CA2391646A1 - Solid preparation - Google Patents

Solid preparation Download PDF

Info

Publication number
CA2391646A1
CA2391646A1 CA002391646A CA2391646A CA2391646A1 CA 2391646 A1 CA2391646 A1 CA 2391646A1 CA 002391646 A CA002391646 A CA 002391646A CA 2391646 A CA2391646 A CA 2391646A CA 2391646 A1 CA2391646 A1 CA 2391646A1
Authority
CA
Canada
Prior art keywords
compound
crystal
drug substance
granules
set forth
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002391646A
Other languages
English (en)
French (fr)
Inventor
Motokazu Iwata
Teruaki Kuriyama
Megumi Fujita
Keiichi Fujiwara
Shiro Kato
Hiroshi Harada
Akihito Fujii
Osamu Odai
Hitoshi Kawashima
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Dainippon Pharmaceutical Co Ltd
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US09/661,577 external-priority patent/US6458824B1/en
Application filed by Individual filed Critical Individual
Publication of CA2391646A1 publication Critical patent/CA2391646A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/14—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
    • C07D209/16—Tryptamines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Indole Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CA002391646A 1999-11-30 2000-11-24 Solid preparation Abandoned CA2391646A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP33954799 1999-11-30
JP11/339547 1999-11-30
US09/661,577 US6458824B1 (en) 1999-11-30 2000-09-14 Solid preparation
US09/661,577 2000-09-14
PCT/JP2000/008283 WO2001040182A2 (en) 1999-11-30 2000-11-24 Solid pharmaceutical preparation

Publications (1)

Publication Number Publication Date
CA2391646A1 true CA2391646A1 (en) 2001-06-07

Family

ID=26576443

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002391646A Abandoned CA2391646A1 (en) 1999-11-30 2000-11-24 Solid preparation

Country Status (14)

Country Link
EP (1) EP1235801A2 (no)
JP (1) JP2003515587A (no)
CN (1) CN1433403A (no)
AU (1) AU1550501A (no)
CA (1) CA2391646A1 (no)
CZ (1) CZ20021833A3 (no)
HU (1) HUP0203865A3 (no)
IL (1) IL149635A0 (no)
MX (1) MXPA02005326A (no)
NO (1) NO20022541L (no)
NZ (1) NZ519086A (no)
PL (1) PL356468A1 (no)
SK (1) SK7362002A3 (no)
WO (1) WO2001040182A2 (no)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR20050010512A (ko) * 2002-06-12 2005-01-27 스미또모 세이야꾸 가부시키가이샤 인돌, 인다졸 및 벤즈아졸류
JP3759949B2 (ja) * 2002-12-17 2006-03-29 湧永製薬株式会社 遮光剤及び皮膜組成物
LT3366283T (lt) * 2004-01-20 2021-12-10 Novartis Ag Tiesioginio presavimo formulė ir procesas

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1070477C (zh) * 1994-11-29 2001-09-05 大日本制药株式会社 吲哚衍生物
JPH11255743A (ja) * 1998-03-06 1999-09-21 Dainippon Pharmaceut Co Ltd 光学活性のインドール誘導体の製造方法及びその製造中間体

Also Published As

Publication number Publication date
NZ519086A (en) 2003-11-28
HUP0203865A3 (en) 2004-05-28
CZ20021833A3 (cs) 2003-02-12
NO20022541D0 (no) 2002-05-29
HUP0203865A2 (hu) 2003-03-28
WO2001040182A3 (en) 2002-06-27
IL149635A0 (en) 2002-11-10
JP2003515587A (ja) 2003-05-07
SK7362002A3 (en) 2003-02-04
NO20022541L (no) 2002-07-29
PL356468A1 (en) 2004-06-28
MXPA02005326A (es) 2003-02-12
WO2001040182A2 (en) 2001-06-07
CN1433403A (zh) 2003-07-30
EP1235801A2 (en) 2002-09-04
AU1550501A (en) 2001-06-12

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Legal Events

Date Code Title Description
FZDE Discontinued