CA2261887A1 - Conjugues lipidiques polaires covalents associes a des composes biologiquement actifs utilisables dans les onguents - Google Patents
Conjugues lipidiques polaires covalents associes a des composes biologiquement actifs utilisables dans les onguentsInfo
- Publication number
- CA2261887A1 CA2261887A1 CA002261887A CA2261887A CA2261887A1 CA 2261887 A1 CA2261887 A1 CA 2261887A1 CA 002261887 A CA002261887 A CA 002261887A CA 2261887 A CA2261887 A CA 2261887A CA 2261887 A1 CA2261887 A1 CA 2261887A1
- Authority
- CA
- Canada
- Prior art keywords
- salves
- drug
- drugs
- agents
- targeting
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/62—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being a protein, peptide or polyamino acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
- A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
- A61K47/54—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic compound
- A61K47/543—Lipids, e.g. triglycerides; Polyamines, e.g. spermine or spermidine
- A61K47/544—Phospholipids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Epidemiology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Dermatology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Biophysics (AREA)
- Organic Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/US1996/012124 WO1998003204A1 (fr) | 1996-07-23 | 1996-07-23 | Conjugues lipidiques polaires covalents associes a des composes biologiquement actifs utilisables dans les onguents |
Publications (2)
Publication Number | Publication Date |
---|---|
CA2261887A1 true CA2261887A1 (fr) | 1998-01-29 |
CA2261887C CA2261887C (fr) | 2007-10-02 |
Family
ID=22255500
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002261887A Expired - Fee Related CA2261887C (fr) | 1996-07-23 | 1996-07-23 | Conjugues lipidiques polaires covalents associes a des composes biologiquement actifs utilisables dans les onguents |
Country Status (5)
Country | Link |
---|---|
EP (1) | EP0917473A1 (fr) |
JP (1) | JPH11514009A (fr) |
AU (1) | AU724421B2 (fr) |
CA (1) | CA2261887C (fr) |
WO (1) | WO1998003204A1 (fr) |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2000033883A1 (fr) * | 1998-12-04 | 2000-06-15 | Oregon Health Sciences University | Conjugues lipides polaires covalents avec medicaments antimicrobiens et antineoplasiques destines a cibler des sites biologiques proteges |
US6464992B2 (en) * | 2000-04-14 | 2002-10-15 | University Of Kentucky Research Foundation | Topical micronutrient delivery system and uses thereof |
US7045543B2 (en) | 2001-11-05 | 2006-05-16 | Enzrel Inc. | Covalent conjugates of biologically-active compounds with amino acids and amino acid derivatives for targeting to physiologically-protected sites |
EA032840B8 (ru) * | 2011-06-22 | 2020-06-18 | Вайоми Терапеутикс Лимитед | Пролекарства на основе конъюгатов противогрибковых агентов и их применение |
WO2024083171A1 (fr) * | 2022-10-20 | 2024-04-25 | 苏州艾博生物科技有限公司 | Composé lipidique et composition de nanoparticules lipidiques |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5264618A (en) * | 1990-04-19 | 1993-11-23 | Vical, Inc. | Cationic lipids for intracellular delivery of biologically active molecules |
JPH05507929A (ja) * | 1990-06-15 | 1993-11-11 | ウェイク フォレスト ユニバーシティー | エーテル脂質―ヌクレオシド共有結合体 |
US5256641A (en) * | 1990-11-01 | 1993-10-26 | State Of Oregon | Covalent polar lipid-peptide conjugates for immunological targeting |
US5543390A (en) * | 1990-11-01 | 1996-08-06 | State Of Oregon, Acting By And Through The Oregon State Board Of Higher Education, Acting For And On Behalf Of The Oregon Health Sciences University | Covalent microparticle-drug conjugates for biological targeting |
US5149794A (en) * | 1990-11-01 | 1992-09-22 | State Of Oregon | Covalent lipid-drug conjugates for drug targeting |
-
1996
- 1996-07-23 CA CA002261887A patent/CA2261887C/fr not_active Expired - Fee Related
- 1996-07-23 JP JP10506883A patent/JPH11514009A/ja active Pending
- 1996-07-23 WO PCT/US1996/012124 patent/WO1998003204A1/fr not_active Application Discontinuation
- 1996-07-23 AU AU65945/96A patent/AU724421B2/en not_active Ceased
- 1996-07-23 EP EP96925431A patent/EP0917473A1/fr not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
JPH11514009A (ja) | 1999-11-30 |
WO1998003204A1 (fr) | 1998-01-29 |
AU6594596A (en) | 1998-02-10 |
EP0917473A1 (fr) | 1999-05-26 |
AU724421B2 (en) | 2000-09-21 |
CA2261887C (fr) | 2007-10-02 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
EEER | Examination request | ||
MKLA | Lapsed |