CA1161036A - Composes de quinazoline-dione, procede de production et applications en pharmacie - Google Patents

Composes de quinazoline-dione, procede de production et applications en pharmacie

Info

Publication number
CA1161036A
CA1161036A CA000377591A CA377591A CA1161036A CA 1161036 A CA1161036 A CA 1161036A CA 000377591 A CA000377591 A CA 000377591A CA 377591 A CA377591 A CA 377591A CA 1161036 A CA1161036 A CA 1161036A
Authority
CA
Canada
Prior art keywords
ethoxycarbonyl
dimethyl
phenyl
compound
group
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA000377591A
Other languages
English (en)
Inventor
Masayuki Ishikawa
Fujinori Sasaki
Yukuo Eguchi
Soyao Moriguchi
Hisashi Ebisawa
Akiko Sugimoto
Katsuhiko Gotoh
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Individual
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP6332880A external-priority patent/JPS56161375A/ja
Priority claimed from JP6708580A external-priority patent/JPS56164172A/ja
Priority claimed from JP8084380A external-priority patent/JPS577471A/ja
Priority claimed from JP8771580A external-priority patent/JPS5714580A/ja
Priority claimed from JP10239680A external-priority patent/JPS5728067A/ja
Priority claimed from JP10239780A external-priority patent/JPS5728068A/ja
Priority claimed from JP10674880A external-priority patent/JPS5731670A/ja
Priority claimed from JP10921280A external-priority patent/JPS5735573A/ja
Application filed by Individual filed Critical Individual
Application granted granted Critical
Publication of CA1161036A publication Critical patent/CA1161036A/fr
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/95—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in positions 2 and 4
    • C07D239/96—Two oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
CA000377591A 1980-05-15 1981-05-14 Composes de quinazoline-dione, procede de production et applications en pharmacie Expired CA1161036A (fr)

Applications Claiming Priority (16)

Application Number Priority Date Filing Date Title
JP63,328/80 1980-05-15
JP6332880A JPS56161375A (en) 1980-05-15 1980-05-15 2,4 1h, 3h -quinazolinedione derivative
JP6708580A JPS56164172A (en) 1980-05-22 1980-05-22 Novel 2,4 1h,3h -quinazolinedione derivative
JP67,085/80 1980-05-22
JP80,843/80 1980-06-17
JP8084380A JPS577471A (en) 1980-06-17 1980-06-17 Novel 2,4 1h,3h -quinazolinedione derivative
JP8771580A JPS5714580A (en) 1980-06-30 1980-06-30 Novel 2,4 1h, 3h -quinazolinedione derivative
JP87,715/80 1980-06-30
JP102,396/80 1980-07-28
JP10239680A JPS5728067A (en) 1980-07-28 1980-07-28 2,4 1h,3h -quinazolinedione derivative
JP102,397/80 1980-07-28
JP10239780A JPS5728068A (en) 1980-07-28 1980-07-28 Novel 2,4 1h,3h -quinazolinedione derivative
JP106,748/80 1980-08-05
JP10674880A JPS5731670A (en) 1980-08-05 1980-08-05 Novel 2,4 1h, 3h -quinazolinedione derivative
JP109,212/80 1980-08-11
JP10921280A JPS5735573A (en) 1980-08-11 1980-08-11 Novel 3-alkyl substituted 2,4(1h,3h)-quinazolinedione derivative

Publications (1)

Publication Number Publication Date
CA1161036A true CA1161036A (fr) 1984-01-24

Family

ID=27572548

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000377591A Expired CA1161036A (fr) 1980-05-15 1981-05-14 Composes de quinazoline-dione, procede de production et applications en pharmacie

Country Status (2)

Country Link
US (1) US4405623A (fr)
CA (1) CA1161036A (fr)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS608274A (ja) * 1983-06-27 1985-01-17 Fujisawa Pharmaceut Co Ltd 新規キナゾリノン誘導体およびその製造法・並びに抗アレルギ−剤
GB8524663D0 (en) * 1985-10-07 1985-11-13 Fujisawa Pharmaceutical Co Quinazoline derivatives
JP2621460B2 (ja) * 1988-02-29 1997-06-18 藤沢薬品工業株式会社 利尿または降圧剤
DE4339209A1 (de) * 1993-11-17 1995-05-18 Hoechst Ag Verfahren zur Herstellung von substituierten Chinazolin-2,4-dionen
DE4429978A1 (de) * 1994-08-24 1996-02-29 Bayer Ag Verfahren zur Herstellung von Chinazolin-2,4-dionen
DE4441145A1 (de) * 1994-11-18 1996-05-23 Hoechst Ag Verfahren zur Herstellung von substituierten Chinazolin-2,4-dionen
EP0742213A1 (fr) * 1995-05-10 1996-11-13 Hoechst Aktiengesellschaft Procédé de préparation de 3-aryl-quinazolines-2,4-diones substitués
DE19517036A1 (de) * 1995-05-10 1996-11-14 Hoechst Ag Verfahren zur Herstellung von substituierten 3-Arylchinazolin-2,4-dionen
DE19517035A1 (de) * 1995-05-10 1996-11-14 Hoechst Ag Verfahren zur Herstellung von substituierten 3-Arylchinazolin-2,4-dionen
US5780628A (en) * 1996-02-01 1998-07-14 Sumitomo Chemical Company, Limited Process for producing dioxoquinazolines
WO2012087938A1 (fr) * 2010-12-20 2012-06-28 Glaxosmithkline Llc Dérivés de quinazolinone en tant qu'agents antiviraux
WO2012125521A1 (fr) * 2011-03-14 2012-09-20 Eternity Bioscience Inc. Quinazolinediones et leur utilisation
TWI527800B (zh) 2011-04-01 2016-04-01 南京英派藥業有限公司 作為聚（二磷酸腺苷酸－核醣）聚合酶（ｐａｒｐ）之抑制劑之１－（芳基甲基）喹唑啉－２，４（１ｈ，３ｈ）－二酮及其應用
WO2023158845A1 (fr) * 2022-02-18 2023-08-24 Musc Foundation For Researchdevelopment Petites molécules ciblant la poche de liaison au nadh vdac pour moduler le métabolisme du cancer

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BE788807A (fr) * 1971-09-15 1973-03-14 Inst Francais Du Petrole Composes dicarboxyliques a noyaux quinazoline-dione-2,4 et resines polyesters en derivant
NZ192392A (en) * 1978-12-19 1983-02-15 M Ishikawa 3-(substituted (phenyl or pyridyl)) -3,4-dihydroquinazolin-4-ones

Also Published As

Publication number Publication date
US4405623A (en) 1983-09-20

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