CA2091057A1 - Derives de substitution de 6,7-dihydroimidazo[1,5,4-ef]-1,5-benzodiazepin-6-ones; methode de preparation; compositions pharmaceutiques - Google Patents

Derives de substitution de 6,7-dihydroimidazo[1,5,4-ef]-1,5-benzodiazepin-6-ones; methode de preparation; compositions pharmaceutiques

Info

Publication number
CA2091057A1
CA2091057A1 CA002091057A CA2091057A CA2091057A1 CA 2091057 A1 CA2091057 A1 CA 2091057A1 CA 002091057 A CA002091057 A CA 002091057A CA 2091057 A CA2091057 A CA 2091057A CA 2091057 A1 CA2091057 A1 CA 2091057A1
Authority
CA
Canada
Prior art keywords
alkyl
formula
integer
paf
substituted
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002091057A
Other languages
English (en)
Inventor
John Steele
Kelvin Cooper
Michael J. Fray
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Ltd
Pfizer Inc
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2091057A1 publication Critical patent/CA2091057A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CA002091057A 1990-09-05 1991-09-02 Derives de substitution de 6,7-dihydroimidazo[1,5,4-ef]-1,5-benzodiazepin-6-ones; methode de preparation; compositions pharmaceutiques Abandoned CA2091057A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB9019409.3 1990-09-05
GB909019409A GB9019409D0 (en) 1990-09-05 1990-09-05 Therapeutic agents

Publications (1)

Publication Number Publication Date
CA2091057A1 true CA2091057A1 (fr) 1992-03-06

Family

ID=10681724

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002091057A Abandoned CA2091057A1 (fr) 1990-09-05 1991-09-02 Derives de substitution de 6,7-dihydroimidazo[1,5,4-ef]-1,5-benzodiazepin-6-ones; methode de preparation; compositions pharmaceutiques

Country Status (8)

Country Link
EP (1) EP0548125A1 (fr)
JP (1) JPH06500091A (fr)
CA (1) CA2091057A1 (fr)
FI (1) FI930967A0 (fr)
GB (1) GB9019409D0 (fr)
IE (1) IE913102A1 (fr)
PT (1) PT98851A (fr)
WO (1) WO1992004354A1 (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5879892A (en) * 1997-04-25 1999-03-09 Ludwig Institute For Cancer Research Leukemia associated genes
US6291430B1 (en) 1997-09-12 2001-09-18 Ludwig Institute For Cancer Research Mage-3 peptides presented by HLA class II molecules
US5965535A (en) * 1997-09-12 1999-10-12 Ludwig Institute For Cancer Research Mage-3 peptides presented by HLA class II molecules

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MY104933A (en) * 1987-09-30 1994-07-30 Pfizer Ltd Platelet activating factor antagonists
DK0389189T3 (da) * 1989-03-23 1994-06-20 Pfizer Diazepin antiallergimidler

Also Published As

Publication number Publication date
PT98851A (pt) 1992-07-31
WO1992004354A1 (fr) 1992-03-19
FI930967A (fi) 1993-03-04
JPH06500091A (ja) 1994-01-06
IE913102A1 (en) 1992-03-11
FI930967A0 (fi) 1993-03-04
EP0548125A1 (fr) 1993-06-30
GB9019409D0 (en) 1990-10-17

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Legal Events

Date Code Title Description
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FZDE Dead