CA2045494A1 - Reduced irreversible bombesin antagonists - Google Patents
Reduced irreversible bombesin antagonistsInfo
- Publication number
- CA2045494A1 CA2045494A1 CA002045494A CA2045494A CA2045494A1 CA 2045494 A1 CA2045494 A1 CA 2045494A1 CA 002045494 A CA002045494 A CA 002045494A CA 2045494 A CA2045494 A CA 2045494A CA 2045494 A1 CA2045494 A1 CA 2045494A1
- Authority
- CA
- Canada
- Prior art keywords
- leu
- residue
- gly
- peptide
- group
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/02—Linear peptides containing at least one abnormal peptide link
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/08—Linear peptides containing only normal peptide links having 12 to 20 amino acids
- C07K7/086—Bombesin; Related peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Genetics & Genomics (AREA)
- Biochemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Saccharide Compounds (AREA)
- Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB898925024A GB8925024D0 (en) | 1989-11-06 | 1989-11-06 | Reduced irreversible bombesin antagonists |
GB8925024.5 | 1989-11-06 | ||
GB9006413.0 | 1990-03-22 | ||
GB909006413A GB9006413D0 (en) | 1990-03-22 | 1990-03-22 | Reduced irreversible bombesin antagonists |
Publications (1)
Publication Number | Publication Date |
---|---|
CA2045494A1 true CA2045494A1 (en) | 1991-05-07 |
Family
ID=26296160
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002045494A Abandoned CA2045494A1 (en) | 1989-11-06 | 1990-11-02 | Reduced irreversible bombesin antagonists |
Country Status (9)
Country | Link |
---|---|
EP (1) | EP0452447A1 (ja) |
JP (1) | JPH04502629A (ja) |
KR (1) | KR920701242A (ja) |
AU (1) | AU6610390A (ja) |
CA (1) | CA2045494A1 (ja) |
HU (1) | HUT58763A (ja) |
IE (1) | IE903958A1 (ja) |
IL (1) | IL96216A0 (ja) |
WO (1) | WO1991006563A1 (ja) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US9839703B2 (en) | 2012-09-25 | 2017-12-12 | Advanced Accelerator Applications Usa, Inc. | Radiolabeled GRPR-antagonists for diagnostic imaging and treatment of GRPR-positive cancer |
Families Citing this family (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5834433A (en) * | 1990-07-26 | 1998-11-10 | Merrell Pharmaceuticals Inc. | Compounds and pharmaceutical uses of peptides of bombesin and GRP |
ES2106188T3 (es) * | 1991-05-23 | 1997-11-01 | Merrell Pharma Inc | Analogos de bombesina. |
WO1993016105A1 (en) * | 1992-02-07 | 1993-08-19 | Merrell Dow Pharmaceuticals Inc. | Phenylalanine analogs of bombesin |
WO2004093807A2 (en) | 2003-04-22 | 2004-11-04 | Societe De Conseils De Recherches Et D'applications Scientifiques S.A.S. | Somatostatin vectors |
EP2848628A1 (en) * | 2010-01-25 | 2015-03-18 | Cornell University | Aromatic-cationic peptides and uses of same |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2795449B2 (ja) * | 1987-09-24 | 1998-09-10 | ジ・アドミニストレーターズ・オブ・ザ・ツーレイン・エデュケイショナル・ファンド | 治療用ペプチド |
GB8808768D0 (en) * | 1988-04-14 | 1988-05-18 | Erba Carlo Spa | Peptide ligands for bombesin receptors |
GR1000608B (el) * | 1988-07-21 | 1992-08-31 | Erba Carlo Spa | Μεθοδος για την παρασκευη ανταγωνιστων bombesin. |
MC2144A1 (fr) * | 1988-10-14 | 1992-02-19 | Univ Tulane | Peptides therapeutiques |
-
1990
- 1990-11-02 AU AU66103/90A patent/AU6610390A/en not_active Abandoned
- 1990-11-02 HU HU912604A patent/HUT58763A/hu unknown
- 1990-11-02 EP EP90915774A patent/EP0452447A1/en not_active Ceased
- 1990-11-02 IL IL96216A patent/IL96216A0/xx unknown
- 1990-11-02 WO PCT/EP1990/001836 patent/WO1991006563A1/en not_active Application Discontinuation
- 1990-11-02 KR KR1019910700701A patent/KR920701242A/ko not_active Application Discontinuation
- 1990-11-02 IE IE395890A patent/IE903958A1/en unknown
- 1990-11-02 JP JP2514747A patent/JPH04502629A/ja active Pending
- 1990-11-02 CA CA002045494A patent/CA2045494A1/en not_active Abandoned
Cited By (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US9839703B2 (en) | 2012-09-25 | 2017-12-12 | Advanced Accelerator Applications Usa, Inc. | Radiolabeled GRPR-antagonists for diagnostic imaging and treatment of GRPR-positive cancer |
US11083805B2 (en) | 2012-09-25 | 2021-08-10 | Advanced Accelerator Applications International Sa | Radiolabeled GRPR-antagonists for diagnostic imaging and treatment of GRPR-positive cancer |
US12064489B2 (en) | 2012-09-25 | 2024-08-20 | Advanced Accelerator Applications International Sa | Radiolabeled GRPR-antagonists for diagnostic imaging and treatment of GRPR-positive cancer |
US12064491B2 (en) | 2012-09-25 | 2024-08-20 | Advanced Accelerator Applications International Sa | Radiolabeled GRPR-antagonists for diagnostic imaging and treatment of GRPR-positive cancer |
US12064490B2 (en) | 2012-09-25 | 2024-08-20 | Advanced Accelerator Applications International Sa | Radiolabeled GRPR-Antagonists for Diagnostic Imaging and Treatment of GRPR-Positive Cancer |
Also Published As
Publication number | Publication date |
---|---|
WO1991006563A1 (en) | 1991-05-16 |
JPH04502629A (ja) | 1992-05-14 |
AU6610390A (en) | 1991-05-31 |
IE903958A1 (en) | 1991-05-08 |
IL96216A0 (en) | 1991-08-16 |
HUT58763A (en) | 1992-03-30 |
EP0452447A1 (en) | 1991-10-23 |
KR920701242A (ko) | 1992-08-11 |
HU912604D0 (en) | 1992-01-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FZDE | Discontinued |