CA2432908A1 - Diamines as modulators of chemokine receptor activity - Google Patents

Diamines as modulators of chemokine receptor activity Download PDF

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Publication number
CA2432908A1
CA2432908A1 CA002432908A CA2432908A CA2432908A1 CA 2432908 A1 CA2432908 A1 CA 2432908A1 CA 002432908 A CA002432908 A CA 002432908A CA 2432908 A CA2432908 A CA 2432908A CA 2432908 A1 CA2432908 A1 CA 2432908A1
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Prior art keywords
amino
methyl
substituted
crr
trifluoromethyl
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Abandoned
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CA002432908A
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English (en)
French (fr)
Inventor
Percy Carter
Robert Cherney
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Bristol Myers Squibb Pharma Co
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Individual
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    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/63—One oxygen atom
    • C07D213/64—One oxygen atom attached in position 2 or 6
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    • C07C237/22—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by amino groups having the carbon atoms of the carboxamide groups bound to acyclic carbon atoms of the carbon skeleton having nitrogen atoms of amino groups bound to the carbon skeleton of the acid part, further acylated
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CA002432908A 2000-12-20 2001-12-20 Diamines as modulators of chemokine receptor activity Abandoned CA2432908A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US25685500P 2000-12-20 2000-12-20
US60/256,855 2000-12-20
PCT/US2001/050619 WO2002050019A2 (en) 2000-12-20 2001-12-20 Diamines as modulators of chemokine receptor activity

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CA2432908A1 true CA2432908A1 (en) 2002-06-27

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CA002432908A Abandoned CA2432908A1 (en) 2000-12-20 2001-12-20 Diamines as modulators of chemokine receptor activity

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