CA2464217A1 - Antimuscarinic aerosol - Google Patents
Antimuscarinic aerosol Download PDFInfo
- Publication number
- CA2464217A1 CA2464217A1 CA002464217A CA2464217A CA2464217A1 CA 2464217 A1 CA2464217 A1 CA 2464217A1 CA 002464217 A CA002464217 A CA 002464217A CA 2464217 A CA2464217 A CA 2464217A CA 2464217 A1 CA2464217 A1 CA 2464217A1
- Authority
- CA
- Canada
- Prior art keywords
- tolterodine
- antimuscarinic agent
- group
- inhalably
- antimuscarinic
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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- 230000001022 anti-muscarinic effect Effects 0.000 title description 4
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- 230000002485 urinary effect Effects 0.000 claims abstract description 33
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/0078—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a nebulizer such as a jet nebulizer, ultrasonic nebulizer, e.g. in the form of aqueous drug solutions or dispersions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/215—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
- A61K31/216—Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids of acids having aromatic rings, e.g. benactizyne, clofibrate
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Emergency Medicine (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Urology & Nephrology (AREA)
- Dispersion Chemistry (AREA)
- Otolaryngology (AREA)
- Pulmonology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US33729801P | 2001-11-05 | 2001-11-05 | |
| US60/337,298 | 2001-11-05 | ||
| PCT/US2002/035335 WO2003039464A2 (en) | 2001-11-05 | 2002-11-04 | Antimuscarinic aerosol |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2464217A1 true CA2464217A1 (en) | 2003-05-15 |
Family
ID=23319948
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002464217A Abandoned CA2464217A1 (en) | 2001-11-05 | 2002-11-04 | Antimuscarinic aerosol |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20030144352A1 (enExample) |
| EP (1) | EP1441706A2 (enExample) |
| JP (1) | JP2005511582A (enExample) |
| AU (1) | AU2002342313A1 (enExample) |
| BR (1) | BR0206300A (enExample) |
| CA (1) | CA2464217A1 (enExample) |
| MX (1) | MXPA04003806A (enExample) |
| NO (1) | NO20033079D0 (enExample) |
| TW (1) | TW200300079A (enExample) |
| WO (1) | WO2003039464A2 (enExample) |
Families Citing this family (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0957073A1 (en) | 1998-05-12 | 1999-11-17 | Schwarz Pharma Ag | Novel derivatives of 3,3-diphenylpropylamines |
| US6974820B2 (en) * | 2002-11-06 | 2005-12-13 | Bridge Pharma, Inc. | Methods for treating urinary incontinence and other disorders using trospium |
| EP1424079A1 (en) * | 2002-11-27 | 2004-06-02 | Boehringer Ingelheim International GmbH | Combination of a beta-3-receptor agonist and of a reuptake inhibitor of serotonin and/or norepinephrine |
| DE10315917A1 (de) * | 2003-04-08 | 2004-11-18 | Schwarz Pharma Ag | Hochreine Basen von 3,3-Diphenylpropylaminmonoestern |
| US20060287347A1 (en) * | 2005-06-21 | 2006-12-21 | Aberg A K G | Methods for treating smooth muscle disorders using trospium |
| US7390816B2 (en) * | 2005-06-21 | 2008-06-24 | Bridge Pharma, Inc. | Methods for treating urinary incontinence in patients suffering from memory disorders |
| US20070004766A1 (en) * | 2005-07-01 | 2007-01-04 | Aberg A K G | Methods for relaxation of smooth muscle contractions using Trospium |
| US9119777B2 (en) | 2008-05-30 | 2015-09-01 | Microdose Therapeutx, Inc. | Methods and compositions for administration of oxybutynin |
| US8415390B2 (en) | 2008-05-30 | 2013-04-09 | Microdose Therapeutx, Inc. | Methods and compositions for administration of oxybutynin |
| CA2859004A1 (en) * | 2007-05-30 | 2008-12-11 | Microdose Therapeutx, Inc. | Methods and compositions for administration of oxybutynin |
