CA2210138A1 - Tocolytic oxytocin receptor antagonists - Google Patents
Tocolytic oxytocin receptor antagonistsInfo
- Publication number
- CA2210138A1 CA2210138A1 CA 2210138 CA2210138A CA2210138A1 CA 2210138 A1 CA2210138 A1 CA 2210138A1 CA 2210138 CA2210138 CA 2210138 CA 2210138 A CA2210138 A CA 2210138A CA 2210138 A1 CA2210138 A1 CA 2210138A1
- Authority
- CA
- Canada
- Prior art keywords
- alkyl
- compound
- hydrogen
- methyl
- piperidin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US37811395A | 1995-01-24 | 1995-01-24 | |
| US378,113 | 1995-01-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2210138A1 true CA2210138A1 (en) | 1996-08-01 |
Family
ID=23491770
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA 2210138 Abandoned CA2210138A1 (en) | 1995-01-24 | 1996-01-19 | Tocolytic oxytocin receptor antagonists |
Country Status (4)
| Country | Link |
|---|---|
| EP (1) | EP0805681A4 (de) |
| AU (1) | AU4763896A (de) |
| CA (1) | CA2210138A1 (de) |
| WO (1) | WO1996022775A1 (de) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2310660A (en) * | 1996-03-01 | 1997-09-03 | Merck & Co Inc | Benzoxazinone oxytocin receptor antagonists |
| GB2326410A (en) * | 1997-06-18 | 1998-12-23 | Merck & Co Inc | Tocolytic Oxytocin Receptor Antagonists |
| AU5620901A (en) | 2000-03-27 | 2001-10-08 | Applied Research Systems | Pharmaceutically active pyrrolidine derivatives as bax inhibitors |
| CA2423933A1 (en) | 2000-10-17 | 2002-04-25 | Applied Research Systems Ars Holding N.V. | Pharmaceutically active sulfanilide derivatives |
| EP1390347B1 (de) | 2001-03-20 | 2008-05-07 | Laboratoires Serono SA | Pyrrolidinesterderivate mit oxytocinmodulierender wirkung |
| US7109193B2 (en) | 2001-04-12 | 2006-09-19 | Wyeth | Tricyclic diazepines tocolytic oxytocin receptor antagonists |
| US6977254B2 (en) | 2001-04-12 | 2005-12-20 | Wyeth | Hydroxy cyclohexenyl phenyl carboxamides tocolytic oxytocin receptor antagonists |
| US6900200B2 (en) | 2001-04-12 | 2005-05-31 | Wyeth | Tricyclic hydroxy carboxamides and derivatives thereof tocolytic oxytocin receptor antagonists |
| US7326700B2 (en) | 2001-04-12 | 2008-02-05 | Wyeth | Cyclohexenyl phenyl carboxamides tocolytic oxytocin receptor antagonists |
| US7022699B2 (en) | 2001-04-12 | 2006-04-04 | Wyeth | Cyclohexenyl phenyl diazepines vasopressin and oxytocin receptor modulators |
| US7202239B2 (en) | 2001-04-12 | 2007-04-10 | Wyeth | Cyclohexylphenyl carboxamides tocolytic oxytocin receptor antagonists |
| US7064120B2 (en) | 2001-04-12 | 2006-06-20 | Wyeth | Tricyclic pyridyl carboxamides and derivatives thereof tocolytic oxytocin receptor antagonists |
| SK15552003A3 (sk) | 2001-06-18 | 2004-05-04 | Applied Research Systems Ars Holding N. V. | Oxadiazolové a tiadiazolové deriváty pyrolidínu, spôsob ich výroby, farmaceutický prostriedok s ich obsahom a ich použitie |
| CA2469042A1 (en) | 2001-12-20 | 2003-07-03 | Applied Research Systems Ars Holding N.V. | Triazoles as oxytocin antagonists |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3026534A1 (de) * | 1980-07-12 | 1982-03-18 | C.H. Boehringer Sohn, 6507 Ingelheim | 3,1-benzoxazin-2-one, ihre herstellung und verwendung |
| TW199153B (de) * | 1990-08-07 | 1993-02-01 | Dtsuka Seiyaku Kk | |
| AU657424B2 (en) * | 1992-07-02 | 1995-03-09 | Otsuka Pharmaceutical Co., Ltd. | Oxytocin antagonist |
| CA2166975C (en) * | 1993-07-16 | 2005-04-05 | Mark G. Bock | Benzoxazinone and benzopyrimidinone piperidinyl tocolytic oxytocin receptor antagonists |
| WO1997025992A1 (en) * | 1996-01-16 | 1997-07-24 | Merck & Co., Inc. | Tocolytic oxytocin receptor antagonists |
-
1996
- 1996-01-19 CA CA 2210138 patent/CA2210138A1/en not_active Abandoned
- 1996-01-19 WO PCT/US1996/000850 patent/WO1996022775A1/en not_active Application Discontinuation
- 1996-01-19 EP EP96903618A patent/EP0805681A4/de not_active Withdrawn
- 1996-01-19 AU AU47638/96A patent/AU4763896A/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| EP0805681A1 (de) | 1997-11-12 |
| WO1996022775A1 (en) | 1996-08-01 |
| AU4763896A (en) | 1996-08-14 |
| EP0805681A4 (de) | 1998-05-06 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| AU691829B2 (en) | Benzoxazinone and benzopyrimidinone piperidinyl tocolytic oxytocin receptor antagonists | |
| US5204349A (en) | Amide-substituted derivatives of spiroindanylcamphorsulfonyl oxytocin antagonists | |
| US5756504A (en) | Tocolytic oxytocin receptor antagonists | |
| EP0533243B1 (de) | Hydantoin und Succinimid-substituierte Spiroindanylcamphorsulfonyl als Oxytocin-Antagonisten | |
| US5756497A (en) | Tocolytic oxytocin receptor antagonists | |
| CA2210138A1 (en) | Tocolytic oxytocin receptor antagonists | |
| CA2055024A1 (en) | N-phenyl piperidinylcamphorsulfonyl oxytocin antagonists | |
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| JP2004503547A (ja) | セリンプロテアーゼインヒビター | |
| JPH082870B2 (ja) | ピペラジニルカンファースルフォニルオキシトシン拮抗物質の置換誘導体 | |
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| AU2005202357A1 (en) | Piperazine derivatives useful as CCR5 antagonists | |
| CA2174650A1 (en) | Piperidinyl camphorsulfonyl oxytocin antagonists | |
| WO1997025992A1 (en) | Tocolytic oxytocin receptor antagonists | |
| JP2004503532A (ja) | セリンプロテアーゼインヒビター | |
| GB2326639A (en) | Piperazine Oxytocin Receptor Antagonists | |
| JPH09500133A (ja) | オキシトシンのアンタゴニストである置換ピペラジニル樟脳誘導体 | |
| GB2326410A (en) | Tocolytic Oxytocin Receptor Antagonists | |
| GB2310660A (en) | Benzoxazinone oxytocin receptor antagonists | |
| TW201720814A (zh) | 用於局部藥物遞送之非類固醇糖皮質激素受體調節劑 | |
| JPH05213865A (ja) | ピペラジニルカンファースルフォニルオキシトシン拮抗物質の置換アルキル誘導体 | |
| US6090805A (en) | Tocolytic oxytocin receptor antagonists | |
| CA2151821A1 (en) | Hydantoin and succinimide-substituted derivatives of spiroindanylcamphorsulfonyl oxytocin antagonists | |
| JP2004083511A (ja) | アクリルアミド誘導体 |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FZDE | Dead |