CA2463675C - Cyclic peptides as g-protein-coupled receptor antagonists - Google Patents
Cyclic peptides as g-protein-coupled receptor antagonists Download PDFInfo
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- CA2463675C CA2463675C CA2463675A CA2463675A CA2463675C CA 2463675 C CA2463675 C CA 2463675C CA 2463675 A CA2463675 A CA 2463675A CA 2463675 A CA2463675 A CA 2463675A CA 2463675 C CA2463675 C CA 2463675C
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- C07K7/56—Cyclic peptides containing at least one abnormal peptide link with at least one abnormal peptide link in the ring the cyclisation not occurring through 2,4-diamino-butanoic acid
Landscapes
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Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AUPR8334A AUPR833401A0 (en) | 2001-10-17 | 2001-10-17 | G protein-coupled receptor antagonists |
| AUPR8334 | 2001-10-17 | ||
| PCT/AU2002/001427 WO2003033528A1 (en) | 2001-10-17 | 2002-10-17 | Cyclic peptides as g-protein-coupled receptor antagonists |
Publications (2)
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| CA2463675A1 CA2463675A1 (en) | 2003-04-24 |
| CA2463675C true CA2463675C (en) | 2012-08-07 |
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| CA2463675A Expired - Fee Related CA2463675C (en) | 2001-10-17 | 2002-10-17 | Cyclic peptides as g-protein-coupled receptor antagonists |
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| US (3) | US7579432B2 (enExample) |
| EP (1) | EP1444251A4 (enExample) |
| JP (1) | JP2005515973A (enExample) |
| CN (2) | CN1604909A (enExample) |
| AU (2) | AUPR833401A0 (enExample) |
| CA (1) | CA2463675C (enExample) |
| WO (1) | WO2003033528A1 (enExample) |
Families Citing this family (34)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AUPO755097A0 (en) | 1997-06-25 | 1997-07-17 | University Of Queensland, The | Receptor agonist and antagonist |
| AUPR833401A0 (en) * | 2001-10-17 | 2001-11-08 | University Of Queensland, The | G protein-coupled receptor antagonists |
| AUPS160602A0 (en) | 2002-04-08 | 2002-05-16 | University Of Queensland, The | Therapeutic method |
| AU2002952086A0 (en) * | 2002-10-16 | 2002-11-07 | The University Of Queensland | Treatment of osteoarthritis |
| CA2542507C (en) * | 2002-10-16 | 2013-04-16 | The University Of Queensland | Treatment of inflammatory bowel disease |
| AU2002952129A0 (en) * | 2002-10-17 | 2002-10-31 | The University Of Queensland | Treatment of hypersensitivity conditions |
| AU2003902586A0 (en) * | 2003-05-26 | 2003-06-12 | The University Of Queensland | Treatment of burns |
| EP1498422A1 (de) * | 2003-07-17 | 2005-01-19 | Jerini AG | C5a-Rezeptor-Antagonisten |
| MXPA06011051A (es) * | 2004-03-26 | 2007-04-13 | Promics Pty Ltd | Tratamiento de condiciones neurologicas usando complemento de moduladores del receptor c5a. |
| WO2006074964A1 (en) * | 2005-01-17 | 2006-07-20 | Jerini Ag | C5a receptor antagonists |
| EP1739078A1 (de) | 2005-05-30 | 2007-01-03 | Jerini AG | C5a-Rezeptor-Antagonisten |
| CN101553244B (zh) * | 2006-07-21 | 2013-01-02 | 普罗米克斯有限公司 | 内膜增生和相关病状的治疗 |
| WO2008153962A2 (en) * | 2007-06-08 | 2008-12-18 | The Trustees Of The University Of Pennylvania | Method of reducing tissue loss in pancreatic islet cell transplantation |
| US8563259B2 (en) * | 2007-06-29 | 2013-10-22 | The Trustees Of The University Of Pennsylvania | Complement-mediated thrombophilic assay |
| US20110142837A1 (en) * | 2007-07-20 | 2011-06-16 | Trustees Of The University Of Pennsylvania | Method Of Treating Acute Respiratory Distress Syndrome |
| US10632170B2 (en) * | 2008-02-19 | 2020-04-28 | The Trustees Of The University Of Pennsylvania | Administration of compstatin to an individual for the treatment of a tumor |
| EP2331113A4 (en) * | 2008-08-20 | 2012-03-14 | Univ Pennsylvania | COMPLEMENTARY TREATMENT FOR THE TREATMENT OF LESIONS DUE TO BRAIN BLEEDING |
| US8445190B2 (en) | 2008-09-30 | 2013-05-21 | The Trustees Of The University Of Pennsylvania | Method of inhibiting biomaterial-induced procoagulant activity using complement inhibitors |