| US20100297225A1 (en) * | 2007-12-20 | 2010-11-25 | Pharmathen S.A. | Sustained-release pharmaceutical formulation containing an antimuscarinic agent and a wetting agent as well as a process for the preparation thereof |
| US9180263B2 (en) | 2009-07-01 | 2015-11-10 | Microdose Therapeutx, Inc. | Laboratory animal pulmonary dosing device |
| JP6017961B2 (ja) | 2010-01-05 | 2016-11-02 | マイクロドース セラピューテクス，インコーポレイテッド | 吸入デバイスおよび方法 |
| GB201402556D0 (en) * | 2014-02-13 | 2014-04-02 | Crystec Ltd | Improvements relating to inhalable particles |
| WO2018071427A1 (en) | 2016-10-11 | 2018-04-19 | Microdose Therapeutx, Inc. | Inhaler and methods of use thereof |
Family Cites Families (15)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL6717123A (enExample) * | 1966-12-29 | 1968-07-01 | ||
| US3505337A (en) * | 1967-12-22 | 1970-04-07 | Boehringer Sohn Ingelheim | N - hydrocarbyl-substituted noratropinium,haloalkylates and o-acyl derivatives thereof |
| US5736577A (en) * | 1995-01-31 | 1998-04-07 | Sepracor, Inc. | Methods and compositions for treating urinary incontinence using optically pure (S)-oxybutynin |
| SE8800207D0 (sv) * | 1988-01-22 | 1988-01-22 | Kabivitrum Ab | Nya aminer, deras anvendning och framstellning |
| US5382600A (en) * | 1988-01-22 | 1995-01-17 | Pharmacia Aktiebolag | 3,3-diphenylpropylamines and pharmaceutical compositions thereof |
| IL91377A (en) * | 1988-09-14 | 1996-09-12 | Nippon Shinyaku Co Ltd | Derivatives of botinylamine glycolate |
| GB8906166D0 (en) * | 1989-03-17 | 1989-05-04 | Pfizer Ltd | Therapeutic agents |
| SE9203318D0 (sv) * | 1992-11-06 | 1992-11-06 | Kabi Pharmacia Ab | Novel 3,3-diphenylpropylamines, their use and preparation |
| US5677346A (en) * | 1995-01-31 | 1997-10-14 | Sepracor, Inc. | Treating urinary incontinence using (S)-desethyloxybutynin |
| AU728395B2 (en) * | 1996-07-19 | 2001-01-11 | Gunnar Aberg | S(-)-tolterodine in the treatment of urinary and gastrointestinal disorders |
| US6124354A (en) * | 1996-07-29 | 2000-09-26 | Pharmacia & Upjohn Ab | Arylcycloalkane carboxylic esters, their use, pharmaceutical compositions and preparation |
| US6383471B1 (en) * | 1999-04-06 | 2002-05-07 | Lipocine, Inc. | Compositions and methods for improved delivery of ionizable hydrophobic therapeutic agents |
| US6545046B2 (en) * | 2000-08-30 | 2003-04-08 | Theramax Inc. | Method for enhanced delivery of oxybutynin and compositions thereof |
| PE20020547A1 (es) * | 2000-10-24 | 2002-06-12 | Upjohn Co | Uso de la tolterodina en tratamientos del asma |
| US20030027856A1 (en) * | 2001-06-29 | 2003-02-06 | Aberg A.K. Gunnar | Tolterodine metabolites |
-
2002
- 2002-11-04 TW TW091132481A patent/TW200300079A/zh unknown
- 2002-11-04 JP JP2003541756A patent/JP2005511582A/ja not_active Withdrawn
- 2002-11-04 BR BRPI0206300-0A patent/BR0206300A/pt not_active IP Right Cessation
- 2002-11-04 MX MXPA04003806A patent/MXPA04003806A/es unknown
- 2002-11-04 EP EP02776444A patent/EP1441706A2/en not_active Withdrawn
- 2002-11-04 CA CA002464217A patent/CA2464217A1/en not_active Abandoned
- 2002-11-04 US US10/287,061 patent/US20030144352A1/en not_active Abandoned
- 2002-11-04 WO PCT/US2002/035335 patent/WO2003039464A2/en not_active Ceased
- 2002-11-04 AU AU2002342313A patent/AU2002342313A1/en not_active Abandoned
-
2003
- 2003-07-04 NO NO20033079A patent/NO20033079D0/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BR0206300A (pt) | 2008-04-08 |
| AU2002342313A1 (en) | 2003-05-19 |
| WO2003039464A3 (en) | 2004-02-26 |
| EP1441706A2 (en) | 2004-08-04 |
| TW200300079A (en) | 2003-05-16 |
| MXPA04003806A (es) | 2005-04-08 |
| JP2005511582A (ja) | 2005-04-28 |
| NO20033079D0 (no) | 2003-07-04 |
| WO2003039464A2 (en) | 2003-05-15 |
| US20030144352A1 (en) | 2003-07-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request | ||
| FZDE | Discontinued |