CA2272927C - Dimesylate salts of neuropeptide y ligands - Google Patents
Dimesylate salts of neuropeptide y ligands Download PDFInfo
- Publication number
- CA2272927C CA2272927C CA002272927A CA2272927A CA2272927C CA 2272927 C CA2272927 C CA 2272927C CA 002272927 A CA002272927 A CA 002272927A CA 2272927 A CA2272927 A CA 2272927A CA 2272927 C CA2272927 C CA 2272927C
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- Prior art keywords
- compound
- diseases
- disorders
- neuropeptide
- treating
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
- C07D295/08—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms
- C07D295/096—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly bound oxygen or sulfur atoms with the ring nitrogen atoms and the oxygen or sulfur atoms separated by carbocyclic rings or by carbon chains interrupted by carbocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Engineering & Computer Science (AREA)
- Obesity (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Biomedical Technology (AREA)
- Child & Adolescent Psychology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US3181596P | 1996-11-26 | 1996-11-26 | |
| US60/031,815 | 1996-11-26 | ||
| PCT/IB1997/001465 WO1998023603A1 (en) | 1996-11-26 | 1997-11-19 | Dimesylate salts of neuropeptide y ligands |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CA2272927A1 CA2272927A1 (en) | 1998-06-04 |
| CA2272927C true CA2272927C (en) | 2003-02-04 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002272927A Expired - Fee Related CA2272927C (en) | 1996-11-26 | 1997-11-19 | Dimesylate salts of neuropeptide y ligands |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US5914329A (enExample) |
| EP (1) | EP0944611B1 (enExample) |
| JP (1) | JP3120861B2 (enExample) |
| AP (1) | AP9701148A0 (enExample) |
| AR (1) | AR010304A1 (enExample) |
| AT (1) | ATE257472T1 (enExample) |
| AU (1) | AU4792497A (enExample) |
| BR (1) | BR9713538A (enExample) |
| CA (1) | CA2272927C (enExample) |
| DE (1) | DE69727155T2 (enExample) |
| DK (1) | DK0944611T3 (enExample) |
| ES (1) | ES2213207T3 (enExample) |
| GT (1) | GT199700123A (enExample) |
| HN (1) | HN1997000154A (enExample) |
| HR (1) | HRP970640A2 (enExample) |
| ID (1) | ID18964A (enExample) |
| MA (1) | MA26450A1 (enExample) |
| PA (1) | PA8441701A1 (enExample) |
| PE (1) | PE17099A1 (enExample) |
| PT (1) | PT944611E (enExample) |
| TN (1) | TNSN97191A1 (enExample) |
| WO (1) | WO1998023603A1 (enExample) |
| ZA (1) | ZA9710587B (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2001232900A1 (en) * | 2000-01-20 | 2001-07-31 | Michael Amling | Methods and compositions for control of bone formation via modulation of neuropeptide y activity |
| JP2005516001A (ja) | 2001-12-05 | 2005-06-02 | ベイラー カレッジ オブ メディスン | 交感神経活動状態の調節による骨形成の制御のための方法及び組成物 |
| NZ533848A (en) | 2002-01-09 | 2006-11-30 | Arexis Ab | Detection of mutations in the flavin-containing monooxygenase (FMO3) gene |
| EP1701722B1 (en) * | 2004-11-23 | 2009-10-14 | Dong Wha Pharmaceutical Co., Ltd. | N-hydroxy-4-{5-[4-(5-isopropyl-2-methyl-1,3-thiazol-4-yl)phenoxy¨]pentoxy}benzamidine 2 methansulfonic acid salt |
| EP1877076A4 (en) * | 2005-04-15 | 2012-02-01 | Regenertech Pty Ltd | USE OF NEUROPEPTIDES Y (NPY) AND AGONIST OF ANTAGONISTS THEREOF FOR REGENERATING TISSUES |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SK57097A3 (en) * | 1994-11-07 | 1998-10-07 | Pfizer | Certain substituted benzylamine derivatives; a new class of neuropeptide y1 specific ligands |
-
1997
- 1997-11-18 PA PA19978441701A patent/PA8441701A1/es unknown
- 1997-11-18 US US08/972,470 patent/US5914329A/en not_active Expired - Fee Related
- 1997-11-19 AU AU47924/97A patent/AU4792497A/en not_active Abandoned
- 1997-11-19 ES ES97910602T patent/ES2213207T3/es not_active Expired - Lifetime
- 1997-11-19 JP JP10524469A patent/JP3120861B2/ja not_active Expired - Fee Related
- 1997-11-19 AT AT97910602T patent/ATE257472T1/de not_active IP Right Cessation
- 1997-11-19 EP EP97910602A patent/EP0944611B1/en not_active Expired - Lifetime
- 1997-11-19 BR BR9713538A patent/BR9713538A/pt not_active Application Discontinuation
- 1997-11-19 DK DK97910602T patent/DK0944611T3/da active
- 1997-11-19 WO PCT/IB1997/001465 patent/WO1998023603A1/en not_active Ceased
- 1997-11-19 DE DE69727155T patent/DE69727155T2/de not_active Expired - Fee Related
- 1997-11-19 CA CA002272927A patent/CA2272927C/en not_active Expired - Fee Related
- 1997-11-19 PT PT97910602T patent/PT944611E/pt unknown
- 1997-11-19 PE PE1997001052A patent/PE17099A1/es not_active Application Discontinuation
- 1997-11-20 AP APAP/P/1997/001148A patent/AP9701148A0/en unknown
- 1997-11-24 AR ARP970105494A patent/AR010304A1/es unknown
- 1997-11-25 ZA ZA9710587A patent/ZA9710587B/xx unknown
- 1997-11-25 TN TNTNSN97191A patent/TNSN97191A1/fr unknown
- 1997-11-25 ID IDP973762A patent/ID18964A/id unknown
- 1997-11-25 MA MA24872A patent/MA26450A1/fr unknown
- 1997-11-25 GT GT199700123A patent/GT199700123A/es unknown
- 1997-11-26 HR HR60/031,815A patent/HRP970640A2/hr not_active Application Discontinuation
- 1997-11-26 HN HN1997000154A patent/HN1997000154A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| AP9701148A0 (en) | 1998-01-31 |
| ES2213207T3 (es) | 2004-08-16 |
| ATE257472T1 (de) | 2004-01-15 |
| AU4792497A (en) | 1998-06-22 |
| JP3120861B2 (ja) | 2000-12-25 |
| GT199700123A (es) | 1999-05-19 |
| JP2000505110A (ja) | 2000-04-25 |
| ID18964A (id) | 1998-05-28 |
| PA8441701A1 (es) | 2000-05-24 |
| CA2272927A1 (en) | 1998-06-04 |
| MA26450A1 (fr) | 2004-12-20 |
| DE69727155D1 (de) | 2004-02-12 |
| PE17099A1 (es) | 1999-02-19 |
| DK0944611T3 (da) | 2004-04-13 |
| TNSN97191A1 (fr) | 2005-03-15 |
| US5914329A (en) | 1999-06-22 |
| DE69727155T2 (de) | 2004-07-08 |
| HRP970640A2 (en) | 1998-10-31 |
| BR9713538A (enExample) | 2000-03-21 |
| HN1997000154A (es) | 1999-02-09 |
| ZA9710587B (en) | 1999-05-25 |
| AR010304A1 (es) | 2000-06-07 |
| PT944611E (pt) | 2004-04-30 |
| EP0944611B1 (en) | 2004-01-07 |
| WO1998023603A1 (en) | 1998-06-04 |
| EP0944611A1 (en) | 1999-09-29 |
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