CA2420012A1 - Derives d'erythromycine substitue en 6-o possedant une tolerance gastro-intestinale amelioree - Google Patents
Derives d'erythromycine substitue en 6-o possedant une tolerance gastro-intestinale amelioree Download PDFInfo
- Publication number
- CA2420012A1 CA2420012A1 CA002420012A CA2420012A CA2420012A1 CA 2420012 A1 CA2420012 A1 CA 2420012A1 CA 002420012 A CA002420012 A CA 002420012A CA 2420012 A CA2420012 A CA 2420012A CA 2420012 A1 CA2420012 A1 CA 2420012A1
- Authority
- CA
- Canada
- Prior art keywords
- hydrogen
- formula
- compound
- diyl
- isoxazol
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- Communicable Diseases (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Abstract
L'invention concerne des composés de formule (I) qui sont utiles dans le traitement des infections bactériennes et permettent d'éviter tout risque concomitant d'intolérance gastro-intestinale. L'invention concerne également des compositions contenant lesdits composés et des méthodes de traitement utilisant ces composés.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US24077700P | 2000-10-16 | 2000-10-16 | |
US60/240,777 | 2000-10-16 | ||
PCT/US2001/032278 WO2002032919A2 (fr) | 2000-10-16 | 2001-10-16 | Derives d'erythromycine substitue en 6-o possedant une tolerance gastro-intestinale amelioree |
Publications (1)
Publication Number | Publication Date |
---|---|
CA2420012A1 true CA2420012A1 (fr) | 2002-04-25 |
Family
ID=22907903
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002420012A Abandoned CA2420012A1 (fr) | 2000-10-16 | 2001-10-16 | Derives d'erythromycine substitue en 6-o possedant une tolerance gastro-intestinale amelioree |
Country Status (9)
Country | Link |
---|---|
EP (1) | EP1328534A2 (fr) |
JP (1) | JP2004529857A (fr) |
AU (1) | AU2002213267A1 (fr) |
BR (1) | BR0109946A (fr) |
CA (1) | CA2420012A1 (fr) |
MX (1) | MXPA03003311A (fr) |
PE (1) | PE20020522A1 (fr) |
UY (1) | UY26964A1 (fr) |
WO (1) | WO2002032919A2 (fr) |
Families Citing this family (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
NZ533282A (en) | 2001-12-05 | 2006-09-29 | Ortho Mcneil Pharm Inc | 6-O-Acyl ketolide derivatives of erythromycine useful as antibacterials |
MXPA04010802A (es) * | 2002-04-30 | 2005-03-07 | Abbott Lab | Compuestos antibacterianos con perfiles farmacocineticos mejorados. |
US6727229B2 (en) * | 2002-08-19 | 2004-04-27 | Enanta Pharmaceuticals, Inc. | 11,12-substituted lactone ketolide derivatives having antibacterial activity |
JPWO2004078771A1 (ja) * | 2003-03-07 | 2006-06-08 | 大正製薬株式会社 | 2−フルオロ−6−o−置換ケトライド誘導体 |
JP2007223900A (ja) * | 2004-02-03 | 2007-09-06 | Taisho Pharmaceut Co Ltd | 6−o−置換ケトライド誘導体 |
JP2007254285A (ja) * | 2004-03-16 | 2007-10-04 | Taisho Pharmaceut Co Ltd | 2−フルオロ−6−o−置換ケトライド誘導体 |
JP5015016B2 (ja) | 2006-02-07 | 2012-08-29 | 大正製薬株式会社 | 10a−アザライド化合物 |
EP2177526A4 (fr) | 2007-08-06 | 2012-08-22 | Taisho Pharmaceutical Co Ltd | Composé 10a-azalide réticulé en position 10a et en position 12 |
US8299035B2 (en) | 2008-05-15 | 2012-10-30 | Taisho Pharmaceutucal Co., Ltd. | 10a-azalide compound having 4-membered ring structure |
CN102234302B (zh) * | 2010-05-07 | 2014-05-07 | 北京理工大学 | 一种酮内酯衍生物、制备方法及其药物组合物 |
AR085286A1 (es) | 2011-02-21 | 2013-09-18 | Taisho Pharmaceutical Co Ltd | Derivado de macrolido sustituido en la posicion c-4 |
AR102810A1 (es) | 2014-08-18 | 2017-03-29 | Taisho Pharmaceutical Co Ltd | Derivado de macrólido sustituido en la posición c-4 |
Family Cites Families (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6054435A (en) * | 1999-03-19 | 2000-04-25 | Abbott Laboratories | 6-O-substituted macrolides having antibacterial activity |
-
2001
- 2001-10-12 UY UY26964A patent/UY26964A1/es not_active Application Discontinuation
- 2001-10-15 PE PE2001001021A patent/PE20020522A1/es not_active Application Discontinuation
- 2001-10-16 CA CA002420012A patent/CA2420012A1/fr not_active Abandoned
- 2001-10-16 BR BR0109946-9A patent/BR0109946A/pt not_active Application Discontinuation
- 2001-10-16 JP JP2002536300A patent/JP2004529857A/ja not_active Withdrawn
- 2001-10-16 AU AU2002213267A patent/AU2002213267A1/en not_active Abandoned
- 2001-10-16 EP EP01981637A patent/EP1328534A2/fr not_active Withdrawn
- 2001-10-16 WO PCT/US2001/032278 patent/WO2002032919A2/fr not_active Application Discontinuation
- 2001-10-16 MX MXPA03003311A patent/MXPA03003311A/es unknown
Also Published As
Publication number | Publication date |
---|---|
BR0109946A (pt) | 2005-08-02 |
UY26964A1 (es) | 2002-06-20 |
WO2002032919A3 (fr) | 2002-09-19 |
AU2002213267A1 (en) | 2002-04-29 |
MXPA03003311A (es) | 2003-09-10 |
WO2002032919A2 (fr) | 2002-04-25 |
EP1328534A2 (fr) | 2003-07-23 |
PE20020522A1 (es) | 2002-06-25 |
JP2004529857A (ja) | 2004-09-30 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FZDE | Dead |