CA1302422C - 5-aminoethyloxazolidin-2-one derivatives, process for the preparation thereofand their therapeutic use - Google Patents

5-aminoethyloxazolidin-2-one derivatives, process for the preparation thereofand their therapeutic use

Info

Publication number
CA1302422C
CA1302422C CA000546004A CA546004A CA1302422C CA 1302422 C CA1302422 C CA 1302422C CA 000546004 A CA000546004 A CA 000546004A CA 546004 A CA546004 A CA 546004A CA 1302422 C CA1302422 C CA 1302422C
Authority
CA
Canada
Prior art keywords
formula
stereoisomers
group
hydrogen atom
mixture
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
CA000546004A
Other languages
English (en)
French (fr)
Inventor
Margherita Strolin-Benedetti
Patrice Renaut
Michel Langlois
Philippe Dostert
Alain-Rene Schoofs
Jean-Francois Rumigny
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Synthelabo SA
Original Assignee
Delalande SA
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR8612369A external-priority patent/FR2603279B1/fr
Priority claimed from FR8618368A external-priority patent/FR2609029B1/fr
Application filed by Delalande SA filed Critical Delalande SA
Application granted granted Critical
Publication of CA1302422C publication Critical patent/CA1302422C/en
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18—Oxygen atoms
    • C07D263/20—Oxygen atoms attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA000546004A 1986-09-03 1987-09-02 5-aminoethyloxazolidin-2-one derivatives, process for the preparation thereofand their therapeutic use Expired - Lifetime CA1302422C (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
FR8612369 1986-09-03
FR8612369A FR2603279B1 (fr) 1986-09-03 1986-09-03 Benzyloxy-phenyl-oxazolidinones, procede de preparation et utilisation en therapeutique
FR8618368A FR2609029B1 (fr) 1986-12-30 1986-12-30 Derives 5-aminoethyles de l'oxazolidinone-2, leur procede de preparation et leur application en therapeutique
FR8618368 1986-12-30

Publications (1)

Publication Number Publication Date
CA1302422C true CA1302422C (en) 1992-06-02

Family

ID=26225458

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000546004A Expired - Lifetime CA1302422C (en) 1986-09-03 1987-09-02 5-aminoethyloxazolidin-2-one derivatives, process for the preparation thereofand their therapeutic use

Country Status (7)

Country Link
US (1) US4897409A (enExample)
EP (1) EP0259228B1 (enExample)
AU (1) AU7778087A (enExample)
CA (1) CA1302422C (enExample)
DE (1) DE3779525T2 (enExample)
ES (1) ES2031921T3 (enExample)
GR (1) GR3005082T3 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA1302422C (en) * 1986-09-03 1992-06-02 Margherita Strolin-Benedetti 5-aminoethyloxazolidin-2-one derivatives, process for the preparation thereofand their therapeutic use
US5380778A (en) * 1992-09-30 1995-01-10 Minnesota Mining And Manufacturing Company Fluorochemical aminoalcohols
US6083967A (en) * 1997-12-05 2000-07-04 Pharmacia & Upjohn Company S-oxide and S,S-dioxide tetrahydrothiopyran phenyloxazolidinones

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2428032A1 (fr) * 1978-06-09 1980-01-04 Delalande Sa Nouvelles oxazolidimones, oxazolidinethiones et pyrrolidinones, leur procede de preparation et leur application en therapeutique
US4348393A (en) * 1978-06-09 1982-09-07 Delalande S.A. N-Aryl oxazolidinones, oxazolidinethiones, pyrrolidinones, pyrrolidines and thiazolidinones
CA1171865A (en) * 1980-06-04 1984-07-31 Alain Lacour N-aryl azolone derivatives, the process for preparing the same and their application in therapeutics
FR2500450A1 (fr) * 1981-02-25 1982-08-27 Delalande Sa Nouveaux derives aminomethyl-5 oxazolidiniques, leur procede de preparation et leur application en therapeutique
FR2528046B1 (fr) * 1982-06-08 1985-06-21 Delalande Sa Derives de l'oxazolidinone-2 n-arylee optiquement actifs, inhibiteurs specifiques et reversibles de la monoamine oxydase de type b et leur procede de preparation
CA1302422C (en) * 1986-09-03 1992-06-02 Margherita Strolin-Benedetti 5-aminoethyloxazolidin-2-one derivatives, process for the preparation thereofand their therapeutic use

Also Published As

Publication number Publication date
DE3779525D1 (de) 1992-07-09
EP0259228B1 (fr) 1992-06-03
ES2031921T3 (es) 1993-01-01
AU7778087A (en) 1988-04-14
US4897409A (en) 1990-01-30
GR3005082T3 (enExample) 1993-05-24
DE3779525T2 (de) 1993-02-11
EP0259228A1 (fr) 1988-03-09

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