CA1256430A - Benzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same - Google Patents

Benzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same

Info

Publication number
CA1256430A
CA1256430A CA000500970A CA500970A CA1256430A CA 1256430 A CA1256430 A CA 1256430A CA 000500970 A CA000500970 A CA 000500970A CA 500970 A CA500970 A CA 500970A CA 1256430 A CA1256430 A CA 1256430A
Authority
CA
Canada
Prior art keywords
group
formula
carbon atoms
hydrogen atom
group represented
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA000500970A
Other languages
English (en)
French (fr)
Inventor
Takehiko Yamane
Takuji Hashizume
Katsuji Yamashita
Kiyoshi Watanabe
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Kanegafuchi Chemical Industry Co Ltd
Original Assignee
Kanegafuchi Chemical Industry Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kanegafuchi Chemical Industry Co Ltd filed Critical Kanegafuchi Chemical Industry Co Ltd
Application granted granted Critical
Publication of CA1256430A publication Critical patent/CA1256430A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA000500970A 1985-02-05 1986-02-03 Benzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same Expired CA1256430A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2038485 1985-02-05
JP20384/1985 1985-02-05

Publications (1)

Publication Number Publication Date
CA1256430A true CA1256430A (en) 1989-06-27

Family

ID=12025537

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000500970A Expired CA1256430A (en) 1985-02-05 1986-02-03 Benzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same

Country Status (4)

Country Link
EP (1) EP0190709B1 (https=)
JP (1) JPS63183587A (https=)
CA (1) CA1256430A (https=)
DE (1) DE3667286D1 (https=)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2544375B2 (ja) * 1986-07-14 1996-10-16 鐘淵化学工業株式会社 アルキル置換ベンゾキサジノリフアマイシン誘導体
DE68924722T2 (de) * 1988-03-18 1996-04-18 Kanegafuchi Chemical Ind Substituiertes Benzoxazinorifamycinderivat, Verfahren zur Herstellung und dieses Derivat enthaltende Bakterizidmittel.
CA1304363C (en) * 1988-11-01 1992-06-30 Takehiko Yamane 3'-hydroxybenzoxazinorifamycin derivative, process for preparing the same and antibacterial agent containing the same
JP2620399B2 (ja) * 1990-08-20 1997-06-11 鐘淵化学工業株式会社 ３′―アルキルまたはアリールシリルオキシベンゾキサジノリファマイシン誘導体
US5981522A (en) * 1995-09-01 1999-11-09 Kaneka Corporation Treatment of disease caused by infection of Helicobacter
KR100407849B1 (ko) * 1995-09-01 2004-05-07 가네가후치 가가쿠고교 가부시키가이샤 헬리코박터의감염에기인하는질환의치료제
JP3963976B2 (ja) 1995-12-08 2007-08-22 株式会社カネカ クラミジア感染症治療剤
EP0861660B9 (en) * 1997-02-28 2006-06-28 Kaneka Corporation Curative medicine for disease caused by infection of Helicobacter
WO1999006047A1 (en) * 1997-07-29 1999-02-11 Kaneka Corporation Use of rifamycin derivative for treating mastitis in a domestic animal
US6486161B1 (en) 1998-07-29 2002-11-26 Kaneka Corporation Use of rifamycin derivative for treating mastitis in a domestic animal
CA2536378A1 (en) * 2003-08-22 2005-03-10 Activbiotics, Inc. Rifamycin analogs and uses thereof
US7256187B2 (en) 2004-03-10 2007-08-14 Cumbre Pharmaceuticals Inc. Rifamycin C-11 oxime derivatives effective against drug-resistant microbes
US7265107B2 (en) 2004-03-10 2007-09-04 Cumbre Pharmaceuticals Inc. Rifamycin C-11 oxime cyclo derivatives effective against drug-resistant microbes
BR112018014355A2 (pt) 2016-03-04 2018-12-18 Genentech, Inc. processos para a preparação de f-benzoxazinorifamicina i e para a preparação de 2-amino-5-fluorobenzeno-1,3-diol iii

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL130099C (https=) * 1963-10-11

Also Published As

Publication number Publication date
EP0190709A1 (en) 1986-08-13
DE3667286D1 (de) 1990-01-11
EP0190709B1 (en) 1989-12-06
JPH0557275B2 (https=) 1993-08-23
JPS63183587A (ja) 1988-07-28

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Legal Events

Date Code Title Description
MKEX Expiry
MKEX Expiry

Effective date: 20060627