CA2405689A1 - Analogues peptidiques vasoactifs intestinaux - Google Patents

Analogues peptidiques vasoactifs intestinaux Download PDF

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Publication number
CA2405689A1
CA2405689A1 CA002405689A CA2405689A CA2405689A1 CA 2405689 A1 CA2405689 A1 CA 2405689A1 CA 002405689 A CA002405689 A CA 002405689A CA 2405689 A CA2405689 A CA 2405689A CA 2405689 A1 CA2405689 A1 CA 2405689A1
Authority
CA
Canada
Prior art keywords
leu
asn
lys
peptide
tyr
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002405689A
Other languages
English (en)
Inventor
Anand C. Burman
Sudhanand Prasad
Rama Mukherjee
Anu T. Singh
Archna Mathur
Neena Gupta
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Dabur Research Foundation
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Priority claimed from PCT/US2000/020871 external-priority patent/WO2001060862A1/fr
Publication of CA2405689A1 publication Critical patent/CA2405689A1/fr
Abandoned legal-status Critical Current

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  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

L'invention concerne de nouveaux analogues peptidiques vasoactifs intestinaux (VIP) contenant des substitutions au niveau des acides aminés convenablement sélectionnés. L'invention concerne plus particulièrement la conception et la synthèse de nouveaux analogues VIP biologiquement actifs contenant des acides aminés .alpha., .alpha.-dialkylés de manière spécifique au site. L'invention concerne plus concrètement la synthèse de dérivés peptidiques VIP qui se lient de manière sélective aux récepteurs VIP sur les cellules cibles. L'invention concerne en outre des procédés permettant l'obtention de ces peptides et de compositions contenant les peptides ainsi que leurs applications pharmacologiques surtout dans le traitement et la prévention du cancer.
CA002405689A 2000-02-18 2000-07-31 Analogues peptidiques vasoactifs intestinaux Abandoned CA2405689A1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
IN136DE2000 2000-02-18
IN136/DEL/2000 2000-02-18
PCT/US2000/020871 WO2001060862A1 (fr) 2000-02-18 2000-07-31 Analogues peptidiques vasoactifs intestinaux

Publications (1)

Publication Number Publication Date
CA2405689A1 true CA2405689A1 (fr) 2001-08-23

Family

ID=11097028

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002405689A Abandoned CA2405689A1 (fr) 2000-02-18 2000-07-31 Analogues peptidiques vasoactifs intestinaux

Country Status (3)

Country Link
AT (1) ATE276273T1 (fr)
CA (1) CA2405689A1 (fr)
DE (1) DE60013912T2 (fr)

Also Published As

Publication number Publication date
DE60013912D1 (de) 2004-10-21
ATE276273T1 (de) 2004-10-15
DE60013912T2 (de) 2005-09-29

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Legal Events

Date Code Title Description
EEER Examination request
FZDE Discontinued