telephone Labor Inc | Time division switching system with time slot interchange |
| US3883847A (en) | 1974-03-28 | 1975-05-13 | Bell Telephone Labor Inc | Uniform decoding of minimum-redundancy codes |
| JPH0763151B2 (ja) | 1985-09-18 | 1995-07-05 | 日本電気株式会社 | 可変長符号複号化回路 |
| US4894456A (en) * | 1987-03-31 | 1990-01-16 | Research Triangle Institute | Synthesis of camptothecin and analogs thereof |
| US4981968A (en) * | 1987-03-31 | 1991-01-01 | Research Triangle Institute | Synthesis of camptothecin and analogs thereof |
| US5552154A (en) * | 1989-11-06 | 1996-09-03 | The Stehlin Foundation For Cancer Research | Method for treating cancer with water-insoluble s-camptothecin of the closed lactone ring form and derivatives thereof |
| US5225404A (en) * | 1989-11-06 | 1993-07-06 | New York University | Methods of treating colon tumors with tumor-inhibiting camptothecin compounds |
| US5162532A (en) * | 1990-12-20 | 1992-11-10 | North Carolina State University | Intermediates and method of making camptothecin and camptothecin analogs |
| US5559235A (en) * | 1991-10-29 | 1996-09-24 | Glaxo Wellcome Inc. | Water soluble camptothecin derivatives |
| JPH05152973A (ja) | 1991-11-28 | 1993-06-18 | Fujitsu Ltd | 可変長符号復号器 |
| JPH05173844A (ja) | 1991-12-19 | 1993-07-13 | Nec Corp | コーディングミス修正方式 |
| JP2842094B2 (ja) | 1992-10-13 | 1998-12-24 | 日本電気株式会社 | ハフマン復号回路 |
| GB9319944D0 (en) * | 1993-09-28 | 1993-11-17 | Erba Carlo Spa | Process for the preparation of 9-amino camptothecin |
| US5731316A (en) * | 1996-01-30 | 1998-03-24 | The Stehlin Foundation For Cancer Research | Derivatives of camptothecin and methods of treating cancer using these derivatives |
| US6096336A (en) * | 1996-01-30 | 2000-08-01 | The Stehlin Foundation For Cancer Research | Liposomal prodrugs comprising derivatives of camptothecin and methods of treating cancer using these prodrugs |
| JPH09307456A (ja) | 1996-05-09 | 1997-11-28 | Matsushita Electric Ind Co Ltd | 可変長符号復号装置及び方法 |
| US5922877A (en) * | 1997-08-05 | 1999-07-13 | The Stehlin Foundation For Cancer Research | Methods of preparing and purifying 9-nitro-20-camptothecin |
| JPH11168391A (ja) | 1997-12-04 | 1999-06-22 | Matsushita Electric Ind Co Ltd | 復号装置 |
| US6291676B1 (en) | 1999-03-03 | 2001-09-18 | University Of Kentucky Research Foundation | Water-soluble derivatives of camptothecin/homocamptothecin |
| US6288072B1 (en) * | 1999-12-29 | 2001-09-11 | Monroe E. Wall | Camptothecin β-alanine esters with topoisomerase I inhibition |
| AU2001240024A1 (en) * | 2000-03-31 | 2001-10-15 | Supergen, Inc. | Camptothecin complexes |
| US6482830B1 (en) * | 2002-02-21 | 2002-11-19 | Supergen, Inc. | Compositions and formulations of 9-nitrocamptothecin polymorphs and methods of use therefor |
-
2002
- 2002-02-21 US US10/081,745 patent/US6482830B1/en not_active Expired - Fee Related
- 2002-02-21 US US10/081,998 patent/US6492379B1/en not_active Expired - Fee Related
- 2002-02-21 US US10/081,991 patent/US6756381B2/en not_active Expired - Fee Related
- 2002-02-21 US US10/080,530 patent/US7071202B2/en not_active Expired - Fee Related
- 2002-02-21 US US10/082,003 patent/US7049322B2/en not_active Expired - Fee Related
- 2002-10-08 US US10/267,909 patent/US6696458B2/en not_active Expired - Fee Related
-
2003
- 2003-02-19 CA CA002476630A patent/CA2476630A1/en not_active Abandoned
- 2003-02-19 AU AU2003215336A patent/AU2003215336A1/en not_active Abandoned
- 2003-02-19 JP JP2003570774A patent/JP2005520819A/ja not_active Abandoned
- 2003-02-19 WO PCT/US2003/005118 patent/WO2003072027A2/en not_active Ceased
- 2003-02-19 EP EP03711157A patent/EP1476159A4/en not_active Withdrawn
-
2006
- 2006-03-28 US US11/277,729 patent/US20060217407A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| US20030166671A1 (en) | 2003-09-04 |
| WO2003072027A2 (en) | 2003-09-04 |
| AU2003215336A1 (en) | 2003-09-09 |
| WO2003072027A3 (en) | 2004-06-10 |
| US20060217407A1 (en) | 2006-09-28 |
| JP2005520819A (ja) | 2005-07-14 |
| US6482830B1 (en) | 2002-11-19 |
| US7049322B2 (en) | 2006-05-23 |
| US20030181476A1 (en) | 2003-09-25 |
| US6696458B2 (en) | 2004-02-24 |
| US7071202B2 (en) | 2006-07-04 |
| US6492379B1 (en) | 2002-12-10 |
| US20030181477A1 (en) | 2003-09-25 |
| EP1476159A4 (en) | 2006-03-01 |
| US20030176453A1 (en) | 2003-09-18 |
| US6756381B2 (en) | 2004-06-29 |
| EP1476159A2 (en) | 2004-11-17 |
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