| US9358266B2 (en) | 2010-02-25 | 2016-06-07 | The Trustees Of The University Of Pennsylvania | Treatment of sepsis using complement inhibitors |
| US20140219999A1 (en) | 2011-04-01 | 2014-08-07 | The Trustees Of The University Of Pennsylvania | Treatment of colon cancer using complement inhibitors |
| WO2012162215A1 (en) | 2011-05-20 | 2012-11-29 | The Trustees Of The University Of Pennsylvania | Promotion of fracture healing using complement inhibitors |
| WO2012174055A1 (en) | 2011-06-13 | 2012-12-20 | The Trustees Of The University Of Pennsylvania | Wound healing using complement inhibitors |
| WO2015103438A2 (en) | 2014-01-02 | 2015-07-09 | Genelux Corporation | Oncolytic virus adjunct therapy with agents that increase virus infectivity |
| US20200325449A1 (en) | 2016-06-02 | 2020-10-15 | The Cleveland Clinic Foundation | Complement inhibition for improving cell viability |
| JP2019532021A (ja) * | 2016-07-29 | 2019-11-07 | ファイザー・インク | Ｃ５ａ受容体アンタゴニストとしての環状ペプチド |
| US10376595B2 (en) | 2017-04-03 | 2019-08-13 | Inflarx Gmbh | Treatment of inflammatory diseases with inhibitors of C5a activity |
| ES2893769T3 (es) | 2017-04-03 | 2022-02-10 | Inflarx Gmbh | Tratamiento de enfermedades inflamatorias con inhibidores de la actividad de C5a |
| CN111201241A (zh) * | 2017-06-23 | 2020-05-26 | 因弗拉克斯有限责任公司 | 用C5a活性抑制剂治疗炎性疾病 |
| SG10201902000YA (en) * | 2019-03-06 | 2020-10-29 | Nat Univ Singapore | Isthmin 1 for treatment of lung inflammation |
| IL296036A (en) | 2020-03-27 | 2022-10-01 | Inflarx Gmbh | Inhibitors of c5a for the treatment of corona virus infection |
| FR3112941B1 (fr) * | 2020-07-30 | 2023-03-03 | Sederma Sa | Traitement cosmétique ou dermatologique à base de peptide(s) de la peau et de ses phanères |
| JP2023117892A (ja) * | 2022-02-14 | 2023-08-24 | 公益財団法人 鷹揚郷 | ヘプシジン結合ペプチド |
| CN116311497A (zh) * | 2023-02-02 | 2023-06-23 | 山东大学 | 一种基于机器视觉的隧道工人异常行为检测方法及系统 |
| US12180274B2 (en) | 2023-05-26 | 2024-12-31 | Inflarx Gmbh | Treatment of pneumonia and ARDS with inhibitors of C5a and IL-6 activity |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5807824A (en) * | 1993-12-06 | 1998-09-15 | Ciba-Geigy Corporation | C5A receptor antagonists having substantially no agonist activity |
| AUPO755097A0 (en) * | 1997-06-25 | 1997-07-17 | University Of Queensland, The | Receptor agonist and antagonist |
| AUPR833401A0 (en) * | 2001-10-17 | 2001-11-08 | University Of Queensland, The | G protein-coupled receptor antagonists |
-
2001
- 2001-10-17 AU AUPR8334A patent/AUPR833401A0/en not_active Abandoned
-
2002
- 2002-10-17 US US10/493,117 patent/US7579432B2/en not_active Expired - Fee Related
- 2002-10-17 JP JP2003536266A patent/JP2005515973A/ja active Pending
- 2002-10-17 EP EP02771873A patent/EP1444251A4/en not_active Withdrawn
- 2002-10-17 CN CNA028252578A patent/CN1604909A/zh active Pending
- 2002-10-17 CN CN2006100067952A patent/CN1847261B/zh not_active Expired - Fee Related
- 2002-10-17 WO PCT/AU2002/001427 patent/WO2003033528A1/en not_active Ceased
- 2002-10-17 CA CA2463675A patent/CA2463675C/en not_active Expired - Fee Related
- 2002-10-17 AU AU2002336783A patent/AU2002336783B2/en not_active Ceased
-
2009
- 2009-07-14 US US12/502,937 patent/US20100331236A1/en not_active Abandoned
-
2012
- 2012-02-02 US US13/365,013 patent/US20120302493A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| AUPR833401A0 (en) | 2001-11-08 |
| US20100331236A1 (en) | 2010-12-30 |
| AU2002336783B2 (en) | 2008-11-06 |
| CN1604909A (zh) | 2005-04-06 |
| EP1444251A1 (en) | 2004-08-11 |
| CA2463675A1 (en) | 2003-04-24 |
| EP1444251A4 (en) | 2005-12-21 |
| JP2005515973A (ja) | 2005-06-02 |
| US20120302493A1 (en) | 2012-11-29 |
| CN1847261A (zh) | 2006-10-18 |
| US20060217530A1 (en) | 2006-09-28 |
| US7579432B2 (en) | 2009-08-25 |
| WO2003033528A1 (en) | 2003-04-24 |
| CN1847261B (zh) | 2010-12-01 |
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| EEER | Examination request | ||
| MKLA | Lapsed |
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